Session Details

Screening/Pharmacologically active compounds

Fri. Mar 29, 2024 4:30 PM - 5:06 PM JST
Fri. Mar 29, 2024 7:30 AM - 8:06 AM UTC
[Room 413] Conference Center 413 (4F)
Chair: Yuko Otani, Hideyo Takahashi

[29-413-pm16S]Discovery of covalent inhibitors based on FBDD approach (1): Evaluation of biocompatibility of CFA library and construction of cell screening system based on metabolic activity

○Ruikang Yin1, Kazuya Inoue, Saki Inoue1, Xiwen Xiao1, Shohei Uchinomiya1, Akio Ojida1 (1. Kyushu University)

[29-413-pm17S]Discovery of covalent inhibitors based on FBDD approach (2) : phenotype screening of CFA fragment library based on β-oxidation activity in cells

○Saki Inoue1, Kazuya Inoue, Ruikang Yin1, Xiwen Xiao1, Shohei Uchinomiya1, Akio Ojida1 (1. Grad. Sch. Pharm. Sci., Kyushu Univ.)

[29-413-pm18]Synthesis of linezolid metabolites (2)

○Naoki Oikawa1, Shogo Ishii1, Takumi Goto1, Hiroaki Saito1, Yasuhiro Tsuji1, Taketo Uchiyama1 (1. Sch. Pharm., Nihon Univ.)