The 144th Annual Meeting of the Pharmaceutical Society of Japan (Yokohama)
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Session Details

Poster Presentation(A) Pharmaceutical Chemistry

Other synthetic studies 1/Structure and physical property 1/Others

Fri. Mar 29, 2024 8:30 AM - 12:00 PM JST
Fri. Mar 29, 2024 11:30 PM - 3:00 AM UTC
[Poster 1] Exhibition Hall AB (1F)

[29P-am001S]Development of a new drug candidate for treatment of Menkes disease

○junna tamura1, Misaki Nakano1, Yoshino Takahashi1, Kayo Nakamura1, Hidetsugu Tabata2, Tetsuta Oshitari2, Hideaki Natsugari3, Kosho Makino4, Kiyomi Ito4, Hideyo Takahashi1 (1. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2. Faculty of Pharma-Science, Teikyo University, 3. Faculty of Pharmaceutical Sciences, The University of Tokyo, 4. Faculty of Pharmacy, Musashino University)

[29P-am002]Simple method for benzothiadiazine dioxide compounds using the redox properties of iron powder

○kyosuke kaneda1,2, Hirotoshi Kabasawa1, Syun Nabeki1, Uki Matsui1, Hiroki Sugiyama1, Takehiro Yamagishi1,2 (1. Pharm. Sci., HUS., 2. CRILS)

[29P-am003]Concise Synthesis of Dehydroanthophyine Derivative with Antimalarial Activity

○Hibiki Tomimori1, Naoto Yamasaki1, Yoshinori Asakawa1, Hirofumi Yamamoto1 (1. Faculy of Pharmaceutical Sciences Tokushima Bunri University)

[29P-am004S]Synthetic studies on tricyclic compounds using 1,3-dipolar cycloaddition reaction

○Nanako Oue1, Kohei Yoshinaga1, Satoshi Yokoshima1 (1. Grad. Sch. Pharm. Sci., Nagoya Univ.)

[29P-am005]Side-chain fluorination of 25-hydroxyvitamin D3 and their biological activity

○Fumihiro Kawagoe1, Sayuri Mototani1, Kaori Yasuda2, Hiroki Mano2, Toshiyuki Sakaki2, Atsushi Kittaka1 (1. Faculty Pharm. Sci., Teikyo Univ., 2. Faculty of Engineering, Toyama Prefectural Univ.)

[29P-am006S]Synthesis and crystal structure analysis of a series of Ac3c peptides having a sulfonamide group at N-terminus

○Kazuma Kondo1, Tomokatsu Enda1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci. Toho Univ.)

[29P-am007]Seven Polymorphs of Quinoline Sulfonamides

○Shoko Kikkawa1, Hiroki Daitoku1, Akihiro Hirata1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci. Toho Univ.)

[29P-am008S]Synthesis and crystal structures of Aib peptides with mesitylene- and naphthalene-sulfonamide.

○Yusuke Saiki1, Tomoka Ishikawa1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci.Toho Univ.)

[29P-am009S]Design and synthesis of electrophilic aminating reagents based on thianthrene scaffold

○Ryutaro Tawara1, Shohei Hamada1, Takumi Furuta1, Yusuke Kobayashi1 (1. Fac. Pharm., Kyoto Pharmaceutical University)

[29P-am010S]Transformation of alkene with hypervalent pnictogen compound

○Nagisa Ishida1, Yuuki Nishida1, Shohei Hamada1, Takumi Furuta1, Yusuke Kobayashi1 (1. Fac. Pharm., Kyoto Pharmaceutical University)

[29P-am011S]Development of odorless dithiophosphoric acid equivalent for hydrothiolysis of nitriles

○Sakura Tsujikawa1, Mei Ikeda1, Shohei Hamada1, Takumi Furuta1, Yusuke Kobayashi1 (1. Fac. Pharm., Kyoto Pharmaceutical University)

[29P-am012S]Structure and Property of Conformationally Controlled Urea and Thiourea by Chalcogen-bonding interaction

○Yui Amijima1, Takumi Inoue1, Moe Ota1, Nami Morita1, Shohei Hamada1, Seikou Nakamura1, Yusuke Kobayashi1, Takumi Furuta1 (1. Kyoto Pharmaceutical Univ.)

