The 143rd Annual Meeting of the Pharmaceutical Society of Japan (Sapporo)
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Session Details

Poster Presentation(A) Pharmaceutical Chemistry

[27P1-pm2]Total synthesis/Biosynthesis/Other synthetic studies/Chemical reactions/Reaction mechanism/Structure and physical property/Molecular recognition/Others

Mon. Mar 27, 2023 3:40 PM - 5:20 PM JST
Mon. Mar 27, 2023 6:40 AM - 8:20 AM UTC
[Room P1] Gymnasium 1F

[27P1-pm2-001S]Detection of Anionic Diastereomers of Diketopiperazines Containing Proline Residues using 13C NMR

○Yuma Fukuba1, Takashi Ishizu1 (1. Faculty of Pharmacy and Pharmaceutical Sciences , Fukuyama University)

[27P1-pm2-002S]Stereochemistry of dibenzoazepinones

○Arisa Chiba1, Mayuno Hotta1, Takuya Namba1, Kayo Nakamura1, Hidetsugu Tabata2, Kosho Makino3, Tetsuta Oshitari2, Hideaki Natsugari4, Hideyo Takahashi1 (1. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2. Faculty of Pharma Sciences, Teikyo University, 3. Faculty of Pharmacy, Musashino University, 4. Faculty of Pharmaceutical Sciences, The University of Tokyo)

[27P1-pm2-003S]Structure-activity relationship of Fentanyl derivatives

○Tsukasa Tomizawa1, Shuntaro Kikukawa1, Hironobu Arita1, Kayo Nakamura1, Kosho Makino2, Hidetsugu Tabata3, Tetsuta Oshitari3, Hideaki Natsugari4, Masahiko Funada5, Hideyo Takahashi1 (1. Pharm.Sci., Tokyo University of Science, 2. Pharm.Sci., Musashino Univ., 3. Pharm.Sci., Teikyo Univ., 4. Pharm.Sci., Tokyo Univ., 5. Pharm.Sci., Shonan Univ.)

[27P1-pm2-004S]Stereochemistry of benzodiazepines

○Ryoko Tanaka1, Kayo Nakamura1, Hidetsugu Tabata2, Kosho Makino3, Tetsuta Oshitari2, Hideaki Natsugari4, Hideyo Takahashi1 (1. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2. Faculty of Pharma Sciences, Teikyo University, 3. Faculty of Pharmacy, Musashino University, 4. Faculty of Pharmaceutical Sciences, The University of Tokyo)

[27P1-pm2-005]Construction of Biopolymer-Functional Molecule Complexes in Bioionic Media

○Kaoru Nobuoka1, Satoshi Kitaoka2 (1. Fac. Sci. Tech., Oita Univ., 2. Fac. Eng. Kindai Univ.)

[27P1-pm2-006S]Synthesis of structually defined axially chiral urea bearing a bipyridyl moiety through chalcogen-bonding interaction

○Haru Takahashi1, Rina Nakamura1, Moe Ota1, Takumi Inoue1, Takuya Murai1, Takahiro Sasamori2, Syohei Hamada1, Yusuke Kobayashi1, Takumi Furuta1 (1. Kyoto pharmaceutical university, 2. Tsukuba university)

[27P1-pm2-007S]Elaboration of indoline-2-carboxylic acid derivatives as a new chiral reagent for the recognition of chiral primary amines by 1H NMR.

○Mao Kawata1, Mashiro Nakagawa1, Risa Inatomi1, Yusuke Kasai1, Hiroshi Imagawa1 (1. Faculty of Pharmaceutical Sciences, Tokushima Bunri University)

[27P1-pm2-008S]Derivatization of amino acids by substitution of their N-methoxymethyl-N-tosylamides.

○Risa Inatomi1, Mao Yamagami1, Yusuke Kasai1, Hiroshi Imagawa1 (1. Faculty of Pharmaceutical Sciences, Tokushima Bunri University)

[27P1-pm2-009]Evaluation of the effect of the type of disubstituted amino acids on the peptide secondary structure in a heteropeptide of leucine and disubstituted amino acids

○Takuma Kato1, Yosuke Demizu2, Masakazu Tanaka3, Akiko Asano1, Mitsunobu Doi1 (1. Fac. Pharm., Osaka Med. Pharm. Univ., 2. Nat. Inst. of Health Sci., 3. Grad. Sch. Biomed. Sci., Nagasaki Univ.)

