The 143rd Annual Meeting of the Pharmaceutical Society of Japan (Sapporo)
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Session Details

Poster Presentation(A) Pharmaceutical Chemistry

[26P1-pm2]Total synthesis/Biosynthesis/Other synthetic studies

Sun. Mar 26, 2023 3:50 PM - 5:30 PM JST
Sun. Mar 26, 2023 6:50 AM - 8:30 AM UTC
[Room P1] Gymnasium 1F

[26P1-pm2-001]Synthesis of fluorescence-labeled thallusin derivatives and their effects on zoospores of green alga Gayralia

○Momoka Takahashi1, Naoto Yamasaki1, Masaya Takehara1, Tomoyuki Esumi1, Hiromichi Kennmoku1, Yoshinori Asakawa1, Hirohumi Yamamoto1 (1. Pharm. Sci., Tokushima bunri Univ.)

[26P1-pm2-002S]Development of N-fluoroalkylation for various nitrogen-containing heterocycles

○Yukari Akamatsu1, Kohei Hamayasu1, Yukiko Karuo1, Atsushi Tarui1, Kazuyuki Sato1, Kentaro Kawai1, Masaaki Omote1 (1. Faculty of Pharmaceutical Sciences, Setsunan University)

[26P1-pm2-003S]Synthetic study of indole-pyrazole type bi-heteroaryl compounds under the common Suzuki coupling conditions

○Natsuki Honda1, Takuya Okawauchi1, Ryota Fujimoto1, Noriyuki Nakajima1,2, Yasuhito Koyama1,2, Masahiro Hamada1,2 (1. Toyama Prefectural University, 2. Biotech. Res. Center, Toyama Pref. Univ.)

[26P1-pm2-004]A concise synthetic route to nobiletin

○Yuka Takahashi1, Hidetsugu Tabata1, Tetsuta Oshitari1 (1. Faculty of Pharma Sciences, Teikyo University)

[26P1-pm2-005S]Synthetic study of specific inhibitors toward a peptide epimerase MurL

○Takumi Yamaoka1, Fumihiro Isikawa1, Yasushi Ogasawara2, Tohru Dairi2, Genzoh Tanabe1 (1. Faculty of Pharmacy, Kindai University, 2. Graduate School of Engineering, Hokkaido University)

[26P1-pm2-006]Synthesis of antitumor cyclic hexapeptide RA-VII analogues with an aromatic amino acid at position 2. Part II.

○Motoki Katoh1, Keiichiro Ogura1, Tomoyo Hasuda1, Haruhiko Fukaya1, Yukio Hitotsuyanagi1 (1. Tokyo Univ. of Pharm. & Life Sci., Sch. of Pharm.)

[26P1-pm2-007S]Evaluation of H-bonding Ability of Chloroalkene Dipeptide Isosteres Using Peptide Catalyst System

○Chihiro Iio1, Fujimoto Junko2, Toyama Daichi1, Sato Kohei1,2, mase Nobuyuki1,2, Narumi Tetsuo1,2 (1. Grad. Sch. Integ. Sci. Tech., Shizuoka Univ., 2. Fac. Eng., Shizuoka Univ.)

[26P1-pm2-008S]Synthesis of amide-to-fluoroalkene peptidomimetic of
Aβ-derived peptide containing Phe-Phe-type fluoroalkene dipeptide isostere

○Ai Sakakibara1, Chihiro Iio2, Kohei Sato1,2, Nobuyuki Mase1,2, Tetsuo Narumi1,2 (1. Fac. Eng., Shizuoka Univ., 2. Grad. Sch. Integ. Sci. Tech., Shizuoka Univ.)

[26P1-pm2-009]Synthesis of a disaccharide, Emmyguyacins B, containing anti influenza virus.