[29P-am013S]Synthesis of benzodichalcogenophene structures containing selenium atom for rhodium paddlewheel complexes.

○Yuumi Ushio1, Shohei Hamada1, Yuusuke Kobayashi1, Takumi Furuta1 (1. Fac.Pharm, Kyoto Pharmaceutical University)

[29P-am014S]Synthesis of C2-symmetrical oxoazahelicenes

○Yuki Arai1, Ryo Ikeda1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci. Toho Univ.,)

[29P-am015S]Synthesis of azahelicenes using stereochemistry of aromatic amide and Yamamoto coupling reaction.

○Ryo Ikeda1, Arai Yuki1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci. Toho Univ.)

[29P-am016S]Towards a synthesis of azananobelt analogs by ring fusion of cyclic aromatic amides

○Akane Ikoshi1, Ayaka Sugiyama1, Akito Miyakoshi1, Hidemasa Hikawa1, Shoko Kikkawa1, Isao Azumaya1 (1. Fac. Pharm. Sci. Toho Univ.)

[29P-am017S]Synthesis of oxoazacoronenes by Yamamoto coupling using Ni(0) reagent

○Yudai Takizawa1, Mariko Ninomiya1, Akihiro Yokoyama2, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci. Toho Univ., 2. Fac. Sci. Tech. Seikei Univ.)

[29P-am018S]One-step synthesis and crystal structures of spherical amides with C3-symmetry

○Haruka Uno1, Daiki Koike1, Hyuma Masu2, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci. Toho Univ., 2. CAI, Chiba Univ.)

[29P-am019S]Synthesis of novel π-conjugated hydrocarbons using McMurry coupling reaction

○Masayoshi Okazaki1, Yuki Saito1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci. Toho Univ.)

[29P-am020S]Synthesis of tetraphenyladamantane derivatives which have fluorescent emitting moieties at the ends of their side chains

○Yurika Yoshida1, Sae Maeda1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci. Toho Univ.)

[29P-am021S]Synthesis and conformational chirality of macrocyclic aromatic amides having diphenyldianthracene moieties

○Hisato Takahashi1, Taku Nakayama1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)

[29P-am022S]Conformational Control of Macrocyclic Peptides Utilizing Stereoisomerism of Benzamide

○Taichi Akahane1, Akira Katsuyama1, Satoshi Ichikawa1 (1. Faculty of Pharmaceutical Sciences, Hokkaido Univ.)

[29P-am023S]Atropisomeric properties of thioamides

○Ryota Takano1, Ryoko Tanaka1, Kayo Nakamura1, Hidetsugu Tabata2, Tetsuta Oshitari2, Hideaki Natsugari3, Hideyo Takahashi1 (1. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2. Faculty of Pharma-Science, Teikyo University, 3. Faculty of Pharmaceutical Sciences, The University of Tokyo)

[29P-am024S]The aggregation-induced intramolecular charge-transfer luminescence of o-carbaboranyl anisole derivatives

○Yui Asano1, Junna Ino1, Naoto Yamasaki1, Yoshinori Asakawa1, Hirofumi Yamamoto1 (1. Faculty of Pharmaceutical Sciences Tokushima Bunri University)

[29P-am025S]Steric properties and conformational preferences of N-(2-azulenyl) aromatic amides

○Mayuko Tomita1, Ai Ito1, Masayuki Yunoki1, Ai Tsuchida1, Mayuko Watanabe1, Ayako Ishii1, Takamasa Amaki1, Ryu Yamasaki1, Iwao Okamoto1 (1. Showa Pharmaceutical University)

[29P-am026S]Development of fluorescein based near-infrared photoredox catalyst

○Masaya Oyama1, Masaru Tanioka1, Yuji Matsuya1 (1. Faculty of Pharm. Sci., University of Toyama)

