Session Details
[26P-pm]反応②／分子認識／反応機構／構造と物性・その他
Thu. Mar 26, 2020 2:00 PM - 4:30 PM JST
Thu. Mar 26, 2020 5:00 AM - 7:30 AM UTC
Thu. Mar 26, 2020 5:00 AM - 7:30 AM UTC
[Room P] Event Hall 1F
[26P-pm001S]One-pot thermal [2+2] cycloaddition of o-silylalkynyl-O-allenylphenol followed by nucleophilic addition of water for the synthesis of arylcyclobutenals
○Ramon Francisco Bernardino Avena1, Shouhei Ohno1, Hiroshi Aoyama1, Hiromichi Fujioka1, Mitsuhiro Arisawa1 (1. Grad. Sch. Pharm. Sci., Osaka Univ.)
[26P-pm002]Development of perfluoroalkylation reactions by using perfluoro acid anhydrides
○Shintaro Kawamura1,2, Valverde Elena2, Daisuke Sekine2, Mikiko Sodeoka1,2 (1. CSRS, RIKEN, 2. CPR, RIKEN)
[26P-pm003]New boroprolinamide organocatalyst for the asymmetric aldol reaction
○Zubeda Begum1, Chigusa Seki1, Yuko Okuyama2, Koji Uwai1, Hiroto Nakano1 (1. Grad. Sch. Eng., Muroran Inst. Tech., 2. Tohoku Med. Pharm. Univ.)
[26P-pm004]Rapid Synthesis of 3,4-Fused Tricyclic Indoles based on C-H Activation using Rhodium-Carbene Species
Mai Yanagawa1, ○Shingo Harada1, Tetsuhiro Nemoto1 (1. Grad. Sch. Pharm. Sci., Chiba Univ.)
[26P-pm005S]Amine/thiol-induced asymmetric Aldol/2,3-sigmatropic rearrangement of optically active sulfoxide
○Misa Kasai1, Motofumi Miura1, Masaharu Toriyama1, Shigeyasu Motohashi1 (1. Sch. of Pharm., Nihon Univ.)
[26P-pm006S]Study on the reaction condition to the Late-Stage C-H Functionalization against β2 stimulator
○Mayuko Seki1, Motofumi Miura1, Masaharu Toriyama1, Shigeyasu Motohashi1 (1. Sch. of Pharm., Nihon Univ.)
[26P-pm007S]Development of the efficient synthesis of skeletal Flavanones
○Sayumi Nakayama1, Toshinori Nakakita2, Motofumi Miura1, Masaharu Toriyama1, Shigeyasu Motohashi1 (1. Sch. of Pharm., Nihon Univ., 2. Yokohama Univ. of Pharm.)
[26P-pm009]Synthesis of Functionalized Monoaryl Iodanes by ipso-Substitution Reactions
○Tatsuhiko Yoshino1, Keitaro Matsuoka1, Narumi Komami1, Ayako Nakano1, Yukino Okabe1, Masahiro Kojima1, Shigeki Matsunaga1 (1. Fac. Pharm. Sci., Hokkaido Univ.)
[26P-pm010S]Synthesis of cyclic carbamates via TM-HAT/RPC mechanism
Takuya Nagai1, Yoshihiro Terada1, Nao Mimata1, ○Chikayoshi Sebe1, Kou Hiroya1, Hiroki Shigehisa1 (1. Pharm. Sci., Musashino Univ.)
[26P-pm011S]Synthesis of cyclic ureas and isoureas via TM-HAT/RPC mechanism
○Nao Mimata1, Takuya Nagai1, Yoshihiro Terada1, Kou Hiroya1, Hiroki Shigehisa1 (1. Pharm. Sci., Musashino Univ.)
