The 141st Annual Meeting of the Pharmaceutical Society of Japan (Hiroshima)
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Session Details

Oral Presentation(A) Organic Chemistry

[27V03-am]ケミカルバイオロジー②

Sat. Mar 27, 2021 10:36 AM - 12:00 PM JST
Sat. Mar 27, 2021 1:36 AM - 3:00 AM UTC
[Room V03] Oral Presentation 3 Online
座長：山次 健三（東大院薬）、家田 直弥（名市大）
10:36 AM - 10:48 AM JST(1:36 AM - 1:48 AM UTC)

[27V03-am08S]Incorporation of a coumarin unit into a PPARγ agonist

○Chisato Yoshikawa1, Hiroaki Ishida1, Nami Ohashi1, Toshimasa Itoh1 (1. Showa Pharm. Univ.)
10:48 AM - 11:00 AM JST(1:48 AM - 2:00 AM UTC)

[27V03-am09]Development of c-di-GMP derivatives with amine skeleton and evaluation of their inhibitory activity against biofilm formation

○Genichiro Tsuji1, Kentaro Ikeda1,2, Yuuta Yanase1,2, Hayashi Katsuhiko1, Kudo Yukiko1, Demizu Yosuke1,2 (1. NIHS, 2. Grad. Sch. Med. Life Sci., YCU)
11:00 AM - 11:12 AM JST(2:00 AM - 2:12 AM UTC)

[27V03-am10S]Development of novel hypoxia-inducible factor-1 (HIF-1) inhibitors with a pyrazole scaffold

○Marina Sakai1, Nobuaki Takahashi1, Yutaka Furutani2, Takehiro Suzuki3, Naoshi Dohmae3, Sayaka Kobayashi1, Akira Hattori1, Hiroshi Harada4, Hideaki Kakeya1 (1. Grad. Sch. Phar. Sci., Kyoto Univ., 2. RIKEN CPR, 3. RIKEN CSRS, 4. GSB, Kyoto Univ.)
11:12 AM - 11:24 AM JST(2:12 AM - 2:24 AM UTC)

[27V03-am11S]Amphiphilic Cationic Triscyclometalated Iridium(III) Complex-Peptide Hybrids Induce Paraptosis-like Cell Death of Cancer Cells via and Intracellular Ca2+-Dependent Pathway

○Kenta Yokoi1, Chandrasekar Balachandran1, Shin Aoki1,2 (1. Fac. Pharm. Sci., 2. Research Institute of Science and Tecnology)
11:24 AM - 11:36 AM JST(2:24 AM - 2:36 AM UTC)

[27V03-am12S]Development of a tumor-selective activatable photosensitizer based on bismuth-rhodamine

○Akari Mukaimine1, Tasuku Hirayama1, Mieko Tsuji1, Hideko Nagasawa1 (1. Gifu Pharm. Univ. )
11:36 AM - 11:48 AM JST(2:36 AM - 2:48 AM UTC)

[27V03-am13S]Elucidation of cell-membrane penetration mechanisms of saporin toxin and application for drug delivery

○Momoko Obuki1, Miku Katayama1, Kosuke Noguchi1, Stefania Zuppone2, Mayu Yamana3, Tomoka Takatani-Nakase4,5, Masashi Ueda3,6, Riccardo Vago2,7, Shiroh Futaki8, Arwyn T. Jones9, Ikuhiko Nakase1 (1. Graduate School of Science, Osaka Prefecture University, 2. IRCCS San Raffaele Hospital, 3. College of Pharmacy, Okayama University, 4. Mukogawa Women’s University, 5. Institute for Biosciences, Mukogawa Women’s University, 6. Graduate School of Medicine, Dentistry, and Pharmaceutical Sciences, Okayama University, 7. University Vita-Salute San Raffaele, 8. Institute for Chemical Research, Kyoto University, 9. Cardiff University)
11:48 AM - 12:00 PM JST(2:48 AM - 3:00 AM UTC)

[27V03-am14]Development of photo-caged compounds to induce intracellular oxidative stress

○Mieko Tsuji1, Tatsuya Aoki1, Haruno Taira1, Susumu Namiki1, Tasuku Hirayama1, Hideko Nagasawa1 (1. Gifu Pharm. Univ.)
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