Session Details
[28P01]その他の合成
Sun. Mar 28, 2021 9:00 AM - 6:00 PM JST
Sun. Mar 28, 2021 12:00 AM - 9:00 AM UTC
Sun. Mar 28, 2021 12:00 AM - 9:00 AM UTC
[Room P01] Poster Presentation Online
[28P01-001]Enantioselective Organocatalytic γ-Position-Selective Mannich Reactions of β-Ketoesters
○Venkati Bethi1, Fujie Tanaka1 (1. Okinawa Institute of Science and Technology Graduate University)
[28P01-002]Pd-catalyzed α-selective C-H arylation of pentavalent organoantimony with benzo[b]furan.
○Yuki Kitamura1, Yuki Murata1, Mizuki Iwai1, Mio Matsumura1, Shuji Yasuike1 (1. Fac. Pharm. Sci., Aichi Gakuin Univ.)
[28P01-003]Synthesis of 6-Unsubstituted 2-Aryldihydropyrimidines by Liebeskind-Srogl Cross-Coupling
○Yoshio Nishimura1, Takanori Kubo1, Ibuki Nakakita1, Yuri Nakamura1, Hidetsura Cho2 (1. Pharm., Yasuda Women's Univ., 2. Grad. Sch. Pharm. Sci., Tohoku Univ.)
[28P01-004]Synthesis of Indolyacetamides by Alkylation•Cyclization•O-Transfer Reactions
○Takumi Abe1, Kenta Noda2, Daisuke Sawada1 (1. Grad. Sch. Pharm., Okayama Univ., 2. Fac. Pharm., Okayama Univ.)
[28P01-005]Annulation via dynamic aldol-oxa-cyclization to construct spirooxindole pyran polycycles
○Muhammad Sohail1, Fujie Tanaka1 (1. Okinawa Institute of Science and Technology Graduate University)
[28P01-006S]Organocatalytic enantioselective Mannich reactions of pyruvates as nucleophiles
○Santanu Mondal1, Fujie Tanaka1 (1. Okinawa Institute of Science and Technology Graduate University )
[28P01-007S]Novel N-alkylational method by use of carboxylic acid as alkyl source under mild condition
○Keigo Sato1, Satoru Tamura1, Aoi Sugawara1, Erika Sato1, Fuka Sato1, Shunsuke Takahashi1, Misaki Tagawa1, Tomikazu Kawano1 (1. School of Pharmacy, Iwate Medical University)
[28P01-008]Synthesis of 1,3-disubstituted isoindoline derivatives via aminalization and subsequent intramolecular aza-Michael cascade reaction
○Tetsuya Tsujihara1, Mizuki Fukkoshi1, Sae Hatakeyama1, Hazuki Yamauchi1, Satoru Tamura1, Tsunayoshi Tekehara2, Takeyuki Suzuki2, Tomikazu Kawano1 (1. Sch. Pharm., Iwate Medical Univ., 2. ISIR, Osaka Univ.)
[28P01-009]Oxidation of isochromans by an electronically tuned nitroxyl radical catalyst
○Shohei Hamada1, Kyoko Yano1, Elghareeb. E. Elboray1, Yusuke Kobayashi1, Takeo Kawabata2, Takumi Furuta1 (1. Kyoto Pharmaceutical Univ., 2. Institute for Chemical Research, Kyoto Univ.)
[28P01-010S]Oxidative deprotection of benzyl-type protecting groups by a nitroxyl radical catalyst
○Maiko Sumida1, Shohei Hamada1, Koichi Sugimoto1, Takeo Kawabata2, Takumi Furuta1 (1. Kyoto Pharmaceutical Univ., 2. ICR, Kyoto Univ.)
[28P01-011S]Development of Synthesis of β,γ-Subsituted-γ-butyrolactones Using Hypervalent Iodine and Nucleophile
○Takuya Matsumoto1, Hiroki Iwasaki1, Masayuki Yamashita1, Naoto Kojima1 (1. Kyoto Pharm. Univ.)
[28P01-012S]The development of one-pot reaction for the synthesis of isoquinoline via isoquinoline N-oxide as reactive intermediate
○Riho Takemi1, Hiroki Iwasaki1, Yumiko Uemura1, Yuna Tsujitani1, Naoto Kojima1, Masayuki Yamashita1 (1. Kyoto Pharmaceutical Univ.)
[28P01-013]Synthesis of N-aminoammonium salts by electrophilic amination of strong organic bases
○Takanari Arai1, Hikaru Fujita1, Munetaka Kunishima1 (1. Faculty of Pharmaceutical Sciences, Institute of Medical, Pharmaceutical, and Health Sciences, Kanazawa University)
[28P01-014]N-Allenylphthalimides as precursors of substituted isoxazoles
○Noriko Okamoto1, Reiko Yanada1, Takuya Sueda1 (1. Hiroshima International University)
[28P01-015]Study on oxone-mediated esterification of aldehydes using tivalent indium reagents
○Tomoko Mineno1, Azusa Sato1, Saika Komiya1 (1. Takasaki Univ. Health Welfare)
[28P01-016]Benzylation reaction of alcohols using alkyl acetimidate activation by gold(I) catalyst
Shintaro Ban1, Tomotake Endo1, Rikako Matsui1, Nobuyoshi Morita1, ○Yoshimitsu Hashimoto1, Kosaku Tanaka III1, Osamu Tamura1 (1. Showa Pharmaceutical University)
[28P01-017]Gold-catalyzed synthesis of 2,3-trans-dihydrobenzofurans in ionic liquid
○Nobuyoshi Morita1, Kanae Ikeda1, Hitomi Chiaki1, Ryuto Araki1, Kosaku III Tanaka1, Yoshimitsu Hashimoto1, Osamu Tamura1 (1. Showa Pharmaceutical University)
[28P01-018]The Pauson-Khand reaction of 1-alkynyl-4-methylenecyclohexanol derivatives
○Yuri Iso1, Koji Ikeda1, Hiroshi Nakamura1, Miyuki Ishizaki1 (1. Fac. Pharm. Sci, Josai International Univ.)
