Session Details
[27P02]全合成・その他の合成
Sat. Mar 27, 2021 9:00 AM - 6:00 PM JST
Sat. Mar 27, 2021 12:00 AM - 9:00 AM UTC
Sat. Mar 27, 2021 12:00 AM - 9:00 AM UTC
[Room P02] Poster Presentation Online
[27P02-001]Study on asymmetric total synthesis of (-)-dichroanal A
Minoru Ozeki1, ○Miyu Yamakita1, Rikako Suzuki1, Aya Niki1, Syui Aoki1, Hiroki Iwasaki2, Naoto Kojima2, Masayuki Yamashita2, Ikuo Kawasaki1 (1. School of Pharmacy and Pharmaceutical Science, Mukogawa Women’s University, 2. Kyoto Pharmaceutical University)
[27P02-002]Efficient synthesis of pyridine-maleimide derivatives and their fluorescence
○Masayori Hagimori1, Yasuhisa Nishimura2, Tasusada Yoshida3, Yukiko Ogawa3, Keitaro Tanaka3 (1. Sch. Pharm., Mukogawa Women's Univ., 2. Sch. Eng., Nagasaki Univ. , 3. Fucl. Pharm. Sci., Nagasaki Int. Univ.)
[27P02-003]Total synthesis of dibenzofuran natural product karnatakafuran B
○Yuhzo Hieda1,2, Tominari Choshi2, Haruto Fujioka2 (1. Common Resources Center Fukuyama university, 2. Faculty of Pharmacy and Pharmaceutical Sciences Fukuyama University)
[27P02-004]Synthetic Study of Gulmirecin A
Shun KITAHATA1, ○Akira KATSUYAMA1, Satoshi ICHIKAWA1,2 (1. Faculty of Pharmaceutical Sciences Hokkaido Univ., 2. GI-CoRE, Hokkaido University,)
[27P02-005]Total Synthesis of Echinomycin
○Satoshi Ichikawa1, Keita Kojima1, Fumika Yakushiji1, Akira Katsuyama1 (1. Faculty of Pharmaceutical Science, Hokkaido University)
[27P02-006S]Total synthetic study of Actinoallolide A, anti-Trypanosoma agent
○Takanori Ohno1, Yoshihiko Noguchi1,2, Akito Watanabe1, Masato Iwatsuki1,2, Yuki Inahashi1,2, Tomoyasu Hirose1,2, Toshiaki Sunazuka1,2 (1. Grad. Sch. of Infect. Control Sci., Kitasato Univ., 2. Ōmura Satoshi memorial Inst., Kitasato Univ.)
[27P02-007S]Synthesis and SAR Study of the Antimalarial agent, Kozupeptin A, Using a Designed Hydrophobic Anchor Molecule
○Akari Ueda1, Tomoyasu Hirose1,2, Yumi Hayashi1, Masato Iwatsuki1,2, Rei Hokari1,2, Aki Ishiyama1,2, Toshiaki Sunazuka1,2 (1. Grad. Sch. Infection. Control Sci., Kitasato Univ., 2. Ōmura Inst., Kitasato Univ.)
[27P02-008S]Synthetic study on celludinones A and B
○Tomoka Sato1, Taichi Ohshiro1, Hiroshi Tomoda1, Tohru Nagamitsu1 (1. Sch. Pharm., Kitasato Univ.)
[27P02-009]Synthtic studies on C-mannosyl tryptophan via Iridium-catalyzed vinylic C-H borylation
○Osamu Hara1, Yasuhiro Nishikawa1, Tatsuaki Baba1, Daiki Kato1, Kazushi Yamakita1, Natsuki Watanabe1, Ken Ito1, Iori Kishihata1 (1. Faculty of Pharmacy, Meijo University)
[27P02-010S]Gymnocin-B synthetic research -ABC and JK fragment synthesis research using common raw materials-
○Shiori Takeuchi1, Mai Kikuyama1, Yuna Aoki1, Yumiko Imai1, Takeo Sakai1, Yuji Mori1 (1. Faculty of Pharmacy, Meijo University)
[27P02-011S]Synthesis of the FG Fragment of Gymnocin-B
○Ryuki Oyachi1, Takeo Sakai1, Yuji Mori1 (1. Faculty of Pharmacy, Meijo Univ.)
[27P02-012S]Synthetic studies on 13-hydroxy-15-oxozoapatlin
○Masahiro Asakawa1, Kokoro Nagasawa1, Matsunaga Kazuma1, Atsushi Kishida1, Kazuhiko Takatori1 (1. Meiji Pharmaceutical University)
[27P02-013S]The molecular basis for the biosynthesis of coprinoferrin, a basidiomycetous siderophore vital to fungal cell development
○Shihori Asai1, Yuta Tsunematsu1, Jun Takanishi1, Tomoki Isogai2, Ichiro Hayakawa3, Akira Sakakura2, Kenji Watanabe1 (1. Dept. Pharm. Sci., Univ. Shizuoka, 2. Grad. Sch. Nat. Sci. Tech., Okayama Univ., 3. Grad. Sch. of Int. Bas. Sci., Nihon Univ.)
