The 143rd Annual Meeting of the Pharmaceutical Society of Japan (Sapporo)
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Session Details

Poster Presentation(A) Pharmaceutical Chemistry

[26P1-am1]Chemical reactions/Reaction mechanism/Structure and physical property/Molecular recognition/Others

Sun. Mar 26, 2023 10:00 AM - 11:40 AM JST
Sun. Mar 26, 2023 1:00 AM - 2:40 AM UTC
[Room P1] Gymnasium 1F

[26P1-am1-001S]Synthesis of substituted pyrrolidines by gold-catalyzed cascade ring opening-cyclization of alkynylazetidines

○TOYA KARIYA1, Hiroto Yuraki1, Masahumi Hayashi1, Tsukasa Hirokane1, Masahiro Yoshida1 (1. Fac. Pharm. Sci., Tokushima Bunri Univ.)

[26P1-am1-002S]Synthesis of [3.1.0]bicyclolactum using iron chloride

○Yuuki IMOTO1,3, Eito YOSHIOKA1,2, Tomohiro YOSHIKAWA2, Tomoko IKEDA2, Ichiro YAMASAKI2, Ryousuke TANAKA2, Hiroki TAKAHASHI1, Naoki HAYASHI2, Hideto MIYABE1,2 (1. Grad. Sch. Pharm., Hyogo Medical University, 2. Sch. Pharm., Hyogo Medical University, 3. Department of Pharmacy, Shiga Prefectural General Hospital)

[26P1-am1-003]The Development of Bismuth-catalyzed Oxidative Cross Coupling Reaction with 3-Hydroxycarbazoles and Aryls

○KENGO KASAMA1, Yuta Koike1, Takayuki Yakura1 (1. University of Toyama)

[26P1-am1-004S]Synthesis of optically active allenes by asymmetric isomerization of aryl propargyl ethers and application to a synthesis of optically active benzofuran derivatives

○Tsuyoshi Kakihara1, Takuya Hirabayashi1, Shinya Minato1, Kenji Matsumoto1, Masahiro Yoshida1 (1. Fac. Pharm. Sci., Tokushima Bunri Univ.)

[26P1-am1-005S]E-Selective synthesis of stapled peptides by using achiral four-membered ring amino acids

○makura yui1, ueda atsushi 1, hisada naoyuki 2, hirayama kazuhiro1, tanaka masakazu1 (1. Grad. Sch. Biomed. Sci., Nagasaki Univ., 2. Sch. Pharm. Sci., Nagasaki Univ.)

[26P1-am1-006]Asymmetric reactions using N-terminal modified helical peptide-catalysts

○Kazuki Satou1, Tomohiro Umeno1, Atsushi Ueda1, Mitsunobu Doi2, Takuma Katou2, Masakazu Tanaka1 (1. Grad. Sch. Biomed. Sci., 2. Fac. Pharm., Osaka Med. Pharm. Univ.)

[26P1-am1-007]Dual functionalization of N-terminus by metal-mediated aldol reaction and Pictet-Spengler reaction

○Kengo Hanaya1, Yuki Morimi1, Kazuaki Taguchi1, Kazuaki Matsumoto1, Shuhei Higashibayashi1, Takeshi Sugai1 (1. Faculty of Pharmacy, Keio University)

[26P1-am1-008]Iron-catalyzed C-H amination of tyrosine derivatives

○Takahiro Yamada1 (1. Showa Pharmaceutical University)

[26P1-am1-009S]Development of asymmetric cyclopropanation using helical peptides as organocatalysts.

