The 144th Annual Meeting of the Pharmaceutical Society of Japan (Yokohama)
Advanced Search

Session Details

Poster Presentation(A) Pharmaceutical Chemistry

Chemical reaction development 1

Fri. Mar 29, 2024 1:30 PM - 5:00 PM JST
Fri. Mar 29, 2024 4:30 AM - 8:00 AM UTC
[Poster 1] Exhibition Hall AB (1F)

[29P-pm001S]Synthetic approach to kainoids via α-sp3C-H cyanation of amines under red-light irradiation

○naoaki yoshihara1, Takehiko Yoshimitsu1 (1. Grad. Sch. Pharm. Sci., Okayama Univ.)

[29P-pm002]Aldol-type macrocyclization reaction catalyzed by peptide foldamer catalysis

○Tomohiro Umeno1, Yuto Yamaberi2, Atsushi Ueda2, Makoto Oba1, Masakazu Tanaka2 (1. Grad. Sch. Med. Sci., Kyoto Prefectural Univ. of Medicine, 2. Grad. Sch. Biomed. Sci., Nagasaki Univ.)

[29P-pm003]Regio- and stereo-selective deuterium-labeling of amino acids under flow conditions

○Tsuyoshi Yamada1, Shuta Ichihara1, Kwihwan Kobayashi1, Takashi Ikawa1, Hironao Sajiki1 (1. Gifu Pharm. Univ.)

[29P-pm004S]Asymmetric Alkylation via Remote Asymmetric Induction: A Practical Approach to the Stereoselective Synthesis of Xaa-Asp-type Chloroalkene Dipeptide Isosteres

○Mio Takeda1, Chihiro Iio2, Daichi Toyama2, Kohei Sato1,2, Nobuyuki Mase1,2, Tetsuo Narumi1,2 (1. Fac. Eng., Shizuoka Univ., 2. Grag. Sch. Integ. Sci. Tech., Shizuoka Univ.)

[29P-pm005]Asymmetric aza-Henry reactions using peptide-catalysts with N-terminal benzothiadiazine

○Kazuki Satou1, Atsushi Ueda1, Masakazu Tanaka1 (1. Grad. Sch. Biomed. Sci., Nagasaki Univ.)

[29P-pm006S]Synthesis of tricyclic amine bearing contiguous tetrasubstituted carbons using a cyclization–3-aza-Cope–Mannich cascade

Mika Sugiyama1, ○Kaito Tozuka1, Yuji Mori1, Takeo Sakai1 (1. Fac.Pharm. Meijo Univ.)

[29P-pm007S]Photosensitizer-mediated racemization of chiral amino acid derivatives

○Ryusei Takada1, Riku Matsuda1, Kayo Nakamura1, Kosho Makino2, Hidetsugu Tabata3, Tetsuta Oshitari3, Hideaki Natsugari4, Hideyo Takahashi1 (1. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2. Faculty of Pharmacy, Musashino University, Faculty of Pharma-Science, 3. Faculty of Pharma-Science, Teikyo University, 4. Faculty of Pharmaceutical Sciences, The University of Tokyo)

[29P-pm008]Intramolucular Hydrophosphimylation of 2-Alkynylaryl-H-phosphinates

○Shino Nakajima1, Kengo Ayabe1, Ryoji Nozawa1, Shintaro Kamio1, Kyosuke Kaneda1,2, Takehiro Yamagishi1,2 (1. Department of Med. Chem., Hokkaido Univ. of Sci., 2. Creation Research Institute of Life Science in KITA-no-DAICHI, Hokkaido Univ. of Sci.)

[29P-pm009]Synthesis of π-conjugated molecules bearing P atom and their photophysical properties

○Yoshitaka Yamashita1, Fumiya Natori1, Shintaro Kamio1, Kyosuke Kaneda1,2, Takehiro Yamagishi1,2 (1. Department of Med. Chem., Hokkaido Univ. of Sci., 2. Creation Research Institute of Life Science in KITA-no-DAICHI, Hokkaido Univ. of Sci.)

[29P-pm010S]Investigation of Desulfurative Borylation in Aqueous Solvents

○Kazuhiro Yamashita1, Yui Hiranaka1, Minjae Kim 1, Hayato Sasamoto1, Daiki Fukue1, Taishi Ichinose1, Manaka Maeda1, Honami Matsumoto1, You Nonaka1, Kohei Yamada1, Yasuchika Yamaguchi1 (1. Nagasaki international university)

[29P-pm011]Development of reductive Heck arylation of unactivated olefin under mild condition

○Takahiro Shirai1, Yusuke Migitera2, Ryo Nakajima1, Takuya Kumamoto1 (1. Grad. Sch. Biomed. Health Sci., Hiroshima Univ., 2. Sch. Pharm. Sci., Hiroshima Univ.)