[26P-pm012]Synthesis of transposed analogues of CJ-14877, a potent production inhibitor of interleukin-1β Part Ⅱ
○Natsumi Yagyu1, Yuna Tsuji1, Eri Nagata1, Yukina Omura1, Nozomi Kitazawa1, Yosiyuki Adachi2, Naohito Ohno2, Reiko Yano1, Yukio Hitotsuyanagi2, Koichi Takeya2, Yutaka Aoyagi1 (1. College of Pharmacy, Kinjo Gakuin University, 2. School of Pharmacy, Tokyo University of Pharmacy and Life Sciences)
[26P-pm013]Lipase TL-mediated kinetic resolution of anisoin Part Ⅱ
○Nami Katagiri1, Rina Shikano1, Reiko Yano1, Yukio Hitotsuyanagi2, Yutaka Aoyagi1, Robert M. Williams3 (1. College of Pharmacy, Kinjo Gakuin University, 2. School of Pharmacy, Tokyo University of Pharmacy and Life Sciences, 3. Department of Chemistry, Colorado State University)
[26P-pm014S]Synthesis of oxidative metabolites of fucoxanthin and their anti-inflammatory effects
○Yuzuru Okada1, Takashi Okitsu1, Akimori Wada1, Naoki Takatani2, Masashi Hosokawa2, Yumiko Yamano1 (1. Kobe Pharm. Univ., 2. Grad. Sch. Fisheries Hokkaido Univ.)
[26P-pm015S]Intramolecular Diels-Alder Reaction of Methoxynaphthalenes and Alkynes
Takashi Okitsu1, ○Kanta Taniguchi1, Hinata Ishii1, Fumitaka Matano1, Akimori Wada1 (1. Kobe Pharm. Univ.)
[26P-pm016S]Domino Reaction of Epoxy-ynamides Leading to Tricyclic Scaffolds
Takashi Okitsu1, ○Kenshi Sakuragi1, Genki Fukui1, Akimori Wada1 (1. Kobe Pharm. Univ.)
[26P-pm017S]Tandem Dehydration-Electrophilic Cyclization Reaction of Silylalkynols
Takashi Okitsu1, ○Mai Morohashi1, Honoka Niwa1, Akimori Wada1 (1. Kobe Pharm. Univ.)
[26P-pm018]Palladium Catalyzed Cyclization-Carbonylation-Cyclization Hetero Coupling Reaction of Alkynes
○Keisuke Kato1, Tomoyuki Mochida2, Taichi Kusakabe1, Keisuke Takahashi1 (1. Pharm. Sci., Toho Univ., 2. Dept. Chem., Kobe Univ.)
[26P-pm019]Palladium catalyzed synthesis of 4,4’-bipyrazoles
○Taichi Kusakabe1, Keisuke Takahashi1, Keisuke Kato1 (1. Faculty of Pharmaceutical Sciences, Toho University)
[26P-pm020S]Synthesis and evaluation of C2-symmetric planar chiral multiple hydrogen-bond donor catalysts
Keisuke Yoshida1, ○chihiro hayakawa1, Hiromu Motoyama1, Takatoshi Matsumoto2, Shinji Kitagaki1 (1. Faculty of Pharmacy, Meijo University, 2. Institute of Multidisciplinary Research for Advanced Materials, Tohoku University)
[26P-pm021S]Total synthesis of Misrametine
Keisuke Yoshida1, Arisa Hidaka1, ○Yuri Imaizumi1, Yuri Fukami1, Shinji Kitagaki1 (1. Faculty of Pharmacy, Meijo University)
[26P-pm022S]Development of N-N coupling reaction of tricyclic biarylamine by using NaOCl・5H2O
Keisuke Yoshida1, Takato Nakayama1, ○Taihei Yamada1, Rina Sako1, Chihiro Ito1, Shinzi Kitagaki1 (1. Faculty of Pharmacy, Meijo University)
[26P-pm023S]Construction of contiguous chiral stereocenter by using bifunctional thiourea catalyst
Keisuke Yoshida1, Syoko Hotokezaka1, ○Koichi Sugito1, Shinji Kitagaki1 (1. Faculty of Pharmacy, Meijo University)
[26P-pm024]Platinum(II)-catalyzed dehydrative C3-benzylation of electron-deficient indoles with benzyl alcohols.
○Hidemasa Hikawa1, Yuuki Matsuura1, Shoko Kikkawa1, Isao Azumaya1 (1. Fac.Pharm.Sci., Toho Univ.)
[26P-pm025S]Palladium-catalyzed dehydrative S-benzylation of thiosalicylic acids in heptane
○Katsuyuki Taoka1, Taku Nakayama1, Hidemasa Hikawa1, Shoko Kikkawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)
[26P-pm026S]Gold(III)/TPPMS-catalyzed dehydrative allylation of anthranilic acids in water
○Ayumi Yamaguchi1, Hidemasa Hikawa1, Shoko Kikkawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)
[26P-pm027S]Palladium-catalyzed dehydrative cascade reactions of isatoic anhydrides in water
○Akihito Sato1, Makiko Takahashi1, Hidemasa Hikawa1, Shoko Kikkawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)
[26P-pm028]Studies on bi-directional nitroaldol reaction (2)
Futaba Nakazawa1, Erika Iwasaki1, Mei Kashihara1, Yusuke Akagi1, ○Toshiya Komatsu1 (1. Fac. Pharm. Sci., Teikyo Heisei Univ.)