○Isao Ohtsuka1, Toshiyuki Atsumi1 (1. Kyushu University Health and Welfare)

[26P1-pm2-010]Effects of sulfated vizantin based on docking simulation analysis

○Yui Asano1, Naoto Yamasaki1, Hironobu Takahashi1, Tomoyuki Esumi, Kenmoku Hiromichi1, Yoshinori Asakawa1, Hirofumi Yamamoto1 (1. Facalty of Pharmaceutical Science, Tokushima Bunri University)

[26P1-pm2-011S]Efforts toward Synthesis of Pericosine E Analogs Bearing A Halogen Atom Other Than Chlorine

○Keika Miyamoto1, Saya Atarashi1, Arisa Nomura1, Yoshihiro Uesawa2, Noboru Hayama1, Hiroki Yoneyama1, Yoshihide Usami1 (1. Fac. Pharm., Osaka Med. Pharm. Univ., 2. Meiji Pharm. Univ.)

[26P1-pm2-012]Synthetic study of C-linked trehalose analogues

Rintaro Nakahashi1, Takahiro Moriyama1, ○Hiroaki Matoba1, Makoto Yoritate1, Go Hirai1 (1. Grad. Sch. Pharm. Sci., Kyushu Univ.)

[26P1-pm2-013]Synthesis of novel entecavir analogues having cyano group and fluorine; Evaluation of their anti-HBV activity

○HIROKI KUMAMOTO1, Nobuyo Kuwata Higashi2, Sanae Hayashi3, Debananda Das4, Haydar Bulut4, Ryoh Tokuda5, Shukei Imoto5, Kengo Onitsuka2, Yuka Honda6, Yuki Odanaka6, Satoko Matsubayashi Shinnbara6, Kazuhiro Haraguchi1, Yasuhito Tanaka3, Hiroaki Mitsuya2,4 (1. Department of Pharmaceutical Sciences, Nihon Pharmaceutical University, 2. NCGM, 3. Kumamoto University, 4. NIH, 5. Sojo University, 6. Showa University)

[26P1-pm2-014S]Photoracemization of chiral sulfoxides by using photocatalysts

○Saki Fukushima1, Kumi Tozawa1, Kosho Makino2, Kayo Nakamura1, Hidetsugu Tabata3, Tetsuta Oshitari3, Hideaki Natsugari4, Hideyo Takahashi1 (1. Pharm.Sci., Tokyo University of Science., 2. Pharm.Sci., Musashino Univ., 3. Pharm.Sci., Teikyo Univ., 4. Pharm.Sci., Tokyo Univ.)

[26P1-pm2-015S]Development of a synthesis method for various fluoroalkenes using Suzuki-Miyaura cross-coupling

○Keita Hirata1, Yukiko Karuo1, Atushi Tarui1, Kazuyuki Sato1, Kentaro Kawai1, Masaaki Omote1 (1. Faculty of Pharmaceutical Sciences, Setsunan University)

[26P1-pm2-016]Synthesis of optically pure erythro-2-amino-1,2-bis(4-methoxyphenyl)ethan-1-ol via Lipase TL-mediated kinetic resolution of anisoin

○Saya Okumura1, Monami Tsukamoto1, Yukiko Otake1, Reiko Yano1, Yukio Hitotsuyanagi2, Yutaka Aoyagi1, Robert M. Williams3 (1. Coll. of Pharm., Kinjo Gakuin Univ., 2. School of Pharm., Tokyo Univ. of Pharm. and Life Sci., 3. Depart. of Chem., Colorado State Univ.)

[26P1-pm2-017]Synthesis of biosynthetic intermediates of vibrioferrin and enzymatic reactions using them as substrates

○Hidemichi Mitome1, Tomotaka Tanabe1, Tatsuya Funahashi1, Kazuki Akira1 (1. Col. Pharm. Sci., Matsuyama Univ.)

