Session Details

[26D-am]Structure-activity relationship/Structure-activity relationship

Sun. Mar 26, 2023 9:00 AM - 10:00 AM JST
Sun. Mar 26, 2023 12:00 AM - 1:00 AM UTC
[Room D] Institute for the Advancement of Higher Education: S2 Bldg. S: 2F
Chair: Naohisa Ogo, Hideaki Fujii

[26D-am01S]Development of PKC activators for HIV cure

○Takahiro Ishii1, Takuya Kobayakawa1, Kouki Matsuda2, Kohei Tsuji1, Kazuhisa Yoshimura3, Hiroaki Mitsuya2,4,5, Kenji Maeda6, Hirokazu Tamamura1 (1. Inst. Biomater. Bioeng., Tokyo Med. Dent. Univ., 2. Natl. Cnr. Glob. Health Med. Res. Inst., 3. Tokyo Metro. Inst. Pub. Health, 4. Natl. Cancer Inst., Natl. Inst. Health, 5. Kumamoto Univ. Hosp., 6. Joint Res. Cnr. Human Retrovirus Infection, Kagoshima Univ.)

[26D-am02S]Structure-Activity Relationship Study of Flavonol Derivatives for Salt-Inducible Kinase

○Yoshiaki Takayama1,2, Tomoya Sugai2, Kei Nishida2,3, Yukiko Ishikawa2, Takeshi Kanda2, Masashi Yanagisawa2,3, Noriki Kutsumura1,2,3 (1. Degree Programs in Pure and Applied Sciences, University of Tsukuba, 2. WPI-IIIS, University of Tsukuba, 3. Ph.D. Program in Humanics, University of Tsukuba)

[26D-am03S]Development of a Novel Salt-Inducible Kinase Activator

○Hiroki Uchiyama1,2, Tomoya Sugai2, Kei Nishida2,3, Yukiko Ishikawa2, Takeshi Kanda2, Masashi Yanagisawa2,3, Noriki Kutsumura1,2,3 (1. Degree Programs in Pure and Applied Sciences, University of Tsukuba, 2. IIIS, University of Tsukuba, 3. Ph.D. Program in Humanics, University of Tsukuba)

[26D-am04S]Design and Synthesis of 2,4,5-Trisubstituted Pyrimidine-centred Kinase Inhibitors

○Ruburika Nagao1,2, Tomoya Sugai2, Kei Nishida2,3, Yukiko Ishikawa2, Takeshi Kanda2, Masashi Yanagisawa2,3, Noriki Kutsumura1,2,3 (1. Degree Program in Pure and Applied Sciences, University of Tsukuba, 2. IIIS, University of Tsukuba, 3. Ph.D. Programs in Humanics, University of Tsukuba)

[26D-am05S]Functional analysis of novel inhibitor for downstream targeting of TGF-β signaling to suppress EMT

○tsugumasa toma1, Hiroshi Tateishi1, Kensaku kawakami2, Yuta Nakashima2, Mikako Fujita1, Masami Otsuka1,3 (1. Grad. Sch. Pharm. Sci., Kumamoto Univ., 2. Grad. Sch. Sci. Tech., Kumamoto Univ., 3. Science Farm Ltd)