[27P02-014]Synthesis of benzothiazole-linked polycyclic compounds via intramolecular C-H bond activation - cyclization and application to macrocyclic compounds
Madoka Waku1, Takumi Abe1, ○Daisuke Sawada1 (1. Grad. Sch. Med. Dent. Pharm. Sci., Okayama Univ.)
[27P02-015]Divergent synthesis of γ-alkylidene butenolides from Thai medicinal plant Melodorum fruticosum and evaluation of those inhibitory effects on melanogenesis
○Genzoh Tanabe1,2, yuri siotani1, katsuki takashima1, toshio morikawa2, kiyofumi ninomiya2, hirofumi isikawa1 (1. Fac. Pharm., Kindai Univ., 2. Pharm. Res. Tech. Inst., Kindai University)
[27P02-016]Synthesis of transposition analogues of CJ-14877 and their inhibitory activity of interleukin-1β
○Nao Watanabe1, Natsumi Yagyu1, Yuna Tsuji1, Izumi Sakai1, Eri Nagata1, Yukina Omura1, Nozomi Kitazawa1, Yoshiyuki Adachi2, Naohito Ohno2, Reiko Yano1, Yukio Hitotsuyanagi2, Koichi Takeya2, Yutaka Aoyagi1 (1. College of Pharmacy, Kinjo Gakuin University, 2. School of Pharmacy, Tokyo University of Pharmacy and Life Sciences)
[27P02-018S]Preparation of chafuroside B, starting from naturally abundant D-arabinosylvitexin
○Kazuki Kurahayashi1, Kengo Hanaya1, Shuhei Higashibayashi1, Takeshi Sugai1 (1. Grad. Sch. Pharm. Sci., Keio Univ.)
[27P02-019]Synthetic Studies of Polymer Libraries using Half-esters Obtained by Practical Selective Monohydrolysis Reactions of Symmetric Diesters
Jianjun Shi1, Wataru Shoji1, Taiga Takayama1, Yuichiro Imura1, ○Satomi Niwayama1 (1. Grad. Sch. Eng. Muroran Institute of Technology)
[27P02-020S]Gold-catalyzed synthesis of 1,2,3-trisubstituted indanes in ionic liquid
○Hitomi Chiaki1, Nobuyoshi Morita1, Kanae Ikeda1, Kosaku III Tanaka1, Yoshimitsu Hashimoto1, Osamu Tamura1 (1. Showa Pharmaceutical University)
[27P02-021]Synthetic study of ζ-carotene geometric isomers
○Chisato Tode1, Naruse Kadowaki1, Kenjirou Sugiyama2, Takashi Maoka3, Atsuko Takeuchi1 (1. Kobe Pharmaceutical Univ., 2. Kogakuin Univ., 3. Research Institute for Production Development)
[27P02-022S]Kinetic study of intramolecular Na-to-Nb acyl migration of peptide agonists selective to neuromedin U receptor type 2
○Daichi Toyama1, Kosuke Arai2, Kohei Sato1,2,3, Nobuyuki Mase1,2,3, Kentaro Takayama4, Tetsuo Narumi1,2,3 (1. Fac. Eng., Shizuoka Univ., 2. Grad. Sch. Integ. Sci. Tech., Shizuoka Univ., 3. Grad. Sch. Sci. Tech., Shizuoka Univ., 4. Kyoto Pharm. Univ.)
[27P02-023S]Chemical Synthesis of Amide Analogues of Ester-Linked Ubiquitin Dimer for Improving Chemical Stability
○Yoshinori Taguchi1, Takuma Nishizawa2, Reon Takeuchi3, Syoko Tanaka3, Nobuyuki Mase1,2,3, Fumiaki Ohtake4, Yasushi Saeki5, Kohei Sato1,2,3, Tetsuo Narumi1,2,3 (1. Fac. Eng., Shizuoka Univ. , 2. Grad. Sch. Integ. Sci. Tech., Shizuoka Univ., 3. Grad. Sch. Sci. Tech., Shizuoka Univ., 4. Hoshi Univ., 5. Tokyo Metropoli. Inst. Med. Sci.)
[27P02-024S]Search for novel guanine quadruplex-binding peptide compounds based on alkene-type peptide bond isostere
○Sayuri Takeo1, Maiko Tabata2, Yuna Kato2, Saki Imai2, Kohei Sato1,2, Nobuyuki Mase1,2, Takanori Oyoshi2, Tetsuo Narumi1,2 (1. Fac. Eng., Shizuoka Univ., 2. Grad. Sch. Integ. Sci. Tech.)