[27P1-pm2-010S]Identification and signal-assignment of deoxynojirimycin derivatives by using 1H-15N HMBC

○Hiroya Kobayashi1, Tetsuya Kajimoto1, Kimiyoshi Kaneko2 (1. Pharm. Sci., Ritsumeikan Univ., 2. Res. Org. Sci. & Tech., Ritsumeikan Univ.)

[27P1-pm2-011S]Structural Properties and conformational preferences of N-(1-azulenyl)aromatic amides

○Masayuki Yunoki1, Ai Ito1, Hirokazu Karasawa1, Marino Asato1, Yuki Asami1, Ayako Ishii1, Takamasa Amaki1, Ryu Yamasaki1, Iwao Okamoto1 (1. Showa Pharm. Univ.)

[27P1-pm2-012S]Synthesis and luminescence properties of substituted benzils

○Masamichi Yasui1, Takashi Fujihara2, Hiroyoshi Ohtsu3, Yuki Wada3, Masaki Kawano3, Kengo Hanaya1, Takeshi Sugai1, Shuhei Higashibayashi1 (1. Fac. Pharm., Keio Univ., 2. Compre. Anal. Cen. Sci., Saitama Univ., 3. Dept. Chem., Tokyo Inst. of Tech.)

[27P1-pm2-013S]Chiral supramolecule formation by heterooligomeric molecular assembly of chiral and achiral diamides

○Ichiho Tanaka1, Miu Hiraizumi1, Junpei Matsuoka1, Akari Miyawaki1, Yasutomo Yamamoto1 (1. Doshisha Women's College of Liberal Arts)

[27P1-pm2-014]Characterization of Emissive Anthyridine Derivatives with Hydrogen Bonding Ability

○Keita Ikeno1, Yasufumi Fuchi2, Kazuteru Usui1, Tomohiro Umeno1, Satoru Karasawa1 (1. Showa Pharmaceutical Uni., 2. Tokushima Bunri Uni.)

[27P1-pm2-015S]Asymmetric Recognition of Diketopiperazines containing Proline Residues using (-)-Epigallocatechin-3-O-gallate in Water

○Yuka Fujitani1, Takashi Ishizu1 (1. Faculty of Pharmacy and Pharmaceutical Sciences,Fukuyama University)

[27P1-pm2-016S]A Peptide-based Gelator for Cyclic Solvents

○Riko Sekiguchi1, Shinya Kimura1, Masashi Yokoya1, Yuiga Nakamura2, Yasuyuki Yamanada3, Masamichi Yamanaka1 (1. Meiji Pharm. Univ., 2. JASRI, 3. Nagoya Univ.)

[27P1-pm2-017]Synthesis of aminopyridine-linked purine bases for 2'-OH acetylation of RNA sugar moiety

○Jeongsu Lee1, Hirotaka Murase1, Mayuko Koga1, Fumika Tasaki1, Chika OOie1, Miharu Takakura1, Katsumi Hongo1, Yosuke Taniguchi2, Shigeki Sasaki1 (1. Grad. Sch. Pharm. Sci, Nagasaki Int. Univ. , 2. Grad. Sch. Pharm. Sci, Kyushu Univ.)

[27P1-pm2-018S]Synthesis and Evaluation of Gelation Abilities of Bis-urea Dimers to Enhance the Strength of Supramolecular Gels

○Kanon Inoue1, Kurea Adachi1, Shinya Kimura1, Masashi Yokoya1, Masamichi Yamanaka1 (1. Meiji Pharm. Univ.)

[27P1-pm2-019S]Exploration of hydrophobic cell-penetrating peptides toward efficient intracellular translocation of antisense nucleic acids

○Saki Tamura1,2, Genichirou Tsuji2, Yousuke Demizu1,2,3 (1. Grad. Sch. Med., Life Sci., Yokohama City Univ., 2. NIHS, 3. Grad. Sch. Med., Dent. & Pharm. Sci., Okayama Univ.)

[27P1-pm2-020S]Design of helical peptides for tissue-selective carriers

○Takahito Ito1,2, Takashi Misawa2, Yosuke Demizu1,2 (1. Grad. Sch. Med. Life Sci., Yokohama City Univ., 2. NIHS)

[27P1-pm2-021S]Induction of an argicyclamide analog by the cyanobacterium Microcystis aeruginosa NIES-88 through the OSMAC approach.