[26P-pm029]Stduies on β-arylation of cyclic α,β-unsaturated oxime ethers
Shiori Fukuyama1, ○Yusuke Akagi1, Toshiya Komatsu1 (1. Fac. Pharm. Sci., Teikyo Heisei Univ.)
[26P-pm030]Synthesis of fluorine-derivatives of benzopyrans toward P2Y6 receptor antagonists
○Misaki Muto1, Asaka Tsutsumi1, Tomoko Mineno1 (1. Takasaki Univ. of Health and Welfare)
[26P-pm031]Synthesis of benzopyran derivatives as P2Y6 receptor antagonists
○Asaka Tsutsumi1, Masaaki Ito1, Isao Matsuoka1, Tomoko Mineno1 (1. Takasaki Univ. of Health and Welfare)
[26P-pm032]Liebeskind-type cross-coupling reaction of azole-thiones with triarylbismuthines
○Yuki Murata1, Misato Kiba1, Aki Terazoe1, Yuki Kitamura1, Mio Matsumura1, Shuji Yasuike1 (1. Sch. Pharm. Sci., Aichi Gakuin Univ.)
[26P-pm033S]Pd catalyzed cascade reaction using pentavalent organoantimony and o-hydroxycinnamic acid for the synthesis of 4-arylcoumarin
○Yuki Kitamura1, Yukari Kato1, Yuki Murata1, Mio Matsumura1, Shuji Yasuike1 (1. Sch. Pharm. Sic., Aichi Gakuin Univ.)
[26P-pm034]Synthesis and physical property of dibenzo[b,h]carbazole derivatives
○Mio Matsumura1, Miyuki Hiraiwa1, Masatoshi Kawahata2, Atsuya Muranaka3, Kentaro Yamaguchi2, Masanobu Uchiyama3,4, Shuji Yasuike1 (1. Sch. Pharm. Sci., Aichi Gakuin Univ., 2. Fac. Pharm. Sci. Kagawa Camp., Tokushima Bunri Univ., 3. Adv. Elem. Chem. Lab., RIKEN, 4. Grad. Sch. Pharm. Sci., Univ. Tokyo)
[26P-pm035]Structural change of diketopiperazines containing proline residue under basic condition
○Takuya Tsujita1, Ryohei Hagiwara1, Marina Ogata1, Takashi Ishizu1 (1. Faculty of Pharm. Sci., Fukuyama Univ.)
[26P-pm036]Molecular capture of diketopiperazines containing proline residue using tea gallate-type catechin (-)-epigallocatechin-3-O-gallate
○Takako Nomoto1, Karen Shinoda1, Miku Tokunaga1, Yukari Takagi1, Takashi Ishizu1 (1. Faculty of Pharm. Sci., Fukuyama Univ.)
[26P-pm037S]Design and synthesis of novel two-point recognition host compounds and research to the selective recognition of dicarboxylic acids
○Akiho Ozawa1, Tomoya Nobuta1, Noriyuki Yamagiwa1 (1. Takasaki University of Health and Welfare)
[26P-pm038]Production of cyclic-heterocyclic-compound : novel binding sites on molecular recognition
○Makoto Fukudome1, Takahiro Ishigaki1, Keita Akagaki1, De-Qi Yuan1 (1. Faculty of Pharmaceutical Sciences, Kobe Gakuin University)
[26P-pm039S]Synthesis and evaluation of 9-(aminoethoxy)phenoxazine conjugated oligonucleotide
○Ryohei Yamaji1, Yuki Kishimoto1, Akane Fujii1, Natsumi Nozaki1, Tomoki Matsumura1, Osamu Nakagawa1, Satoshi Obika1 (1. Grad. Sch. Pharm. Sci., Osaka Univ.)
[26P-pm040S]Development and self-assembly behavior of a fluorescent molecular tweezer that recognizes heme
○Koki Otani1, Yosuke Hisamatsu1, Naoki Umezawa1, Tsunehiko Higuchi1 (1. Grad. Sch. Pharm. Sci., Nagoya City Univ.)