○Akihiro Iyoshi1, Atsushi Ueda1, Kazuki Sato1, Masakazu Tanaka1 (1. Grad. Sch. Biomed. Sci., Nagasaki Univ)

[26P1-am1-010]Concise synthesis and application to 2,5-diketopiperazines based on catalytic peptide bond formation

○Masayoshi Koshizuka1, Kaito Shinoda1, Kazuishi Makino1, Naoyuki Shimada2 (1. Department of Pharmaceutical Sciences, Kitasato University, 2. Department of Chemistry, Nihon University)

[26P1-am1-011S]6-Step total synthesis of quercetin glycosides using boronic acid-catalyzed site-selective acylations

○Shinnosuke Nakagawa1, Yuuki Nakamura2, Naoya Takahasi2, Kazuishi Makino2, Naoyuki Shimada1 (1. Department of Chemistry, Nihon Univercity , 2. Department of Pharmaceutical Sciences, Kitasato Univercity )

[26P1-am1-012S]Development of Glucuronidation Reaction by using Methyl 1,2,3,4-Tetra-O-acetyl-D-glucuronate as a Glycosyl Donor

○Tianqi DU1, Kimiyoshi Kaneko2, Yuki Sakai1, Masato Tsunoi1, Tenchi Yoshitake1, Aki Kotera1, Yasuyuki Matsushima3, Tsuyoshi Miura3, Tetsuya Kajimoto1 (1. Pharm. Sci., Ritsumeikan Univ., 2. Res. Org. Sci. & Tech., Ritsumeikan Univ., 3. Pharm, Tokyo Univ. Pharm. & Life Sci.)

[26P1-am1-013]Steric Effect of Side Chain in Ring-Closing Metathesis of Ene-Ynamides

○Hideaki Wakamatsu1, Mizuki Sato1, Yuichi Yoshimura1 (1. Fac. Pharm. Sci., Tohoku Medical and Pharmaceutical Univ.)

[26P1-am1-014S]PNP pincer acridine ligand enabling visible light-induced transition metal catalyzed reaction.

○Yu Matsuda1, Masaya Nakajima1, Tetsuhiro Nemoto1 (1. Grad. Sch. Pharm. Sci., Chiba Univ.)

[26P1-am1-015]Ruthenium-catalyzed construction of aminovinylcyclopropane scaffold from ynamide and ethylene

○Masanori Tayu1, Mizuki Masutani1, Misa Ejima1, Sayaka Ohrui1, Keiichi Saito2, Yoshihiro Sato2, Nozomi Saito1 (1. Meiji Pharm. Univ., 2. Fac. Pharm. Sci., Hokkaido Univ.)

[26P1-am1-016S]Development of nickel catalyzed cycloaddition reaction of 2,3-bis-silylcyclopropanone and 1,6-diyne

○Yuki Sato1, Satoshi Yagi1, Sayaka Ohrui1, Masanori Tayu1, Nozomi Saito1 (1. Meiji Pharm. Univ.)

[26P1-am1-017S]Development of rhodium-catalyzed Ullmann-type coupling reaction.

○satoki teranishi1, kazuyuki sato1, masaaki omote1, atsushi tarui1, yukiko karuo1, kentaro kawai1 (1. Setsunan Univ. Pharm Sciences, Med. Chem. Lab.)

[26P1-am1-018]Regioselective Epoxidation of Olefins Using Fluorous Fe(III) Salen Complex and Air

○Yamato Kato1, Kazuki Ishihara1, Takayuki Shioiri1, Masato Matsugi1 (1. Grad. Sch. Agri., Meijo Univ.)

[26P1-am1-019S]Bridging ligands library construction in chiral paddle-wheel diruthenium catalysts

○Kohei Mori1, Kotoko Makino1, Shoichi Kiryu2, Yuhei Kumagai2, Taku Miyazawa2, Tatsuhiko Yoshino2,3, Masahiro Kojima2, Shigeki Matsunaga2,3 (1. Fac. Pharm. Sci., Hokkaido Univ., 2. Grad. Sch. Pharm. Sci., Hokkaido Univ, 3. GI-CoRE)

[26P1-am1-020S]Development of highly enantioselective Henry reaction of trifluoromethyl enones using organocatalysts.