[29P-pm012]Steric Effect of Substitution on the Nitrogen in Ring-Closing Metathesis of Ene-Ynamides

○Hideaki Wakamatsu1, Saya Matsuzaka1, Ryoka Okamoto1, Yuichi Yoshimura1 (1. Fac. Pharm. Sci., Tohoku Med. Pharm. Univ.)

[29P-pm013S]Regio- and enantioselective synthesis of succinimides bearing all-carbon quaternary centers using a chiral phenanthroline-Pd catalyst

○Midori Adachi1, Masafumi Tamura1 (1. Dept. Pharm. Sci., Sanyo-Onoda City Univ.)

[29P-pm014S]Asymmetric Henry Reaction Using Bisoxazoline Ligands Bearing Two Fluorous Tags

Kazuki Ishihara1, ○Toya Natsume1, Yamato Kato1, Narisa Takeuchi1, Yuka Hayashi1, Yuna Hagiwara1, Shota Shibuya1, Takayuki Shioiri1, Masato Matsugi1 (1. Grad. Sch. Agri., Meijo Univ.)

[29P-pm015S]Dehydration of tertiary alcohols under the neutral conditions using Ru/C

○Shuki Oyama1, Shuji Akai2, Yoshinari Sawama2 (1. Sch. Pharm. Sci., Osaka Univ., 2. Grad. Sch. Pharm. Sci., Osaka Univ.)

[29P-pm016S]Synthesis of Acylglycosides Using Hypervalent Iodine Reagents and Their Use as Glycosyl Donors

○KANA YANASE1, KOJI MORIMOTO1,2, TETSUYA KAJIMOTO1, KITA YASUYUKI2 (1. Grad. Sch. Pharm. Sci., Ritsumeikan Univ., 2. Res. Org. Sci and Tech., Ritsumeikan Univ.)

[29P-pm017]Fluorous Lewis acid-catalyzed Ring-opening Reactions of 1,6-Anhydroglucopyranose

○Akihiro Yoshida1, Miki Namiki1, Ryo Sagara1, Chikako Takahashi1, Hiroshi Akutsu1, Takashi Yamanoi1 (1. Faculty of Pharmacy and Pharmaceutical Sciences, Josai University)

[29P-pm018]Asymmetric synthesis of benzyl alcohol using optically active 2-(tolylsulfinyl)phenyl ketones

○Toshinori Nakakita1, Karin Shigematsu2, Yoshinori Okuno1, Yasuo Sato1, Masashi Asai1, Yasuhito Nobushi2, Masaharu Toriyama2, Motofumi Miura2 (1. YOKOHAMA UNIVERSITY OF PHARMACY, 2. SCHOOL OF PHARMACY. NIHON UNIVERSITY)

[29P-pm019S]Development of the butenolide radical-mediated dimerization

○Mizuki Oda1, Maho Naito1, Souhei Teshigawara1, Tohru Nagamitsu1, Masaki Ohtawa1 (1. Sch. Pharm., Kitasato Univ.)

[29P-pm020]Effects of Reactant 1,3-Cyclohexanedione on Catalytic Reactions: Limiting the Loading Enables the Use of Less Catalyst in Spiro Ring Formations

○Muhammad Sohail1, Fujie Tanaka1 (1. Okinawa Institute of Science and Technology Graduate University)

[29P-pm021S]Synthesis of cyclic acetal by MHAT/RPC mechanism

○Takuma Sugimura1, Bartłomiej Szarłan2, Hiroki Shigehisa1 (1. Musashino Univ., 2. Adam Mickiewicz Univ.)

[29P-pm022]Alkynyl thioesters in halocyclization/oxidative aromatization to form thiophenes

Miari Kurihara1, Airi Ide1, ○hiroki shigehisa1 (1. Musashino Univ.)

[29P-pm023]Electrophilic epoxidation of α,β-unsaturated oximes and following ring-opening

○Yoshimitsu Hashimoto1, Kiwamu Yoshida1, Miyu Furugoori1, Toru Yoshino1, Kosaku Tanaka III1, Nobuyoshi Morita1, Osamu Tamura1 (1. Showa Pharm. Univ.)

