The 144th Annual Meeting of the Pharmaceutical Society of Japan (Yokohama)
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Session Details

Poster Presentation(A) Pharmaceutical Chemistry

Total synthesis/Other synthetic studies 2

Sat. Mar 30, 2024 8:30 AM - 12:00 PM JST
Sat. Mar 30, 2024 11:30 PM - 3:00 AM UTC
[Poster 1] Exhibition Hall AB (1F)

[30P-am001S]Synthetic study of Lycopladine H

Hiroshi Takikawa2, ○Yoshiaki Yoh1, Chiho Yorozuya2, Kiyosei Takasu2 (1. Fac. Pharm. Sci., Kyoto Univ., 2. Grad. Sch. Pharm. Sci., Kyoto Univ.)

[30P-am002]Synthetic study of dalomycin T

Ryuto Watanabe1, Yasutaka Chino1, ○Yusuke Akagi1, Erika Iwasaki1, Toshiya Komatsu1 (1. Fac. Pharm. Sci., Teikyo Heisei Univ.)

[30P-am003S]Total Synthesis of Dragmacidins G and H

○Keita Yamazaki1, Yuma Okuda1, Akiko Takaya1, Tetsuhiro Nemoto1 (1. Grad. Sch. Pharm. Sci., Chiba Univ.)

[30P-am004S]Synthetic Studies on Catharanthine

○Sakiko Namba1, Hirofumi Ueda1, Hidetoshi Tokuyama1 (1. Grad. Sch. Pharm. Sci., Tohoku Univ.)

[30P-am005S]Synthetic studies on discorhabdin alkaloids by desymmetrization approach using thio-Michael addition

○Shunta Kitao1, Masashi Shimomura1, Kohta Ide1, Juri Sakata1, Hidetoshi Tokuyama1 (1. Grad. Sch. Pharm. Sci., Tohoku Univ.)

[30P-am006S]Synthetic Studies on (+)-Pericyclivine via Radical Cyclization

Sota Nishimuro1, ○Keita Moriyasu1, Hirofumi Ueda1, Hidetoshi Tokuyama1 (1. Grad. Sch. Pharm. Sci., TOHOKU Univ.)

[30P-am007S]Total Synthesis of Furo[3,2-c]quinoline Alkaloid Using Intramolecular Biaryl Coupling Reaction

○Nana Kusaka1, Keito Murayama2, Naoto Matsuba2, Hitoshi Abe2 (1. Fac. Eng., Toyama Univ. , 2. Grad. Sch. Sci. and Eng., Toyama Univ.)

[30P-am008S]Studies toward total synthesis of neostenine

Anri Yamamoto1, ○Mizuki Shiratori1, Hiroki Kumazaki1, Rika Goto1, Chihiro Ueda1, Yuji Mori1, Takeo Sakai1 (1. Fac. Pharm., Meijo Univ.)

[30P-am009]Synthetic study of Batzelladine O

○Taichi Kusakabe1, Yue Tianci1, Takuya Tsukamoto1, Keisuke Takahashi1, Keisuke Kato1 (1. Faculty of Pharmaceutical Sciences, Toho University)

[30P-am010S]Synthetic study of crambescin A2 392 analogues based on cyclization-carbonylation reaction

○Kyoka Someya1, Fujino Sakata1, Natsuki Murase1, Takuya Tsukamoto1, Taichi Kusakabe1, Keisuke Takahashi1, Keisuke Kato1 (1. Grad. Sch. Pharm. Sci., Toho Univ.)

[30P-am011S]Synthesis of α-Tocopherol

○Ayaka Nakamine1, Kei Kitamura1, Hiroto Kaku1 (1. Fac. Pharm. Sci., Tokushima Bunri Univ.)

[30P-am012S]Total synthesis of lamellolactones

○Yuto Fuse1, Tohru Nagamitsu1, Masaki Ohtawa1 (1. Sch. Pharm., Kitasato Univ.)

[30P-am013S]Total synthesis of Alanense A

○Rio Fukuda1, Kosho Makino1,2, Shunsuke Sueki1,2, Masahiro Anada1,2 (1. Fac. Pharm., Musashino Univ., 2. Res. Inst. Pharm. Sci., Musashino Univ.)

[30P-am014S]Synthetic Study of Antimalarial Meroterpene Natural Products

○Masahiro Iwahori1, Goh Sennari1,2, Soichiro Kimura1, Yoshihiro Watanabe1,2, Masato Iwatsuki1,2, Tomoyasu Hirose1,2, Toshiaki Sunazuka1,2 (1. Grad. Sch. of Infect. Ctl., Kitasato Univ., 2. Omura Satoshi Memorial Inst., Kitasato Univ.)

[30P-am015S]Synthetic study of tricyclic skeleton of kitungolide B.