○Ryo Tsuyusaki1, Miki Shimomura1, Masahiro Kawada1, Kosuke Nakashima1, Yasuyuki Matsushima1, Shin-ichi Hirashima1, Tsuyoshi Miura1 (1. Tokyo University of Pharmacy and Life Sciences)

[26P1-am1-021S]Preparation of alkylslufonium salts and their application to C-C bond formation

○shunsuke nakamura1, kai yamamoto1, airi takagi1, haruma abe1, haruka naruse1, motoki ito1, kazuhiro higuchi1, shigeo sugiyama1 (1. Meiji Pharmaceutical University)

[26P1-am1-022S]Hetero Cope-type hydroamination reaction with isocyanate

○Ayaka Yamamoto1, Ryo Makita1, Kosaku Tanaka,Ⅲ1, Yoshimitsu Hashimoto1, Nobuyoshi Morita1, Osamu Tamura1 (1. Showa Pharm. Univ.)

[26P1-am1-023S]Cyclization of 2-alkynylaryl-H-phosphinates

○Kengo Ayabe1, Ryoji Nozawa1, Makoto Tatamiya1, Makoto Tatamiya1,2, Takehiro Yamagishi1,2 (1. Dept. of Med. Chem., Hokkaido University of Science, 2. CRILS)

[26P1-am1-024S]Enantioselective desymmetrization of meso-aziridines with chalcogen phosphinic acids

○Ryo Fujino1, Shin-ichi Hiashima1, Tomoka Iki1, Takuki Baba1, Naoki Noda1, Yasuyuki Matsushima1, Kosuke Nakashima1, Tsuyoshi Miura1 (1. Tokyo University of Pharmacy and Life Sciences)

[26P1-am1-025S]One-pot asymmetric synthesis of stilbene oxide via desymmetrical monosulfonylation of meso-hydrobenzoin directed to the synthesis of multivalent chiral amines

Kenji Yatsuzuka1, ○Shiori Fukuoka1, Seine Nakano1, Akari Shimmoto1, Midori Kawasaki2, Ryuichi Shirai2 (1. Fac. Pharm. Sci., Doshisha Women's Col., 2. Grad. Sch. Pharm. Sci., Doshisha Women's Col.)

[26P1-am1-026]Asymmetric Luche reduction of optically active 2-(Arylsulfinyl)phenyl ketones

○Toshinori Nakakita1, Karin Shigematsu2, Yoshinori Okuno1, Yasuo Sato1, Masashi Asai1, Yasuhito Nobushi2, Masaharu Toriyama2, Kouwa Yamashita1, Motofumi Miura2 (1. YOKOHAMA UNIVERSITY OF PHARMACY, 2. SCHOOL OF PHARMACY. NIHON UNIVERSITY)

[26P1-am1-027]A Facile Preparation of Silylacetals via Anodic Oxidation of 2-Silyl-1,3-dithianes

○Masahiro Noji1, Sho Ishimaru1, Haruki Obata1, Ayano Kumaki1, Taichi Seki1, Satoshi Hayashi1, Toshikatsu Takanami1 (1. Meiji Pharmaceutical University)

[26P1-am1-028S]Photocatalytic deuteration of sulfur-containing organic substrates

○Miyu Mae1, Riku Ogasahara1, Shuji Akai1, Yoshinari Sawama1 (1. Osaka univ.)

[26P1-am1-029]Trifluoromethylthiolation of alfa bromoamides with nucleophilic trifluoromethylthiolating reagents

○Satoshi Mizuta1, Masahiro Tabira2, Yuki Morii1, Jun Ishihara1, Takeshi Ishikawa2 (1. Grad. Sch. Biomed. Sci., Nagasaki Univ., 2. Grad. Sch. Sci. Eng., Kagoshima Univ.)

[26P1-am1-030]Synthesis of Carbamoyl Azides via Lossen Rearrangement Utilizing DPPA

Kotaro Ishihara1, ○Yota Tanaka1, Kazuki Ishihara1, Takayuki Shioiri1, Masato Matsugi1 (1. Grad. Sch. Agri., Meijo Univ.)

[26P1-am1-031S]Photocatalytic Decoration of Simple Alkanes by Superacidic Carbon Acid Functionality

Shoki Hoshikawa1, ○Rikuto Fujimoto1, Takashi Matsumoto1, Hikaru Yanai1 (1. Tokyo Univ. Pharm. Life Sci.)