[27P02-025S]Design and synthesis of vitamin D3 derivatives with fluorinated side chain
○Sayuri Mototani1, Fumihiro Kawagoe1, Kaori Yasuda2, Toshiyuki Sakaki2, Atsushi Kittaka1 (1. Faculty Pharm. Sci., Teikyo Univ., 2. Faculty of Engineering, Toyama Prefectural Univ.)
[27P02-026]Stereoselective synthesis of 24-hydroxylated vitamin D3 analogues
○Fumihiro Kawagoe1, Sayuri Mototani1, Kaori Yasuda2, Toshiyuki Sakaki2, Atsushi Kittaka1 (1. Faculty Pharm. Sci., Teikyo Univ., 2. Faculty of Engineering, Toyama Prefectural Univ.)
[27P02-027S]Design and synthesis of proline-based thioglycosides for programmed oligosaccharide synthesis
○Ryota Naoi1, Tomohiro Tanaka1, Shin Aoki1,2 (1. Tokyo University of Science, 2. Research Institute for Science & Technology)
[27P02-028]A Synthetic Study of Oridamycin Analogs
○Naoto Yamasaki1, Esumi Tomoyuki1, Hiromichi Kenmoku1, Yoshinori Asakawa1, Hirofumi Yamamoto1 (1. Fac. Pharm. Sci., Tokushima Bunri Univ.)
[27P02-029]The Fluorescence-Activity Relationship Study of Dehydroantofine
Ikumi Iwasaki1, Naoto Yamasaki1, Rei Hokari2, Masato Iwatsuki2, Aki Ishiyama2, Tomoyuki Esumi1, Hiromichi Kenmoku1, Yoshinori Asakawa1, ○Hirofumi Yamamoto1 (1. Fac. Pharm. Sci., Tokushima Bunri Univ., 2. Ōmura Inst., Kitasato Univ.)
[27P02-030S]Chemical conversion of aphid pigments: red uroleuconaphin A1 to green viridaphin A2
○Chiharu Ozakai1, Kei Kitamura1, Tosho Hoshiyama1, Akari Imamura1, Mitsuyo Horikawa1, Tatsuro Yoneyama1, Akemi Umeyama1, Tetsuto Tsunoda1, Hiroto Kaku1 (1. Faculty of Pharm. Sci., Tokushima Bunri Univ.)
[27P02-031S]The Synthesis of FG-beads linked Thallusin
○Ayari Oshiro1, Kento Sumitomo1, Naoto Yamasaki1, Tomoyuki Esumi1, Hiromichi Kenmoku1, Yoshinori Asakawa1, Yusuke Kasai1, Hiroshi Imagawa1, Takashi Kuzuhara1, Hirofumi Yamamoto1 (1. Fac. Pharm. Sci., Tokushima Bunri Univ.)
[27P02-032]Synthesis of benzothiophene using ring-opening cyclization of spirocyclopropanes with sulfur nucleophile
○Hisanori Nambu1, Yuki Seto1, Yuta Onuki1, Takayuki Yakura1 (1. Fac. Pharm. Sci., Univ. Toyama)
[27P02-033]A concise synthesis of thiosugar skeleton
○Hiroko Kakuda1, Yasutake Takahashi1 (1. Institute of Liberal Arts and Sciences, Univ. of Toyama)
[27P02-034]Studies on the synthesis and reaction of spiro-epoxy-pyrazol-3-one derivatives
○Hayate Nagabuchi1, Eiichi Masumoto1, Mayu Hikita1, Fumi Okabe-Nakahara1, Hiroshi Maruoka1 (1. Pharm. Sci., Fukuoka Univ.)
[27P02-035]Synthetic Studies of Novel Spiro[pyrazole-4,2′-quinazoline]-5,4′-dione Derivatives
○Eiichi Masumoto1, Hayate Nagabuchi1, Azusa Mikuriya1, Chijiiwa Risa1, Fumi Okabe-Nakahara1, Hiroshi Maruoka1 (1. Fac. Pharm. Sci., Fukuoka Univ.)
[27P02-036]Synthetic study of benzo[b]phosphole oxide derivatives focusing on the substituents of phosphorus atom
○Takehiro Yamagishi1, Kouki Nakahara1, Moe Kato1, Kyosuke Kaneda1 (1. Faculty of Pharmaceutical Sciences, Hokkaido University of Science)
[27P02-037S]Synthesis and SAR study of the antimalarial troponoids
○Asuka Nakajima1, Ryo Saito1, Goh Sennari1, Masato Iwatsuki1,2, Aki Ishiyama1,2, Rei Hokari2, Kazuhiko Otoguro2, Tomoyasu Hirose1,2, Toshiaki Sunazuka1,2 (1. Grad. Sch. Infection Control Sci., Kitasato Univ., 2. Ōmura Inst., Kitasato Univ.)