[26P-pm041S]Inclusion crystals of V-shaped host molecule having trimethoxyphenyl groups with o-carborane
○Ryota Komatsu1, Masatoshi Kawahata2, Masahide Tominaga1, Tadashi Hyodo1, Kentaro Yamaguchi1 (1. Tokushim Bunri Univ., 2. Showa Pharmaceutical Univ.)
[26P-pm042S]Inclusion and structural analysis of six-membered cyclic ethers by a benzophenonediimide-based macrocycle
○Kosuke Mizuno1, Masahide Tominaga1, Tadashi Hyodo1, Kentaro Yamaguchi1 (1. Tokushima Bunri Univ.)
[26P-pm043S]Inclusion and structural analysis of five-membered cyclic ethers by a benzophenonediimide-based macrocycle
○Haruka Yamamoto1, Masahide Tominaga1, Tadashi Hyodo1, Kentaro Yamaguchi1 (1. Tokushima Bunri Univ.)
[26P-pm044S]Inclusion behavior of aromatic hydrocarbons obtained from porous crystals of cyclic compounds
○tadashi hyodo1, masatoshi kawahata2, masahide tominaga1, kentaro yamaguchi1 (1. Tokushima Bunri Univ., 2. Showa Pharm Univ.)
[26P-pm045S]Asymmetric transport of dicarboxylic acids through bulk liquid membrane using optically active norbornane derivatives as a carrier molecule
○Natsumi Tada1, Hiroto Kaku1, Ayaka Ise1, Sara Otsuru1, Jinuk Lee1, Mitsuyo Horikawa1, Kei Kitamura1, Tetsuto Tsunoda1 (1. Faculty of Pharm. Sci., Tokushima Bunri Univ.)
[26P-pm046S]Trial of the inclusion ability improvement by the β-cyclodextrin multimerizationⅡ -For medicine raw material-
○Tominaga Tatsuro1, Makoto Fukudome2, De-Qi Yuan1 (1. Grad. Sch. Pharm. Sci., Kobe Gakuin Univ., 2. Fac. Pharm. Sci., Kobe Gakuin Univ.)
[26P-pm047]Synthesis of fluorescent cyclodextrin modified dendrimer and application to drug carriers
○koki fukuda1, deti yuen1, makoto fukudome1 (1. kobegakuin Univ)
[26P-pm048S]Mechanism study of 1,4-dihydropyridine formation in water
○Mayu Anzai1, Yukie Yabe1, Shigeki Isomura1, Yoshinori Okuno1, Isao Azumaya2, Yasuo Sato1 (1. Yokohama University of Pharmacy, 2. Faculty of Pharmaceutical Science, Toho University)
[26P-pm049]Chennat-type synthesis of 1,4-dihydropyridine derivatives in water
○Chieka Kobayashi1, Ryuya Fujiyoshi1, Shigeki Isomura1, Yoshinori Okuno1, Yasuo Sato1 (1. Yokohama University of Pharmacy)
[26P-pm050S]Computational Augmentation about Diels-Alder reactions of 3-carbamoyl-2,4-dinitrophenylpyridinium
○Masataka Nakahara1, Kengo Hanaya1, Takeshi Sugai1, Shuhei Higashibayashi1 (1. Grad. Sch. Pharm. Sci., Keio Univ.)
[26P-pm051S]Development of chiral ligand grafted polymer catalysts and application to asymmetric alkylation using flow system.
○Airi Kakita1, Yoshinori Okuno1, Madoka Kamiharako1, Shouji Aoki2, Junichi Kanno2, Shigeki Isomura1, Yasuo Satou1 (1. Yokohama University of Pharmacy, 2. ECE Co.,Ltd.)
[26P-pm052]Effect of magnesium ion on the scavenging reaction of water-solubilized 2,2-diphenyl-1-picrylhydrazyl radical by caffeic acid in aqueous media
○Ikuo Nakanishi1, Yoshimi Shoji1, Kei Ohkubo1,2,3, Toshihiko Ozawa4, Shunichi Fukuzumi5, Ken-ichiro Matsumoto1 (1. Natl. Inst. Radiol. Sci., Natl. Inst. Quant. Radiol. Sci., 2. Inst. Adv. Co-Creation Stud., Osaka Univ., 3. Open Transdisciplinary Res. Initiatives, Osaka Univ., 4. Nihon Pharm. Univ., 5. Grad. Sch. Sci. Technol., Meijo Univ.)