○Nandani Balloo1, Chin-Soon Phan2, Tatsufumi Okino1,2 (1. Graduate School of Environmental Science, Hokkaido University, 2. Faculty of Environmental Earth Science, Hokkaido University)

[27P1-pm2-022S]Synthesis of spherical amides with benzyl groups on the amide nitrogen and optical activity thereof

○Fumiko Shibata1, Daiki Koike1, Hyuma Masu2, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ., 2. CAI, Chiba Univ)

[27P1-pm2-023S]Synthesis of spherical amides with pyrenyl groups and optical activity thereof

○Emiri Karigome1, Arisa Okuda1, Daiki Koike1, Hyuma Masu2, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ., 2. CAI, Chiba Univ.)

[27P1-pm2-024S]A short step synthesis of azacoronene analogs via the cyclic trimer of dibromo-p-aminobenzoic acid

○Mariko Ninomiya1, Miho Takeno1, Sayaka Futami1, Hinata Suganuma1, Akito Miyakoshi1, Ayaka Sugiyama1, Akihiro Yokoyama2, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ., 2. Fac. Sci. Tech., Seikei Univ.)

[27P1-pm2-025S]Synthesis of functionalizable macrocyclic aromatic amides

○Ayaka Sugiyama1, Hinata Suganuma1, Sayaka Futami1, Hidemasa Hikawa1, Shoko Kikkawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)

[27P1-pm2-026S]Synthesis of cyclic oligomers of dibromo-para-aminobenzoic acid and effect of N-alkyl groups on the properties

○Akito Miyakoshi1, Sayaka Futami1, Hinata Suganuma1, Hidemasa Hikawa1, Syoko Kikkawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ)

[27P1-pm2-027S]Construction of supramolecular architectures using tetraphenyladamantane skeleton

○Sae Maeda1, Akira Tanaka1, Misaki Okayasu1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)

[27P1-pm2-028]Three-component 1,3-dipolar cycloaddition at N-Terminus of peptide

○Kazuya Kanemoto1, Haruka Machida2, Haruhiko Fuwa2 (1. Graduate School of Pharmaceutical Sciences, Tohoku University, 2. Department of Applied Chemistry, Chuo University)

[27P1-pm2-029]Silver-catalyzed 1,3-dipolar cycloaddition of azomethine ylides with dehydroalanine derivatives

○Masaki Iwata1, Kazuya Kanemoto1, Naohiko Yoshikai1 (1. Graduate School of Pharmaceutical Sciences, Tohoku University)

[27P1-pm2-030S]Investigation of desulfurative borylation at cysteine residues

○Hayato Sasamoto1, Daiki Fukue1, Taishi Ichinose1, Manaka Maeda1, Honami Matsumoto1, You Nonaka1, Tatsusada Yoshida1, Kohei Yamada1, Yasuchika Yamaguchi1 (1. Facult. Pharm. Sci., Nagasaki Int. Univ.)

[27P1-pm2-031S]Identification of a phosphorus-containing co-product in desulfurative borylation and its formation mechanisms

○Daiki Fukue1, Taishi Ichinose1, Hayato Sasamoto1, Manaka Maeda1, Honami Matsumoto1, You Nonaka1, Tatsusada Yoshida1, Kohei Yamada1, Yasuchika Yamaguchi1 (1. Facult. Pharm. Sci., Nagasaki Int. Univ.)

[27P1-pm2-032]Molecular behavior of cyclodextrin heterodimers with cross-linker containing biphenyl: the tumbling motion of modified sugar units

○Kazutaka Koga1, Kei Kitayama2, Kento Kimura2, Makoto Fukudome2, De-Qi Yuan2 (1. Fac. Pharm., Daiichi Univ. of Pharm., 2. Fac. Pharm. Sci., Kobe Gakuin Univ.)

[27P1-pm2-033]Vector-selective functionalization on the primary side of cyclodextrins via bifunctional catalysis

Tatsuro Tominaga1, Koki Fukuda1, Kazutaka Koga2, Makoto Fukudome1, ○De-Qi Yuan1 (1. Fac. Pharm. Sci., Kobe Gakuin Univ., 2. Fac. Pharm., Daiichi Univ. of Pharm.)

[27P1-pm2-034S]Gold-catalyzed cascade ring opening-cyclization reaction of alkynylcyclopropanes with anilines

○Kaede Nakazato1, Tsukasa Hirokane1, Masahiro Yoshida1 (1. Fac. Pharm. Sci., Tokushima Bunri Univ.)