[29P-am027S]Peptide Design to Control Gel-to-Sol Transition Rate

○Yoshika Hara1, Atsuya Yaguchi1, Hirotsugu Hiramatsu2, Takahiro Muraoka1,3 (1. Grad. Sch. Eng., Tokyo Univ. of Agri. and Tech., 2. NYCU, 3. KISTEC)

[29P-am028S]Conformational behavior of N,N'-diaryl sudstituted Tf2C=C(NR2)2 type push-pull ethylene

Hikaru Yanai1, ○Masahi Shiozawa1, Tomoki Sakaguchi1, Takashi Matsumoto1 (1. Tokyo Univ. Pharm. Life Sci)

[29P-am029]Evaluation of the stability of helical structure by metal ion-mediated side chain cross-linking of peptides containing picoryl esters in the side chain

○takuma kato1, Yukino Yamamoto1, Naoki Kosukegawa1, Akari Yoshikawa1, Akiko Asano1, Mitsunobu Doi1 (1. Osaka. Med. Pharm. Univ.)

[29P-am030S]Synthesis of peptides with amino acids protected by a photoremovable group and their conformational analyses.

○Motoki Naka1, Tomohiro Umeno1, Hiroyasu Takemoto1, Atsushi Ueda2, Masakazu Tanaka2, Makoto Oba1 (1. Grad. Sch. Med. Sci., Kyoto Prefecture Univ. of Medicine, 2. Grad. Sch. Biomed. Sci., Nagasaki Univ.)

[29P-am031S]Synthesis of thioamides structurally controlled by sulfur-sulfur chalcogen bonds and their application to heterocyclic compounds

○Rika Sakai1, Takumi Inoue1, Shohei Hamada1, Yusuke Kobayashi1, Takumi Furuta1 (1. Fac. Pharm, Kyoto Pharmaceutical University)

[29P-am032]Elucidation of thermal behavior and single crystal structure determination of acetaminophen form III

○Kasumi Kihara1, Taiji Yamamoto1, Yasuaki Masuda1, Hiroyasu Sato1, Akito Sasaki1 (1. Rigaku Corporation)

[29P-am033]Synthesis, Characterization, and DNA cleavage activity of ZnII–Ant-[12]aneN3

○Yoshimi Ichimaru1, Koichi Kato1, Hiromasa Kurosaki2, Masaaki Kurihara1 (1. Fac. Pharm. Sci., Shonan Univ. Med. Sci., 2. Coll. Pharm., Kinjo Gakuin Univ.)

[29P-am034S]Synthesis of unnatural fluorinated dipeptides with protease inhibitory activity and their effects on the stereochemistry

○Airi Ginyama1, Yuya Miyasato1, Atsushi Tarui1, Ryuji Yamazawa1, Yukiko Karuo1, Kazuyuki Sato1, Kentaro Kawai1, Masaaki Omote1 (1. Pharm. Sci., Setsunan Univ.)

[29P-am035S]Synthesis and Properties of the Optically Active Ladder Oligonaphthalenes

○Misa Sakura1, Shunsuke Noda2, Takahiro Kimoto3, Keita Okada3, Yoshitane Imai3, Ayumi Imayoshi2, Kazunori Tsubaki2 (1. Faculty of Life and Environmental Sciences, Kyoto Prefectual University, 2. Graduate School of Life and Environmental Sciences, Kyoto Prefectual University, 3. Graduate School of Engineering, Kindai University)

[29P-am036]Development of influenza virus NA specific fluorescent probe

○Tadamune Otsubo1, Daiki Syuto1, Yutaka Narimichi2, Tadanobu Takahashi2, Yuuki Kurebayashi2, Akira Minami2, Fumiteru Teraoka1, Hideyuki Takeuchi2, Kiyoshi Ikeda1 (1. Faculty of Pharm. Sci., Hiroshima International Univ., 2. Sch. Pharm. Sci., University of Shizuoka)

[29P-am037]Synthetic research on sulfate monosaccharide type anti-dengue virus drug (4)

○fumiteru teraoka1, Takuma Miyamoto1, Chie Ustubo2, Kazuya IRJ Hirari3, Tadamune Otsubo1, Kiyoshi Ikeda1 (1. Grad. Sch. Pharm. Sci., Hiroshima Int. Univ., 2. Grad. Sch. Health. Sci., Kobe Univ., 3. Dpt. Food, Nutrition Scie., Aizu Jun. Univ.)