[26P-pm053]Reactivity of highly stabilized carbanions in intramolecular nucleophilic addition of vinyl carbocation intermediates
○Hikaru Yanai1, Yuuki Fujimoto1, Takashi Matsumoto1, Irene Martín-Mejías2, Aragoncillo Cristina3, Pedro Almendros2 (1. Tokyo Univ. Pharm. Life Sci., 2. CSIC, 3. UCM)
[26P-pm054]Theoretical Studies for Conformations of Symmetric Diesters Considering Solvent Effects
○Satomi Niwayama1, Kento Osada1, Shota Matsushima1 (1. Graduate School of Engineering, Muroran Institute of Technology)
[26P-pm055S]Synthesis and crystal structure analysis of a series of Aib peptides having a sulfonamide moiety
○Ayaka Suzuki1, Ayaka Takahashi1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)
[26P-pm056S]Synthesis and crystal structure analysis of a series of short Aib-based peptides.
○Yuusuke Haga1, Mami Tanihira1, Naruka Sato1, Yoshiki Takahashi1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)
[26P-pm057S]Synthesis and crystal structure analysis of a series of Cbz-protected Aib peptides
○Miho Sakai1, Yuki Hirano1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)
[26P-pm058]Solid-state vibrational circular dichroism spectroscopy of aromatic sulfonamides
○Daichi Inoue1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)
[26P-pm059]Structural Features of Quinoline Sulfonamides: Their Polymorphs and Phase Transitions
○Hiroki Daitoku1, Shoko Kikkawa1, Akihiro Hirata1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)
[26P-pm060]Synthesis of macrocyclic aromatic hydrocarbons and conformational analysis thereof
○Ryota Nakagawa1, Hana Hirayama1, Ryohei Tsuchiya1, Yuuki Saito1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)
[26P-pm061]Synthesis of tetrapodal adamantane derivatives and structural analysis thereof
○Takaya Namikawa1, Riho Hakura1, Toshiki Sunakawa1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)
[26P-pm062S]Atropisomeric properties of N-alkyl-4-substituted 5H-dibenz[b,f]azepine
○Ayana Nabae1, Yuki Kanase2, Hidetsugu Tabata2, Kosho Makino1, Tetsuta Oshitari2, Hideaki Natsugari3, Hideyo Takahashi1 (1. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2. Faculty of Pharma Sciences, Teikyo University, 3. Faculty of Pharmaceutical Sciences, The University of Tokyo)
[26P-pm063S]Atropisomeric and conformational properties of fentanyl analogues
○Hironobu Arita1, Yuki Kanase2, Kosho Makino1, Hidetsugu Tabata2, Tetsuta Oshitari2, Hideaki Natsugari3, Hideyo Takahashi1 (1. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2. Faculty of Pharma Sciences, Teikyo University, 3. Faculty of Pharmaceutical Sciences, The University of Tokyo)
[26P-pm064S]Stereochemistry of 1, 4-benzodiazepines
○Ryoko Tanaka1, Yuki Kanase2, Kosho Makino1, Hidetsugu Tabata2, Tetsuta Oshitari2, Hideaki Natsugari3, Hideyo Takahashi1 (1. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2. Faculty of Pharma Sciences, Teikyo University, 3. Faculty of Pharmaceutical Sciences, The University of Tokyo)
[26P-pm065S]Synthesis and atropoisomeric properties of dibenzoazepine analogs
○Mayuno Hotta1, Takuya Namba1, Kosho Makino1, Hidetsugu Tabata2, Tetsuta Oshitari2, Hideaki Natsugari3, Hideyo Takahashi1 (1. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2. Faculty of Pharmaceutical Sciences, Teikyo University, 3. Faculty of Pharmaceutical Sciences, The University of Tokyo)
[26P-pm066S]Synthesis of macrocyclic aromatic amides which can be functionalized on their aromatic rings
○Masako Tashiro1, Yuu Aoyama1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. pharm. Sci., Toho Univ.)
[26P-pm067S]Synthesis of cylindrical aromatic amides having ethynylene group and structural analysis thereof
○Yuuki Saito1, Misa Satake1, Kozue Tsuneizumi1, Ryoko Sakagami1, Ryuichi Mori1, Hyuma Masu2, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ., 2. CAI, Chiba Univ.)
