The 141st Annual Meeting of the Pharmaceutical Society of Japan (Hiroshima)
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Session Details

Poster Presentation(A) Organic Chemistry

[27P02]構造活性相関①

Sat. Mar 27, 2021 9:00 AM - 6:00 PM JST
Sat. Mar 27, 2021 12:00 AM - 9:00 AM UTC
[Room P02] Poster Presentation Online

[27P02-062]Examination of the antimicrobial activity of C-terminal amide derivatives of myticalin A6 (3-23)-OH

○Keiko Okimura1, Tamako Shiratori1, Atsuya Sawada1, Chinami Katsui1, Tohru Daikoku1 (1. Fac. Pharm. Sci., Hokuriku Univ.)

[27P02-063S]Development of helical peptides containing non-proteinogenic amino acids inhibiting VDR-coactivator interaction

○Mami Takyo1,2, Yuumi Sato1,2, Hiroaki Ishida3, Keiko Yamamoto3, Takashi Misawa2, Yosuke Demizu1,2 (1. Grad. Sch. Med. Life Sci., Yokohama city Univ., 2. NIHS, 3. Showa Pharm. Univ.)

[27P02-064S]Synthesis and biological evaluation of cinnamoylchromone derivatives as monoamine oxidase inhibitors

○Yuri Takemura1, Tomoka Aiba2, Koichi Takao2, Hitoshi Kamauchi2, Yoshiaki Sugita2 (1. Grad. Sch. Pharm. Sci., Josai Univ., 2. Pharm. Sci., Josai Univ.)

[27P02-065S]Synthesis and biological evaluation of gingerol derivatives as neuroprotective agents

○Takumi Oda1, Koichi Takao2, Hitoshi Kamauti2, Yoshiaki Sugita2 (1. Grad. Sch. Pharm. Sci., josai Univ, 2. Pharm. Sci., josai Univ)

[27P02-066S]Synthesis and evaluation of selective tumor cell death induction by kukoamine derivatives.

○Asuka Aoyama1, Koichi Takao2, Hitoshi Kamauchi2, Yoshiaki Sugita2 (1. Grad. Sch. Pharm. Sci., Josai Univ., 2. Pharm. Sci., Josai Univ.)

[27P02-067S]Synthesis of strychnos alkaloid derivatives and evaluation of their cholinesterase inhibitory activity.

○Koki Ueno1, Hitoshi Kamauchi2, Koichi Takao2, Yoshiaki Sugita2 (1. Grad. Sch. Pharm. Sci., Josai Univ., 2. Pharm. Sci., Josai Univ.)

[27P02-068S]Synthesis and biological evaluation of piperic acid and cinnamic acid derivatives

○Daiki Taki1, Koichi Takao2, Hitoshi Kamauchi2, Yoshiaki Sugita2 (1. Grad. Sch. Pham. Sci., Josai Univ., 2. Pham. Sci., Josai Univ.)

[27P02-069]Structure-Activity Relationship Study of the Metallo-β-lactamase Inhibitor, ODTAA

○Kiki Nakazato1, Akari Ikeda1,2, Akihiro Tomiyama1, Yoshiki Ikegaya1, Masako Honsyou2, Hiroyuki Asami1,2, Tomoyasu Hirose1,2, Toshiaki Sunazuka1,2 (1. Grad. Sch. Infection Control Sci., Kitasato Univ., 2. Ōmura Inst. Kitasato Univ.)

[27P02-070S]Synthesis and biological evaluation of aromatic polyketide derivatives

○Masafumi Takanashi1, Hitoshi Kamauchi2, Koichi Takao2, Yoshiaki Sugita2 (1. Grad. Sch. Pharm. Sci., Josai Univ., 2. Pharm. Sci., Josai Univ.)

[27P02-071S]Synthesis of polycyclic pyridone derivatives and their anti-hyphae formation and biofilm formation activity

○Yu Kimura1, Hitoshi Kamauchi1, Mikoto Ushiwatari1, Taishi Seki1, Koichi Takao1, Yoshiaki Sugita1 (1. Pham. Sci., Josai Univ.)

[27P02-072]Discovery of novel isothiourea derivatives as potent dual inhibitors of IDO1 and TDO for cancer immunotherapy

○Naohisa Ogo1, Masaya Nonaka1, Momoko Ishihara1, Mito Watanabe1, Katsumi Ota1, Hisashi Murakami1, Osamu Takikawa2, Akira Asai1 (1. Grad. Div. of Pharma. Sci., Univ. of Shizuoka, 2. AMED)

[27P02-073S]Synthesis and evaluation of antimicrobial fluorine-containing naphthoquinone derivatives

○Ayuka Tatsumi1, Mitsuaki Yamashita1, Jun Sawano1, Ryuji Umeda1, Yuko Kumeda2, Youichi Fukuda1, Akira Iida1 (1. Faculty of Agriculture, Kindai Univ., 2. Research Center for Microorganism Control, Osaka Prefecture Univ.)

[27P02-074S]Synthesis of α-methylenecyclopentanones for the development of NFκB inhibitors

○Aya Shiuchi1, Aki Kohyama1, Rei Yokoyama1, Zhou Yue1, Hiroaki Sakurai1, Yuji Matsuya1 (1. Faculty of Pharmaceutical Sciences, University of Toyama)

[27P02-075]Synthesis of 4’-substituted 2’-deoxy-4’-thiocytidines and its Evaluation for Antineoplastic and Antiviral Activities

○Kazuhiro Haraguchi1, Hiroki Kumamoto1, Kiju Konno2, Hideki Yagi2, Yutaka Tatano3, Yuki Odanaka4, Satoko Shimbara Mastubayashi4, Robert Snoeck5, Graciela Andrei5 (1. DDepartment of Pharmaceutical Sciences, Nihon Pharmaceutical University, 2. Department of Pharmaceutical Sciences, International University of Health and Welfare, 3. International University of Health and Welfare Department of Pharmaceutical Sciences, School of Pharmacy at Fukuoka, 4. School of Pharmacy, Showa University, 5. Rega Institute for Medical Research, Katholieke Universiteit Leuven)

[27P02-076]Antitumor effects of 6-TMNQ and its derivatives on Colon-26 colon cancer cells

○Yu Jin1, Aika Ohno1, Kaho Ono1, Hiyo Okamoto1, Haruka Toda1, Sakura Fuchiwaki1, Michiko Wada1, Tetsutaro Kimachi1, Satoru Takahashi1 (1. Sch. Pharmcy & Pharm. Sci., Mukogawa Women's Univ.)

[27P02-077S]Structure-activity relationships of SR-12813 for HMG-CoA reductase degradation

○Kota Kawamura1, Hiromasa Yoshioka2, Koji Kuramochi1, Kenji Ohgane1 (1. Tokyo Uni. of Science, 2. RIKEN)
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