[29P-pm024S]Catalytic Enantioselective Mannich Reactions of Ketones with Cyclic Ketimino Esters and Their Reverse Retro-Mannich Reactions to Afford Tetrasubstituted α-Amino Acid Derivatives

○Kuan-Lin Chen1, Fujie Tanaka1 (1. Okinawa Institute of Science and Technology Graduate University)

[29P-pm025S]Three-component coupling reaction by direct generation of nitrones and its application

○Ayaka Yamamoto1, Tatsuya Kouchi1, Riku Saito1, Kosaku Tanaka,Ⅲ1, Yoshimitsu Hashimoto1, Nobuyoshi Morita1, Osamu Tamura1 (1. Showa Pharm. Univ.)

[29P-pm026]DMAPO/Boc2O-Mediated One-Pot Direct N-Acylation of Less Nucleophilic N-Heterocycles with Carboxylic Acids

○atsushi umehara1, Soma Shimizu1, Makoto Sasaki1 (1. Grad. Sch. Life Sci. Tohoku Univ.)

[29P-pm027S]Palladium on carbon-catalyzed conversion of azides to nitriles

○Takanori Kitazono1, Naoya Sakurada1, Seiya Ohtori1, Takashi Ikawa1, Tsuyoshi Yamada1, Hironao Sajiki1 (1. Gifu Pharm. Univ.)

[29P-pm028]Synthesis of sulfonium salts from arylbenziodoxaborole with sulfides

○Akira Yoshimura1, Mekhman s Yusubov2, Nami Ogura1, Tatsuya Suzuki1, Akiharu Ueki1, Akio Saito3, Viktor V Zhdankin4 (1. Aomori Univ., 2. Tomsk Polytechnic University, 3. Tokyo University of Agriculture and Technology, 4. University of Minneota)

[29P-pm029]Development of the cyclization reaction with alkene and trifluoroacetamide group as radical precursor mediated by samarium(II) diiodide

○Hiroki Iwasaki1, Saho Ito1, Yuzuha Iwamoto1, Hisanori Nambu1 (1. Kyoto Pharmaceutical Univ.)

[29P-pm030]Alkylidene transfer from 1,3-dipoles to iminoiodanes

○Noriko Okamoto1, Haruto Ogino1, Keiji Konishi1, Takuya Sueda1 (1. Hiroshima International University)

[29P-pm031S]Development of synthesis for α-amino-β-lactam equivalent using N-Alkynylimide via the Kinugasa reaction

○Chie Nakamo1, Keiji Konishi1, Noriko Okamoto1, Takuya Sueda1 (1. Hiroshima International University)

[29P-pm032]Regioselective [3+2] Cycloaddition of Ynimides with Azomethine Imines to Generate N,N-Bicyclic 3-Pyrazolidinones

○Risako Hashimoto1, Keiji Konishi1, Noriko Okamoto1, Takuya Sueda1 (1. Hiroshima International University)

[29P-pm033]Environmentally benign thio-Michael reaction using acidic resin

○Yasunari Monguchi1, Arisa Kumagai1, Yuki Yoshida1, Shuri Yokotake1, Aika Matsuzono1, Natsuki Matsumura1, Kazutaka Koga1, Sayuri Yokoyama1 (1. Daiichi University of Pharmacy)

[29P-pm034]A general strategy for nucleophilic fluorination with Et3N・3HF complex via Halogen exchange

○Satoshi Mizuta1, Takeshi Ishikawa2 (1. Grad. Sch. Biomed. Sci., Nagasaki Univ., 2. Grad. Sch. Sci. Eng., Kagoshima Univ.)

[29P-pm035S]Kharasch addition to α,β-unsaturated oximes

Yuki Honda1, ○Tomohiro Hitoe1, Ayaka Yamamoto1, Yoshimitsu Hashimoto1, Kosaku Tanaka Ⅲ1, Nobuyoshi Morita1, Osamu Tamura1 (1. Showa Pharm. Univ.)

[29P-pm036S]Catalytic Direct Synthesis of Primary Amides from Carboxylic Acids Using Hexamethyldisilazane as the Nitrogen Source

○Shunsuke Kataoka1, Takashi Ohshima1 (1. Grad. Sch. Pharm. Sci., Kyushu Univ.)