[26P-pm068]Synthesis of macrocyclic aromatic amides which have diphenyldianthracene skeletons and conformational analysis thereof
○Hisato Takahashi1, Akane Yoshida1, Ryosuke Kori1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)
[26P-pm069S]Synthesis of macrocyclic aromatic amides which have adamantane skeletons.
○Shun Hashimoto1, Rina Shimizu1, Kei Takamatsu1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)
[26P-pm070]Short step syntheis of spherical aromatic amides and structural analysis thereof
○Rintaro Nimoda1, Ayako Chiba1, Hyuma Masu2, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ., 2. CAI, Chiba Univ.)
[26P-pm071]Sythesis of spherical aromatic amides which can be functionalized and stereochemistry thereof
○Shogo Suzuki1, Ayako Chiba1, Hyuma Masu2, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ., 2. CAI, Chiba Univ.)
[26P-pm072]Synthesis and properties of π-extended dihydro[5]helicenyl phosphine
○Kazuteru Usui1, Nozomi Narita1, Takahiro Fukunaga1, Atsushi Yokoo2, Kosuke Yamamoto2, Yasufumi Fuchi1, Kazunobu Igawa3, Katsuhiko Tomooka3, Satoru Karasawa1 (1. Faculty of Pharm. Sci., Showa Pharm. Univ., 2. Grad. Sch. of Pharm. Sci., Kyushu Univ. , 3. Inst. Mat. Chem. and Eng., Kyushu Univ.)
[26P-pm073S]Synthesis of low symmetrical ball-shaped metal complexes with cyano groups
○Sari Ishikawa1, Hajime Maeda1, Masahito Segi1, Taniyuki Furuyama1,2 (1. Grad. Sch. of Nat. Sci. and Tech. Kanazawa Univ., 2. JST PRESTO)
[26P-pm074]Synthesis and fluorescence properties of diarylmethyleneimidazolinones bearing NADH-NAD+-like structures
○Aki Fujisaka1, Yuki Shimozono1, Aya Ikeshita1, Sakiho Hamakubo1, Masahiro Ikejiri1, Kazuyuki Miyashita1 (1. Faculty of Pharmacy, Osaka Ohtani University)
[26P-pm075S]Reactivities and physical properties of emissive diquinolylamine derivatives
○Ami Amano1, Yasufumi Fuchi1, Kazuteru Usui1, Ryusuke Hagihara2, Satoru Karasawa1 (1. Faculty of Pharm. Sci. Showa Pharmaceutical Univ., 2. Grad. Sch. Pharm. Sci., Kyushu Univ.)
[26P-pm076S]Conformational analysis and functionalization of peptides containing a chiral nitrogen-containing five-membered ring α,α-disubstituted amino acid
○Yuto Yamaberi1, Ryo Eto2, Tomohiro Umeno2, Makoto Oba2, Masakazu Tanaka2 (1. Sch. Pharm. Sci., Nagasaki Univ., 2. Grad. Sch. Bio. Sci., Nagasaki Univ.)
[26P-pm077S]Intermolecular interactions in the coexistence of cell-penetrating peptides and drug molecules
○Takamasa Matsuo1, Shino Kinugasa1, Reji Ishida1, Kazuhiro Kudo1,2, Komei Okabe1,2, Hiroshi Enomoto2, Takahiro Honda1,2 (1. NAIST, 2. Santen Pham.)
[26P-pm078S]Synthesis and binding properties of chloroalkene-type PBB3 compounds targeting neurofibrillary tangles
○Hiro Takeda1, Ryuji Kyan2, Kohei Sato1,3, Nobuyuki Mase1,2,3, Tetsuo Narumi1,2,3 (1. Fac. Eng., Shizuoka Univ., 2. Grad. Sch. Sci. Tech., Shizuoka Univ., 3. Grad. Sch. Integ. Sci. Tech., Shizuoka Univ.)
[26P-pm079S]Development of G-quadruplex selective binding RGG peptides containing Gly-Gly-type (E)-methylalkene dipeptide isosteres
○Hikari Okita1, Yuna Kato2, Takuma Nishizawa2, Kohsuke Arai2, Kohei Sato1,2, Nobuyuki Mase1,2, Takanori Oyoshi2, Tetsuo Narumi1,2 (1. Fac. Eng., Shizuoka Univ., 2. Grad. Sch. Integ. Sci. Tech., Shizuoka Univ.)