[26P1-am1-032S]Asymmetric construction of chiral phosphorous center by using chiral sulfonamide

○Mizuki Nakamoto1, Miku Murata1, Yurika Kambara1, Ayase Matsumoto1, Aya Sakaki1, Akari Miyawaki1, Junpei Matsuoka1, Yasutomo Yamamoto1 (1. Doshisha Women's College of Liberal Arts)

[26P1-am1-033S]Inverse-electron-demand Diels–Alder reactions of α,β-unsaturated hydrazones with methyl coumalate

○Yuki Maeda1, Kyoka Inoue1, Yoshimitsu Hashimoto1, Kosaku Tanaka III1, Nobuyoshi Morita1, Osamu Tamura1 (1. Showa Pharm. Univ)

[26P1-am1-034S]Cp*Rh(III)/chiral carboxylic acid-catalyzed enantioselective synthesis of thiazin-1-imines via catalytic C–H activation

○Yuta Kitakawa1, Kodai Yamada2, Futa Kamiyama2, LongTao Huang2, Masahiro Kojima2, Tatsuhiko Yoshino2,3, Shigeki Matsunaga2,3 (1. Fac. Pharm. Sci., Hokkaido Univ., 2. Grad. Sch. Pharm. Sci., Hokkaido Univ., 3. GI-CoRE GSD, Hokkaido Univ.)

[26P1-am1-035S]Development of Reagent Converted into Hydrodisulfide under Acidic Condition

○Masaki Kobayashi1, Mako Nishigaki1, Tsubasa Inokuma1, Ken-ichi Yamada1 (1. FAC. Pharm. Sci. Tokushima Univ.)

[26P1-am1-036]Synthesis of fluorinated dihydropyrido[1,2-a]indolones facilitated by fluorinative cyclohexanedione ring-opening reaction

○Hirotaka Sasa1, Hideyasu China2, Yusuke Yoto1, Kotaro Kikushima1, Toshifumi Dohi1 (1. College of Pharmaceutical Sciences, Ritsumeikan University, 2. Faculty of Bioscience, Nagahama Institute of Bio-Science and Technology)

[26P1-am1-037]N-Heterocyclic carbene catalyzed cross dehydrogenative coupling of aldehydes with methanol: Combined use of eosin Y and hexachloroethane

○Eito YOSHIOKA1,2, Hiroki TAKAHASHI1, Akane KUBO2, Miki OHNO2, Fuuka WATANABE2, Rino SHIONO2, Yuuki MIYAZAKI2, Hideto MIYABE1,2 (1. Grad. Sch. Pharm., Hyogo Medical University, 2. Sch. Pharm., Hyogo Medical University)

[26P1-am1-038S]Ring formation of acetylene derivatives in water

○Hina Ishimaru1, Ayano Suzuki1, Yoshinori Okuno1, Shigeki Isomura1, Yasuo Sato1 (1. Yokohama University of Pharmacy)

[26P1-am1-039]Synthesis of boronic acid derivatives TDBFB for F-18 indirect labeling using Suzuki coupling

○Yusuke Yagi1,2,3,4, Hiroyuki Kimura2, Takahiro Higuchi3,4,5 (1. Kyoto College of Medical Science, Faculty of Medical Science, Department of Radiological Technology, 2. Grad. Sch. Pharm. Sci., Kyoto Pharmaceutical Univ., 3. Department of Nuclear Medicine, University Hospital Würzburg, 4. Comprehensive Heart Failure Center, University Hospital of Würzburg, 5. Grad. Sch. Med. Dent. Pharm. Sci., Okayama Univ.)