[29P-pm037S]Development of One-Pot Transformation of Silyl Ethers to Nitriles

○Suzuka Kubozono1, Yuka Tanaka1, Yusuke Kobayashi1, Takumi Furuta1, Shohei Hamada1 (1. Fac. Pharm., Kyoto Pharmaceutical University)

[29P-pm038]Samarium-catalyzed pinacol coupling using a visible-light-absorbing antenna ligand

○Takahito Kuribara1, Ayahito Kaneki1, Yu Matsuda1, Tetsuhiro Nemoto1 (1. Grad. Sch. Pharm. Sci., Chiba Univ.)

[29P-pm039]Synthesis of azoxybenzene derivatives from nitroarenes via a reductive reaction using a catalytic amount of azastibocine

○yuki murata1, Seiya Nakashima1, Tomohiro Fujita1, Mio Matsumura1, Shuji Yasuike1 (1. Sch. Pharm. Sci., Aichi Gakuin Univ.)

[29P-pm040]Copper-catalyzed three component Se-arylation of selenium powder with pyrazolones and triarylbismuthanes

○Mio Matsumura1, Ayaka Nakamura1, Atsuki Yanagida1, Yuki Murata1, Shuji Yasuike1 (1. Sch. Pharm. Sci., Aichi Gakuin Univ.)

[29P-pm041S]Synthesis of novel benzoxazoloisoquinoliniums and optical properties

○Masato Kawakubo1, Megu Morishita2, Yuki Ohno2, Yuki Murata2, Mio Matsumura2, Shuji Yasuike2 (1. Grad. Sch. Pharm. Sci., Aichi Gakuin Univ., 2. Sch. Pharm. Sci., Aichi Gakuin Univ.)

[29P-pm042S]Synthesis of triphenylamines bearing a silicon substituent at the ortho position

○Yuria Sato1, Hikaru Fujita1, Shiori Kobayashi1, Munetaka Kunishima1,2 (1. Faculty of Pharmaceutical Sciences, Institute of Medical, Pharmaceutical, and Health Sciences, Kanazawa University, 2. Faculty of Pharmaceutical Sciences, Kobe Gakuin University)

[29P-pm043]Manganese(III)-catalyzed diastereoselective oxygenative aminoperoxidation

○Daisuke Yamamoto1, Yuki Narushima1, Issei Hirano1, Masayuki Soga1, Hiromasa Ansai1, Kazuishi Makino1 (1. School of Pharmacy, Kitasato Univ.)

[29P-pm044S]Hydrosilylation of Selenoesters and Its Synthetic Application

○Mustapha Kobina Abeka1, Alex Boateng1, Yuhei Ohta1, Masaharu Sugiura1 (1. Dept. Pharm. Sci., Sojo University)

[29P-pm045S]Development of highly efficient bifunctional asymmetric organocatalyst from conformationally rigid cis-1,2-diamines
~Search for hydrogen bond donor sites~

○Yuki Kurosawa1, Kento Muneta1, Satsuki Matsumoto1, Takuro Yasuyama1, Hirofumi Matsunaga1 (1. Fac. Pharm. Sci., Sanyo-Onoda City Univ.)

[29P-pm046S]Development of asymmetric organocatalyst with cis-1,2-diamine framework derived from indane skeleton

○Yuki Yamada1, Naoki Kawakami1, Rei Hodumi1, Takuro Yasuyama1, Hirofumi Matsunaga1 (1. Fac. Pharm. Sci., Sanyo-Onoda City Univ.)

[29P-pm047S]Synthesis of β-carboline via oxidative Pictet-Spengler reactions/DBU-mediated aerobic oxidation cascade

○Masakazu Kobayashi1, Shoko Kikkawa1, Isao Azumaya1, Hidemasa Hikawa1 (1. Fac. Pharm. Sci. Toho Univ.)

[29P-pm048S]Au(Ⅲ)-catalyzed dehydrative Bischler-Möhlau type indole synthesis

○Yuuka Kumono1, Taku Nakayama1, Shoko Kikkawa1, Isao Azumaya1, Hidemasa Hikawa1 (1. Fac. Pharm. Sci. Toho Univ.)

[29P-pm049S]Construction of imidazopyridine skeleton via Pd-catalyzed dehydrogenative oxidation of benzyl alcohol in water

○Nanoka Kobori1, Masakazu Kobayashi1, Taku Nakayama1, Shoko Kikkawa1, Isao Azumaya1, Hidemasa Hikawa1 (1. Fac. Pharm. Sci. Toho Univ.)