[28P01-019S]Reductive indole synthesis accompanied with N-N bond and cyclopropane cleavage via [3, 3]-sigmatropic rearrangement
○Hiroki Fujioka1, Motohiro Yasui1, Norihiko Takeda1, Masafumi Ueda1 (1. Kobe Pharm. Univ.)
[28P01-020S]Development of alkylated 1,2,4-triazole synthesis utilizing the C-nucleophilicity of hydrazones
○Haruo Matsuzaki1, Norihiko Takeda1, Mayuko Okazaki1, Seishin Suzuki1, Motohiro Yasui1, Masafumi Ueda1 (1. Kobe Pharmaceutical University)
[28P01-021]6-Chloro-2-pyridone as an efficient catalyst for ester aminolysis
○Takeshi Yamada1, Yusuke Watanabe1, Sentaro Okamoto1 (1. Dept. Mater. Life Chem., Kanagawa Univ.)
[28P01-022S]Oxidation of Allylic and Benzylic Alcohol with Lindlar Catalyst under Hydrogen Atmosphere
○Namika Atsumi1, Naoto Okutomi1, Shogo Kamo1, Shinya Adachi1, Akinobu Matsuzawa1, Kazuyuki Sugita1 (1. Hoshi University)
[28P01-023]Development of a synthetic method for 1,1-difluoroethyl ethers with Halothane
○Yukiko Karuo1, Ayaka Kametani1, Atsushi Tarui1, Kazuyuki Sato1, Kentaro Kawai1, Masaaki Omote1 (1. Faculty of Pharmaceutical Sciences, Setsunan University)
[28P01-024S]Yb(OTf)3·nH2O accelerated cascade reaction of Krapcho decarboxylation and aldol reaction for the synthesis of α,α-difluoro-β-hydroxy ketones and its related compounds
○Yohei Yasuno1, Atsushi Tarui1, Hiroshi Shimomura1, Yukiko Karuo1, Kazuyuki Sato1, Kentaro Kawai1, Masaaki Omote1 (1. Dep. Pharm. Sci., Setsunan Univ.)
[28P01-025]One-pot synthesis of (diarylmethylene)imidazolinones
○Masahiro Ikejiri1, Atsufumi Watanabe1, Mari Katsuda1, Mayu Funakoshi1, Aki Fujisaka1, Kazuyuki Miyashita1 (1. Faculty of Pharmacy, Osaka Ohtani University)
[28P01-026S]E-selective ring-closing metathesis for i, i+4 stapled peptides
○Yui Makura1, Atsushi Ueda1, Tomohiro Umeno1, Takuma Kato2, Kazuhiro Hirayama1, Mitsunobu Doi2, Makoto Oba3, Masakazu Tanaka1 (1. Grad. Sch. Biomed. Sci., Nagasaki Univ., 2. Osaka Univ. Pharm. Sci., 3. Kyoto Pref. Univ. Med.)
[28P01-027]A concise synthetic route to flavonoids via 1,3-dipolar cycloaddition reaction
○Yuka Takahashi1, Hidetsugu Tabata1, Tetsuta Oshitari1 (1. Faculty of Pharma Sciences, Teikyo University)
[28P01-028]Studies on bi-directional nitroaldol reaction (3)
Rio Kadowaki1, Fumihiro Fukuhara1, Futaba Nakazawa1, Yusuke Akagi1, ○Toshiya Komatsu1 (1. Fac. of Pharm. Sci., Teikyo Heisei Univ.)
[28P01-029]Studies of direct arylation of 1,4-naphthoquinones
Kohei Harasawa1, Madoka Taniguchi1, ○Yusuke Akagi1, Toshiya Komatsu1 (1. Fac. Pharm. Sci., Teikyo Heisei Univ.)
[28P01-030]Asymmetric construction of optically active benzochromens via SNAr toward total synthesis of teretifolione B
Yuki Wakamiya2, ○Takuya Kumamoto1 (1. Grad. Sch. Biomed. Health Sci., Hiroshima Univ., 2. School Pharm. Sci., Hiroshima University)
[28P01-L001]One-pot preparation of the phenanthridinone derivatives from the biaryl dicarboxylic acids
○Mayu Kurokawa1, Takuya Murai1, Yongning Xing2, Elghareeb Elboray1, Syouhei Hamada1, Yusuke Kobayashi1, Takahiro Sasamori3, Takeo Kawabata2, Takumi Furuta1 (1. Department of Pharmaceutical Chemistry, Kyoto Pharmaceutical Univ., 2. ICR, Kyoto Univ., 3. Faculty of Pure and Applied Sciences, Univ. Tsukuba)