[26P1-am1-040]Catalytic oxidation of aromaric aldehydes and benzyl alcohols without adding of water

○Yasunari Monguchi1, Yuka Yamasaki1, Minami Moriuchi1, Yui Higashikayama1, Taiga Komura1, Kazutaka Koga1, Sayuri Yokoyama1 (1. Daiichi University of Pharmacy)

[26P1-am1-041S]Environmentally benign intramolecular HAT hydroarylation of alkenes by the merger of photoredox and cobalt catalysis

○Yuto Yamaguchi1, Yusuke Seino1, Akihiko Suzuki1, Yuji Kamei1, Tatsuhiko Yoshino1,2, Masahiro Kojima1, Shigeki Matsunaga1,2 (1. Grad. Sch. Pharm. Sci., Hokkaido Univ., 2. GI-CoRE)

[26P1-am1-042S]Synthesis of chiral indane derivatives using Michael-Michael domino reaction of nitroalkanes to o-substituted nitrostyrenes catalyzed by planar chiral bisthiourea

○Kaho Ishida1, Naohiro Kojima1, Shun Yoshioka1, Yukino Morita1, Keisuke Yoshida1, Shinji Kitagaki1 (1. meijo university)

[26P1-am1-043S]Development of catalytic regioselective halo-phosphorylation of epoxides by using 4-methylpyridine N-oxide

○Yuka Kimura1, Mima Nitta1, Keisuke Yoshida1, Shinji Kitagaki1 (1. Meijo university)

[26P1-am1-044S]Amine-free O-phosphorylation of alcohols by using 4-methylpyridine N-oxide

○Wataru Hirano1, Keisuke Yoshida1, Shinji Kitagaki1 (1. Meijo university)

[26P1-am1-045S]Synthesis of alpha-amino acid derivatives bearing beta-sulfonyl group

Yusuke Kobayashi1, ○Yuta Ishimoto1, kaori motoki1, takuma kinsho1, nana suzuki1, shohei hamada1, takumi furuta1 (1. Fac. Pharm., Kyoto Pharmaceutical University)

[26P1-am1-046S]Synthesis and property of hypervalent pnictogen compound-Brønsted acid complex

○Nagisa Ishida1, Yuuki Nishida1, Shohei Hamada1, Takumi Furuta1, Yusuke Kobayashi1 (1. Fac. Pharm., Kyoto Pharmaceutical University)

[26P1-am1-047]Synthesis of sialidase inhibitors for aiming to development of anti-diabetic drugs (2)

○Kiyoshi Ikeda1, Masahiro Tanaka1, Naoya Shibao1, Kazu Koyama2, Akira Minami2, Tomoya Hikita3, Yuuki Kurebayashi2, Tadanobu Takahashi2, Hideyuki Takeuchi2, Takashi Suzuki2, Fumiteru Teraoka1, Tadamune Otsubo1 (1. Dep. Pharm. Sci., Hiroshima International Univ., 2. Sch. Pharm. Sci., Univ. of Shizuoka, 3. Aichi Cancer Center Research Insti.)

[26P1-am1-048]Synthetic study of sulfate monosaccharide anti-dengue virus drug (3)

○fumiteru teraoka1, Takahiro Osaki1, Utsubo Chie2, kazuya hidari3, tadamune otsubo1, Kiyoshi Ikeda1 (1. Pharmaceutical Sci., Hiroshima International Univ., 2. Grad. Sch. Health Sci., Kobe Univ., 3. Sch. Food and Nutririon. Sci., Aizu Jnr. Coll.)

[26P1-am1-049]Design and synthesis of a novel selective fluorescence sialidase probe

○tadamune otsubo1, Hiroto Ueda1, Daiki Syuto1, Yutaka Narimichi2, Tadanobu Takahashi2, Yuuki Kurebayashi2, Akira Minami2, Fumiteru Teraoka1, Hideyuki Takeuchi2, Kiyoshi Ikeda1 (1. Dept. Pharm. Sci., Hiroshima International Univ., 2. Sch. Pharm. Sci., Univ. Shizuoka)

[26P1-am1-050S]Development of catalytic enantioselective aza-Henry reaction utilizing stereo-characteristics of aromatic layered ureas

○Mamika Ogura1, Mayumi Kudo2, Tatsuya Orihara3, Minami Odagi3, Kazuo Nagasawa3, Aya Tanatani1 (1. Grad. Sch. Adv. Sci., Ochanomizu Univ., 2. NIT Gunma College, 3. Department of Biotechnology, Tokyo University of Agriculture & Technology)
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