Session Details
[S09]How was the original drug discovery research born? --2020 Breakthrough Award of the Division of Medicinal Chemistry, PSJ and 2019 Award for Excellent General Presentation in the Medicinal Chemistry Symposium--
Sat. Mar 27, 2021 1:15 PM - 3:15 PM JST
Sat. Mar 27, 2021 4:15 AM - 6:15 AM UTC
Sat. Mar 27, 2021 4:15 AM - 6:15 AM UTC
[Room I] Oral Presentation I Online
Organizer: Habashita Hiromu (Ono Pharmaceutical Co., Ltd.), Otaka Akira (Faculty of Pharm. Sci., Tokushima Univ.), Aoki Kazumasa (Daiichi Sankyo Co., Ltd.)
Division of Medicinal Chemistry at The Pharmaceutical Society of Japan commends research results, including innovative content that contributes to the development of drug discovery, as Breakthrough Award of the Division of Medicinal Chemistry, PSJ. Specifically, the awards are given to original research on drugs or bioactive compounds that have a novel chemical structure as pharmaceuticals, and original research that contributes to drug discovery with new technologies and methods. In addition, from the general oral presentations and poster presentations at the Medical Chemistry Symposium, several research results including remarkable contents that contribute to the progress and future development of drug discovery are commended as Award for Excellent General Presentation in the Medicinal Chemistry Symposium. At this symposium, the award ceremony and award lecture of the 2020 Breakthrough Award of the Division of Medicinal Chemistry, PSJ, and the award lecture of the 2019 Award for Excellent General Presentation in the Medicinal Chemistry Symposium will be given. We hope that through the active sharing of knowledge and experience of these excellent research results, new ideas that will lead to the identification of breakthrough new drugs will be born.
オーガナイザー挨拶:巾下 広(小野薬品工業)
[S09-1]Design, construction, and screening of a one-bead-one-compound library for discovery of potent analogues of antibiotic lysocin E
○Kotaro Tokumoto1, Takuya Kaji1, Hiroaki Itoh1, Masayuki Inoue1 (1. Grad. Sch. Pharm. Sci., The Univ. of Tokyo)
[S09-2]Discovery of TAS-116 as a novel orally available HSP90 inhibitor
○Takao Uno1, Yuichi Kawai1, Satoshi Yamashita1, Hiromi Oshiumi1, Chihoko Yoshimura1, Takashi Mizutani1, Tatsuya Suzuki1, Khoon Tee Chong1, Kazuhiko Shigeno1, Mitsuru Ohkubo1, Yasuo Kodama1, Hiromi Muraoka1, Kaoru Funabashi1, Koichi Takahashi1, Shuichi Ohkubo1, Makoto Kitade1 (1. Taiho Pharmaceutical Co., Ltd.)
医薬化学部会賞 授賞式&記念撮影
[S09-3]Discovery of delgocitinib as a novel JAK inhibitor
○Satoru Noji1, Yoshinori Hara1, Tomoya Miura1, Hiroshi Yamanaka1, Makoto Shiozaki1 (1. JAPAN TOBACCO INC)
[S09-4]The discovery of a novel siderophore cephalosporin Cefiderocol
○Toshiaki Aoki1, Kenji Yamawaki2, Takafumi Sato2, Yasuhiro Nishitani2, Yoshinori Yamano2 (1. CMC R&D Division, SHIONOGI & CO., LTD., 2. Pharmaceutical Research Division, SHIONOGI & CO., LTD.)
