Session Details

[28P02]天然物・生体由来医薬品/薬理活性物質/その他

Sun. Mar 28, 2021 9:00 AM - 6:00 PM JST
Sun. Mar 28, 2021 12:00 AM - 9:00 AM UTC
[Room P02] Poster Presentation Online

[28P02-050S]Decomposition profile data analysis identifies unrecognized multiple effects of a natural product, Rescinnamine.

○Shumpei Nemoto1, Katsuhisa Morita1, Tadahaya Mizuno1, Hiroyuki Kusuhara1 (1. Grad. Sch. Pharm Sci., Univ of Tokyo.)

[28P02-051S]STAT3 inhibitory activity of naphthoquinones isolated from Tabebuia avellanedae

○Keita Saito1, Teruyuki Tahara1, Mitsuaki Yamashita1, Youichi Fukuda1, Akira Iida1 (1. Faculty of Agriculture, Kindai Univ.)

[28P02-052]Coffee reduces histologic and biochemical hepatic inflammation in a well characterized NAFLD mouse model

Sandra A. LaSalle1,2, Daniel Rodriguez-Agudo1,2, Kei Minowa3, Mitsuyoshi Suzuki3, William M. Pandak1,2, ○Genta Kakiyama1,2 (1. Sch. Med., Virginia Commonwealth Univ., 2. McGuire VA Med. Ctr., 3. Sch. Med., Juntendo Univ.)

[28P02-053S]Synthesis of heterocyclic rocaglamide derivatives with inhibitory activity on Ascl1 expression

○Yoshinori Makita1,2,3, Masami Ishibashi2,3, Midori A. Arai1 (1. Fac. Sci. Tech., Keio Univ., 2. Grad. Sch. Pharm. Sci., Chiba Univ., 3. Plant Mol. Sci. Cent., Chiba Univ.)

[28P02-054]Immortalized hypothalamic neurons (GT1-7 cells) by tamoxifen by geranium essential oil Toxicity enhancement mechanism

○Dai Mizuno1, Keiko Mizuno1, Masahiro Kawahara2, Kentaro Yamazaki1 (1. Faculty of Medicine, Yamagata Univ., 2. Faculty of Pharmacy, Musashino Univ.)

[28P02-055]Studies on isomerization of vitamin D3 and its related compounds in the presence of palladium catalyst

○Masayuki Morikawa1, Natsumi Kouno1, Toshie Fujishima1 (1. Faculty of Parmaceutical Sciences at Kagawa Campus Tokushima Bunri University)

[28P02-056]The mechanism of action of Brefeldin A from a fungus having HIF-1α accumulation restraint action

○Tadahiro Etoh1, Emi Watanabe1, Shou Takaki1, Karin Hashimoto1, Yongpil Kim1,2 (1. Iryo sosei Univ. Faculty of Pharmacy, 2. Iryo sosei Univ. Graduate School of Science and Engineering)

[28P02-057S]Synthesis of derivatives to modulate carboxylation activity for vitamin K-dependent proteins

○Natsuko Furukawa1, Jian-Ke Tie2, Yoshitomo Suhara1 (1. Department of Bioscience and Engneering, College of Systems Engineering and Science, Shibaura Institute of Technology, 2. Department of Biology, University of North Carolina at Chapel Hill)

[28P02-058]Purity determination of cyclophosphamide hydrate by 31P-quantitative-NMR (2)

Nahoko Uchiyama1, Junko Hosoe1, Naoki Sugimoto1, Kyoko Ishizuki1, Tatsuo Koide1, MIka Murabayashi2, Miyashita Naoto3, Kengo Kobayashi3, Yoshinori Fujimine4, Toshiyuki Yokose4, Katsuya Ofuji5, Hitoshi Shimizu5, Takashi Hasebe6, Yumi Asai6, Eri Ena6, Junko Kikuchi7, Kohei Kiyota7, Kazuhiro Fujita7, Yoshinobu Makino8, Naoko Yasobu9, Yoshiaki Iwamoto10, Toru Miura10, Koji Mizui10, Katsuo Asakura11, Takako Suematsu12, Ai Kohama13, Takashi Goto14, Masu Yasuda14, Tomohiko Ueda15, ○Yukihiro Goda1 (1. National Institute of Health Sciences, 2. Takeda Pharmaceutical Co., Ltd., 3. Daiichi Sankyo Co., Ltd., 4. Otsuka Pharmaceutical Co., 5. Chugai Pharma Manufacturing Co., Ltd., 6. Eisai Co., Ltd., 7. SHIONOGI & Co., Ltd, 8. Juzen Chemical Corp., 9. FUJIFILM Corporation, 10. FUJIFILM Wako Pure Chemical Corporation, 11. JEOL Ltd, 12. JEOL RESONANCE Inc, 13. Pharmaceutical and Medical Device Regulatory Science Society of Japan, 14. Nippon Shinyaku Co.,Ltd., 15. Sumitomo Dainippon Pharma Co., Ltd)

[28P02-059S]Fmoc synthesis and affinity evaluation of (2S,4S)-pyrrolidine PNA

○Yukari Yasutomi1, Chisato Terada2, Asako Yamayoshi2, Tsuyoshi Yamamoto2 (1. Sch. Pharm. Sci., Nagasaki Univ., 2. Grad. Sch. Pharm. Biomed Sci., Nagasaki Univ.)

[28P02-060]Development of Nano Particle Containing BSH and Cationic Polymer for Boron Neutron Capture Therapy

○Tomohiro Tanaka1, Hiroki Ueda1, Minoru Suzuki2, Yoshinori Sakurai2, Shin Aoki1,3 (1. Faculty of Pharmaceutical Sciences, Tokyo Unversity of Science, 2. Institute for Integrated Radiation and Nuclear Science, Kyoto University, 3. Research Institute for Science & Technology, Tokyo Unversity of Science)