[27P1-pm2-035S]Development of gold-catalyzed cascade ring opening-cyclization reaction using alkynylcyclopropanes with phenols

○Haruki Inoue1, Tsukasa Hirokane1, Masahiro Yoshida1 (1. Fac. Pharm. Sci., Tokushima Bunri Univ.)

[27P1-pm2-036]Synthesis of C2-Symmetric Bisisoquinoline Derivatives.

○Shunsuke Shimomura1, Makoto Furutachi1 (1. Fukuoka University)

[27P1-pm2-037]Flow Synthesis of Chromane Derivatives by Rearrangement Reaction

○Tetsu Tsubogo1, Fumiya Okamura2, Hiromi Uchiro2 (1. Fac. Pharm. Sci., Health Sciences Univ. of Hokkaido, 2. Fac. Pharm. Sci., Tokyo Univ. of Science)

[27P1-pm2-038]Development of highly stabilized polymeric palladium catalyst for continuous flow Suzuki-Miyaura coupling reaction

○Zhenzhong Zhang1, Aya Ohno1, Hikaru Takaya2, Yoichi M. A. Yamada1 (1. RIKEN CSRS, 2. Fac. of Life & Envir. Sci., Teikyo Univ. of Sci.)

[27P1-pm2-039]Predicting Highly Enantioselective Catalysts Using Machine Learning

○Nobuya Tsuji1, Pavel Sidorov1, Chendan Zhu2, Yuuya Nagata1, Timur Gimadiev1, Alexandre Varnek1,3, Benjamin List1,2 (1. Hokkaido University, ICReDD, 2. Max-Planck-Institut für Kohlenforschung, 3. University of Strasbourg)

[27P1-pm2-040]Novel natural compounds that control differentiation in the life cycle of Neopyropia tenera.

○Junna Ino1, Hiroto Kaku1, Naoto Yamasaki1, Tomoyuki Esumi1, Hiromiti Kennmoku1, Yoshinori Asakawa1, Hirofumi Yamamoto1 (1. Tokushima Bunri University)

[27P1-pm2-041S]Total Syntheses of Oregonensin A and Related Natural Products

○Kazuki Hori1, Shogo Kamo1, Kazuyuki Sugita1 (1. Hoshi University)

[27P1-pm2-042]Racemization study in aqueous peptide synthesis at low temperatures with continuous microwave irradiati

Nanami Shimizu1, ○Keiko Hojo1,2, Toshiki Kitagawa1, Tomoyo Uda1, Yuki Manabe1, Yuuta Ohki3, Takahiro Tanaka3, Naoyuki Takahashi3, Yuko Tsuda1,2 (1. Fac. Pharm. Sci., Kobe Gakuin Univ., 2. Ctr. Life Sci., Kobe Gakuin Univ., 3. Tokyo Rikakikai Co., Ltd)

[27P1-pm2-043S]Synthesis and α-Glucosidase Inhibitory Activity of Ribose Derived Bicyclic Pyrrolopyrazole-Iminosugars

○Kanako Yamawaki1, Hiroki Yoneyama1, Noboru Hayama1, Yoshihide Usami1 (1. Fac. Pharm., Osaka Med. Pharm. Univ.)

[27P1-pm2-044]Rapid Isomerization of Prostaglandin H2 and Related Endoperoxide Catalyzed by Thiolate-Coordinated Heme Complex and Its Derivatives

○Yuto Tsuzuki1, Tsunehiko Higuchi2, Yuuki Yano2, Takehiro Yamane2, Yosuke Hisamatsu2, Naoki Umezawa2 (1. Fac. Sch. Pharm. Sci., Nagoya City Univ., 2. Grad. Sch. Pharm. Sci., Nagoya City Univ.)

[27P1-pm2-045]Synthetic studies on 4’-thionucleoside analogue of cordycepin using ring-opening of three-membered sulfonium ion by acetate ion as a key step

○Yoshihiro Natori1, Nishi Yoshiyuki1, Watanabe Yoshiyuki1, Hideaki Wakamatsu1, Yukako Saito1, Asako Kaise1, Kentaro Yamaguchi2, Tadashi Hyodo2, Yuichi Yoshimura1 (1. Faculty of Pharmaceutical Sciences, Tohoku Medical and Pharmaceutical University, 2. Faculty of Pharmaceutical Sciences at Kagawa Campus, Tokushima Bunri University)
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