[29P-am038S]Steric Effects in Functional Amine Compounds for CO2 Absorbent

○Hisayo Oka1, Chika Suefusa1, Ryo Murakami1, Fuyuhiko Inagaki1 (1. Fac. Pharm. Sci., Kobegakuin Univ.)

[29P-am039S]Electronic Effects in Functional Amine Compounds for CO2 Absorption/Desorption Performance

○Sako Yoshida1, Chika Suefusa1, Ryo Murakami1, Fuyuhiko Inagaki1 (1. Fac. Pharm. Sci., Kobegakuin Univ.)

[29P-am040S]Synthesis and properties of an activator with a ahydrophobic unit for oligonucleotide synthesis

○Koichi Mizuno1, Yuta Ito1, Yasufumi Fuchi1, Yoshiyuki Hari1 (1. Fac. Pharm. Sci., Tokushima Bunri Univ.)

[29P-am041S]Development of novel bifunctional asymmetric organocatalysts

○Souki Sakai1, Teruyuki Ota1, Shinya Kimura1, Masamichi Yamanaka1, Masashi Yokoya1 (1. Meiji Pharm. Univ.)

[29P-am042]Evaluation of temperature-responsive self-assembly behavior of 4-aminoquinoline amphiphile: Selective construction of perforated vesicles and nanofibers

○Yosuke Hisamatsu1, Go Toriyama1, Katsuhiro Yamamoto2, Naoki Umezawa1 (1. Grad. Sch. Pharm. Sci., Nagoya City Univ., 2. Grad. Sch. Eng., Nagoya Inst. Tech.)

[29P-am043]Efficient fluorination on vitamin D3 side-chain using electrophilic fluorination reagent

○sayuri mototani1, Fumihiro Kawagoe 1, Kaori Yasuda2, Hiroki Mano2, Toshiyuki Sakaki2, Atsushi Kittaka1 (1. Faculty Pharm. Sci., Teikyo University, 2. Faculty of Engineering, Toyama Prefectural University)

[29P-am044]Synthesis and properties of 2-amino-4-fluoro-3-formylpyridine-C-nucleoside for covalent inhibition of protein function

○Kousuke Sato1, Masaru Morikawa1, Momoko Tsuruya1, Tetsushi Yamamoto1, Takahiro Sasaki1, Tsuyoshi Murai1 (1. Sch. Pharm. Sci., Health Sci. Univ. Hokkaido)

[29P-am045S]Dynamic Kinetic Resolution of 2-Phenylpropionic Acid esters by Chiral Quaternary Ammonium Salts

○Kokoro Kimura2, Kawasaki Midori1, Yatsuzuka Kenji2, Shirai Ryuichi1 (1. Grad. Sch. Pharm. Sci.,Doshisha Women's Col., 2. Fac. Pharm. Sci.,Doshisha Women's Col.)

[29P-am046S]Synthesis and evaluation of Perylene Diimides based CO2 absorbents

○Sayaka Kono1, Rie Shinohara1, Ryo Murakami1, Fuyuhiko Inagaki1 (1. Fac. Pharm. Sci., Kobegakuin Univ.)

[29P-am047S]Synthesis and characterization of Sulfinic acid-responsive fluorescent molecules

○Aoi Otsuki1, Shogo Kyogaku1, Hiroki Tanimoto1, Takenori Tomohiro1 (1. Dep. Pharm. Sci., Univ. Toyama)
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