[26P1-pm2-018]A synthetic method for enyne compounds using highly halogenated alkenes

○yukiko karuo1, Atsushi Tarui1, Kazuyuki Sato1, Kentaro Kawai1, Masaaki Omote1 (1. Faculty of Pharmaceutical Sciences, Setsunan University)

[26P1-pm2-019S]Construction of successive three asymmetric carbons toward synthesis of rearranged-vibsanines

○SHINO BANDO1, KENICHI HARADA1, DAI HAMAMOTO1, MIWA KUBO1, YOSHIYASU FUKUYAMA1 (1. Tokushima Bunri University)

[26P1-pm2-020]Synthetic studies of polymers from half-esters having the norbornadiene skeleton by ring-opening metathesis polymerizations and the saturated derivatives

Xiaoxue Lin2, Jianjun Shi1,2, ○Satomi Niwayama1 (1. Grad. Sch. Eng., Muroran Institute of Technology, 2. Grad. Sch. Chem. Eng.,Hainan Normal University)

[26P1-pm2-021]Synthesis of 14β-estradiol to improve estrogen β receptor selectivity

Hinako Sato1, Takayuki Kanaya1, Noriyuki Kogure1, ○Kohei Inomata1 (1. Pharm. Sci., Int. Univ. Health and Welfare)

[26P1-pm2-022S]Synthetic study of sphingomyelinase inhibitor SMY-540 analogues.

○Mao Yamaguchi1, Shino Inishi1, Kotono Kamei1, Yusuke Kasai1, Hiroshi Imagawa1 (1. Faculty of Pharmaceutical Sciences, Tokushima Bunri University)

[26P1-pm2-023S]A short-step synthesis for optically active norbornane derivative with lactam structure

○Mayu Terauchi1, Hiroto Kaku1, Natsuki Kyan1, Natsumi Tada1, Jinuk Lee1, Yuki Ujihara1, Kei Kitamura1, Tetsuto Tsunoda1 (1. Fac. Pharm. Sci., Tokushima Bunri Univ.)

[26P1-pm2-024]Development of a synthetic method for dihydrosphingomyelin and Its application for RNA delivery

○Rina Fujihara1, Yuki Nakasaku1, Naofumi Fukata1, Kimitada Terao1 (1. nippon fine chemical co., ltd.)

[26P1-pm2-025S]Asymmetric total synthesis of β-carboline alkaloid (S)-brevicolline as antiviral agents.

○Koharu Sakoguchi1, Takashi Nishiyama1, Ryouya Shouno1, Natsumi Nakanishi1, Manami Obata1, Tominari Choshi1 (1. Fukuyama Univ.)

[26P1-pm2-026S]Total synthesis of camptothecin analogues rosettacin and synthesis of its derivatives

○Shota Mizuno1, Takashi Nishiyama1, Mai Endo1, Takaki Yoshiura1, Toshio Motoyashiki1, Noriyuki Hatae2, Tominari Choshi1 (1. Fukuyama Univ., 2. Yokohama univ. of pharm.)

[26P1-pm2-027S]Total synthesis indolo[3,2-a]carbazole alkaloid racemosin B

○Nanaka Fukada1, Takashi Nishiyama1, Yuria Takeo1, Tominari Choshi1 (1. Fukuyama University)

[26P1-pm2-028]Total synthesis of calothrixin B and its analogs.

○Takashi Nishiyama1, Yushi Yamaguchi1, Aoi Okubo1, Haruna Okihara1, Toshio Motoyashiki1, Noriyuki Hatae2, Tominari Choshi1 (1. Fukuyama Univ., 2. Yokohama univ. of pharm.)

[26P1-pm2-029S]Synthesis of novel pyridoimidazoisoquinoliniums via silver-mediated intramolecular cyclization and application for live cell imaging

○Masato Kawakubo1, Yoshikazu Inoh1, Yuki Murata1, Mio Matsumura1, Tadahide Furuno1, Shuji Yasuike1 (1. Sch. Pharm. Sci., Aichi Gakuin Univ.)