[29P-pm050S]Dehydrative/decarboxylative coupling of quinoline-4-carboxylic acids with allylic alcohols in water

○En Kenmochi1, Taku Nakayama1, Tomokatsu Enda1, Shoko Kikkawa1, Isao Azumaya1, Hidemasa Hikawa1 (1. Fac. Pharm. Sci. Toho Univ.)

[29P-pm051S]Extension of the Newman-Kwart Rearrangement to Heterocycles

○Yuma Okuda1, Keita Yamazaki1, Tetsuhiro Nemoto1 (1. Grad. Sch. Pharm. Sci., Chiba Univ.)

[29P-pm052S]HFIP accelerates the oxidation of alcohol using TEMPO and PIDA

○Kaori Sakamoto1, Wakana Oda1, Yusuke Kobayashi1, Takumi Furuta1, Shohei Hamada1 (1. Fac. Pharm., Kyoto Pharmaceutical University)

[29P-pm053S]Investigation of intermolecular anti-Markownikov Wacker-type reaction

Yasuhiro Nishikawa1, ○Sayaka Suzuki1, Momoka Suzuki1, Sara Kawanishi1, Kazuma Mizuno1, Mikako Aoki1, Osamu Hara1 (1. Fac. Pharm. , Meijo Univ.)

[29P-pm054S]The development of trivalent bismuth catalyzed oxidative coupling for arenols

Kengo Kasama1, ○HaoYang Dai1, Kousuke Umezawa1, Takayuki Yakura1 (1. University of Toyama)

[29P-pm055S]Site-selective deuteration of thioacetals using a potassium deuteroxide solution in D2O

○Hyoga Shimizu1, Shuji Akai2, Yoshinari Sawama2,3 (1. Sch. Pharm. Sci., Osaka Univ., 2. Grad. Sch. Pharm. Sci., Osaka Univ., 3. Deuterium Science Research Unit, Center for the Promotion of Interdisciplinary Education and Research, Kyoto University)

[29P-pm056S]Palladium-catalyzed construction of B,N-naphthalene scaffold

Yuto Iseya1, Ryotaro Kume1, ○Ryo Yanagida2, Ozora Sasamoto1,3, Yoshinori Kondo1, Masanori Shigeno1,4 (1. Grad. Sch. Pharm. Sci., Tohoku Univ., 2. Pharm. Sci., Tohoku Univ., 3. RCPD, 4. PRESTO, JST)

[29P-pm057S]Catalyst-Free Aziridination using In Situ Generated Iminoiodanes

○Asaka Kodama1, Shun Sunagawa1, Akira Tsubouchi1, Akio Saito1 (1. Grad. Sch. Eng., Tokyo Univ. Agric. Tech.)

[29P-pm058]Generation and Cycloaddition of Functionalized Arynes Generated from o-Triazenylarylboronic Acids

○Motoki Ito1, Haruna Yamazaki1, Yuta Takishima1, Aguri Ito1, Ryuhei Oda1, Moeka Komiya1, Kazuhiro Higuchi1, Shigeo Sugiyama1 (1. Meiji Pharmaceutical Univ.)

[29P-pm059S]Reactions for the introduction of perfluoroalkyl groups into carbonyl compounds

Tsuyoshi Yamada1, ○Mana Kumazawa1, Yutaro Yamada1, Takashi Ikawa1, Hironao Sajiki1 (1. Gifu. Pharm. Univ.)

[29P-pm060S]Synthesis of 1,2-dihydroisoquinoline derivatives by palladium-catalyzed cascade cyclization of allenamides and arylboronic acids

○Ryunosuke Imaji1, Shinya Shiomi1, Masahiro Yoshida1 (1. Faculty of Pharmaceutical Sciences, Tokushima Bunri University)

[29P-pm061S]Development of a new method for constructing benzazetine using dual-wavelength light irradiation

○Kaito Nakajima1, Masaru Tanioka1, Yuji Matsuya1 (1. Faculty of Pharm. Sci., University of Toyama)

[29P-pm062S]Nitrogen-containing heterocycle synthesis utilizing the nucleophilic imino carbon of the hydrazone

○Ayano Ichimonji1, Miku Nakayama1, Norihiko Takeda1, Motohiro Yasui1, Hiroshi Matsubara2, Masafumi Ueda1 (1. Kobe Pharmaceutical University, 2. Osaka Metropolitan University)
Back to Category List