[26P-pm080S]p-type hydrogen bonding potential of (Z)-fluoroalkene dipeptide isostere
○Takaya Kawaguchi1, Yuki Kodama2, Kohei Sato1,3, Nobuyuki Mase1,2,3, Tetsuo Narumi1,2,3 (1. Fac. Eng., Shizuoka Univ., 2. Grad. Sch. Sci. Tech., Shizuoka Univ., 3. Grad.Sch. Integ. Sci. Tech., Shizuoka Univ.)
[26P-pm081S]Spontaneous resolution of the chiral crystal and crystal structure analysis of N,N'-dimethylpyridine-2,6-dicarboxamides bearing pyrimidine
○Youhei Fujii1, Ai Ito1, Ruri Kozono1, Tatsuya Yamaguchi1, Yuichi Sugiki1, Kazuo Fukuda1, Ryu Yamasaki1, Iwao Okamoto1 (1. Showa Pharm. Univ.)
[26P-pm082S]Structures and Reactivities of N-Ethynylated N-Benzyl Amide Compounds
○Shuya Nakamura1, Ryu Yamasaki1, Kento Morita1, Kazuo Fukuda1, Ai Ito1, Iwao Okamoto1 (1. Showa Pharm. Univ.)
[26P-pm083]Study of molecular configuration of peptide-based drugs using NMR finger-print analysis
○Takashi Misawa1, Yosuke Demizu1,2 (1. NIHS, 2. Grad. Sch. Med. Life Sci. Yokohama city Univ.)
[26P-pm084]Synthesis and evaluation of FICA derivatives as chiral derivatizing agents
○Tamiko Takahashi1, Tomoyo Kamei1, Jyunichi Koyanagi1, Hiroyuki Teramae2 (1. Fac. Pharm. Sci., Josai Intl. Univ., 2. Grad. Sch. Sci., Josai Univ.)
[26P-pm085S]Cyclization of glutathione and a new radical scavenging mechanism
○Hiyori Furumachi1, Yuta Morishita1, Takashi Fujimoto2, Tomoyuki Fujita1,3, Ayumi Tsutsui1,3 (1. Fuct.Agric.Shinsyu Univ., 2. Col.Sci.Tech.Meisei Univ., 3. Grad.Sch.Agric.Shinsyu Univ.)
[26P-pm086]Development of highly sensitive fluorescent probe for cellular glucose uptake assay.
○Norio Hirakawa1, Takashi Shimomura1, Reina Kitamura1, Katsuya Noguchi1, Yuya Ohuchi1, Munetaka Ishiyama1 (1. Dojindo Laboratories.)
[26P-pm087]The tumbling of the modified glucose unit in a 6-bridged cyclodextrin dimer: a new route to the pseudo-rotaxane structure
○Kazutaka Koga1, Kanna Nishida2, Makoto Fukudome2, De-Qi Yuan2 (1. Daiichi Univ. Pharm., 2. Fac. Pharm. Sci., Kobe Gakuin Univ.)
[26P-pm088]Primer extension reactions through formation of CuI-mediated base pairs by DNA polymerase
○Mizuki Hakuba1, Ken Nakata1, Junsuke Hayashi1, Shun-ichi Wada1, Hidehito Urata1 (1. Osaka Univ. Pharm. Chem)
[26P-pm089S]Direct Visible Light-Excitation of Alkylborates Enabling Ni-Catalyzed Cross-Couplings
○Yukiya Sato1, Kei Nakamura1, Yuto Sumida1,3, Takamitsu Hosoya2,3, Hirohisa Ohmiya1 (1. Division of Pharmaceutical Sciences, Graduate School of Medical Sciences, Kanazawa University, 2. Laboratory of Chemical Bioscience, Institute of Biomaterials and Bioengineering, Tokyo Medical and Dental Univ. (IBB,TMDU), 3. Laboratory for Chemical Biology, RIKEN Center for Biosystems Dynamics Research (BDR))
[26P-pm090S]Design and synthesis of supramolecular complexes formed by the self-assembly of monoalkyated dizinc(II) complex, copper and diimide units functionalized with lewis acid or crown ether moieties
○Akib Bin Rahman1, Yuya Miyazawa1, Shin Aoki1 (1. Faculty of Pharmaceutical Sciences, Tokyo University of Science)
[26P-pm091]Effects of fermentation by lactic acid bacteria on skin of HR-AD fed hairless mice
○Tsuyoshi Tamane1,2, Yoshihiro Tokudome2 (1. Koei-science, 2. Josai Univ.)