[26P1-pm2-030]Synthesis of 2-aminodibenzo[d,f][1,3]oxazepines from 2′-amino-2-hydroxybiphenyl and isothiocyanates via iodine-mediated cyclodesulfurization

○Yuki Murata1, Arisu Koyanagi1, Mako Izawa1, Yukako Hayashi2, Tadashi Hyodo2, Mio Matsumura1, Kentaro Yamaguchi2, Shuji Yasuike1 (1. Sch. Pharm. Sci., Aichi Gakuin Univ., 2. Sch. Phram Sci., Tokushima Bunri Univ.)

[26P1-pm2-031S]Synthesis of 2-arylbenzoazoles from thioamides and aminophenols via Ph3BiCl2-promoted desulfurization

○Arisu Koyanagi1, Yuki Murata1, Shiori Hayakawa1, Mio Matsumura1, Shuji Yasuike1 (1. Sch. Pharm. Sci., Aichi Gakuin Univ.)

[26P1-pm2-032]Syntehsis of 5-FU selene analog: Ag catalyzed regioselective C-H selenation of uracils

○Mio Matsumura1, Saori Tsuchida1, Rena Nezaki1, Yuki Murata1, Shuji Yasuike1 (1. Sch. Pharm. Sci., Aichi Gakuin Univ.)

[26P1-pm2-033]Synthetic Studies of Novel Heterocyclic Linking Pyrazole Derivatives based on 4-Hydroxypyrazoles

Eiichi Masumoto1, ○Saori Shindo1, Kohei Kobayashi1, Fumi Okabe-Nakahara1, Hiroshi Maruoka1 (1. Fac. Pharm. Sci., Fukuoka Univ.)

[26P1-pm2-034S]Synthetic Studies of Novel Spiro-1,3,4-Oxaziazole-Pyrazolone Derivatives

Eiichi Masumoto1, ○Kazutoshi Ihara1, Hanae Seki1, Fumi Okabe-Nakahara1, Hiroshi Maruoka1 (1. Fac. Pharm. Sci., Fukuoka Univ.)

[26P1-pm2-035]Synthetic Studies of fused tricyclic imidazo[1,2-a]pyridine derivatives.

Fumi Okabe-Nakahara1, ○Yuuna Mihara1, Eiichi Masumoto1, Hiroshi Maruoka1 (1. Fac. Pharm. Sci., Fukuoka Univ.)

[26P1-pm2-036S]Synthetic Studies of Matrine Analogues

○Hana Uemura1, Haruki Obata1, Takeshi Noda2 (1. Kanagawa Institute of Technology, 2. Kanagawa institute of technology)

[26P1-pm2-037S]Synthetic Studies of Sparteine and Anagyrine Analogues

○Daiki Arai1, Takeshi Noda2 (1. Kanagawa Institute of Technology, 2. Kanagawa institute of technology)

[26P1-pm2-038S]Synthetic Studies of New Bicyclic Pipecolic Acid Derivatives

○Masahiko Yamamoto1, Takeshi Noda2 (1. Kanagawa Institute of Technology, 2. Kanagawa institute of technology)

[26P1-pm2-039]Synthesis and properties of 4-chloropyrimidine-C-nucleoside for inhibition of DNA cytosine-5 methyltransferase (DNMT)

○Kousuke Sato1, Yuria Chiba1, Mayu Ohyama1, Takahiro Sasaki1, Tsuyoshi Murai1 (1. Sch. Pharm. Sci., Health Sci. Univ. Hokkaido)

[26P1-pm2-040]Design and synthesis of ApoB-targeted prodrug siRNA containing partial modifications for improvement of nuclease resistance

○Junsuke Hayashi1, Yosuke Ochi1, Shun-ichi Wada1, Fumito Wada2, Mariko Harada-Shiba2, Hidehito Urata1 (1. Osaka Med. and pharm. Univ., 2. National Cerebral and Cardiovascular Center)
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