○Masaki Yonekura1, Toyoharu Kobayashi1, Yuichiro Kawamoto1, Hisanaka Ito1 (1. Tokyo University of Pharmacy and Life Sciences)

[30P-am016S]Asymmetric total synthesis of (–)-lemnalemnane A

○Rina Sugitate1, Toyoharu Kobayashi1, Yuichiro Kawamoto1, Hisanaka Ito1 (1. Tokyo University of Pharmacy and Life Sciences)

[30P-am017S]Synthetic Study of Meroterpenoid Manginoid E

○Koki Hosoi1, Naoya Endo1, Toyoharu Kobayashi1, Yuichiro Kawamoto1, Hisanaka Ito1 (1. Tokyo University of Pharmacy and Life Sciences)

[30P-am018S]Synthetic Study of Tetracyclic Diterpenoid Venezuelaene B

○Zen Suzuki1, Yuichiro Kawamoto1, Toyoharu Kobayashi1, Hisanaka Ito1 (1. Tokyo University of Pharmacy and Life Sciences)

[30P-am019S]Synthesis and biological activity evaluation of curcusone A and B

Hideki Abe1, ○Chiharu Arai1, Akino Morikawa1, Yoshima Ide2, Ryohei Saito-Moriya1, Yuichiro Kawamoto2, Toyoharu Kobayashi2, Akihito Yokosuka3, Yoshihiro Mimaki3, Hisanaka Ito2 (1. Fac. Sci., Japan Women's Univ., 2. Sch. Life Sci., Tokyo Univ. Pharm. Life Sci., 3. Sch. Pharm., Tokyo Univ. Pharm. Life Sci.)

[30P-am020S]Total syntheses and biological activity evaluation of tricyclic natural products from the soft coral

Hideki Abe1, ○Nanako Inaba1, Mayu Nomura1, Yuta Ogura2, Ryohei Saito–Moriya1, Yuichiro Kawamoto2, Toyoharu Kobayashi2, Akihito Yokosuka3, Yoshihiro Mimaki3, Hisanaka Ito2 (1. Fac. Sci., Japan Women's Univ., 2. Sch. Life Sci., Tokyo Univ. Pharm. Life Sci., 3. Sch. Pharm., Tokyo Univ. Pharm. Life Sci.)

[30P-am021S]Protecting-Group-Free Total Syntheses of Boscartins

○Airi Miyazaki1, Misaki Niizato1, Hiroto Aihara1, Daisuke Kounai1, Akihiko Kasamatsu1, Junya Shiraiwa1, Shogo Kamo1, Akinobu Matsuzawa1, Kazuyuki Sugita1 (1. Hoshi Univ.)

[30P-am022]Synthetic study of wickerols, potent anti-influenza activities

○Takuma Miyata1, Goh Sennari1,2, Tomoyasu Hirose1,2, Toshiaki Sunazuka1,2 (1. Grad. Sch. of Infect. Ctl., Kitasato Univ., 2. Ōmura Satoshi Memorial Inst., Kitasato Univ.)

[30P-am023S]Improvement study of Michael–Michael–alkylation reaction toward a synthesis of antheridiogen–An

○Soichiro Fujiwara1, Satoshi Kaneko1, Kokoro Nagasawa1, Kazuma Matsunaga1, Hiroto Nagaoka1, Kazuhiko Takatori1 (1. Meiji Pharmaceutical University)

[30P-am024S]A novel synthetic approach to brianthein W

○Hiromi Arai1, Kazuma Matsunaga1, Atsushi Kishida1, Kazuhiko Takatori1 (1. Meiji Pharmaceutical University)

[30P-am025S]Total Synthesis of Cryptolaevilactone

○Tomoya Nishida1, Yuta Miura1, Yohei Saito1, Kyoko Nakagawa-Goto1,2 (1. Grad. Sch. Pharm. Sci., Kanazawa Univ., 2. UNC)

[30P-am026S]Total synthesis of marine natural product Dysibetaine by oxidative modification of hydrocarbon compound

Yasuhiro Nishikawa1, ○Mikako Aoki1, Yuka Takeda1, Nanaka Kurumiya1, Rino Hishiki1, Chifumi Yasuda1, Jun Baku1, Nao Sato1, Shiori Sakakibara1, Yuuki Ito1, Shuuto Nakayama1, Osamu Hara1 (1. Faculty of Pharmacy, Meijo University)

[30P-am027S]Synthetic study of oxypinnatanine

○Kurumi Shoji1, Nao Hayashida1, Nanase Sekiguch1, Akari Miyawaki1, Junpei Matsuoka2, Yasutomo Yamamot1 (1. Doshisha Women's College of Liberal Arts, 2. Kindai University)

[30P-am028]Concise synthesis of pleurocybellaziridine

Sora Nose1, Fuma Shiosawa1, Takashi Matsuda1, Danya He1, ○Tomohiro Asakawa1 (1. Tokai University, School of Marine Science and Technology, Department of Fisheries)

[30P-am029S]Synthesis of cytosamine

Hanaka Sato1, ○Eri Saima1, Daiki Lee1, Shiho Arima1, Taichi Ohshiro1, Hiroshi Tomoda1, Tohru Nagamitsu1 (1. Sch. Pharm., Kitasato Univ.)

[30P-am030S]Study on Enantio-divergent Synthesis of (+)- and (−)-Uvaridacol L Using Desymmetriyation of Dialdose by Chiral NHC-catalyzed Benzoin Reaction

○Yuki Takahara1, Tsubasa Inokuma1, Ken-ichi Yamada1 (1. Grad. Sch. Pharm. Sci. Tokushima Univ.)

[30P-am031S]Synthetic study of hypocreolide A

○Shiuto Soma1, Daiki Lee1, Shiho Arima1, Taichi Ohshiro1, Tohru Nagamitsu1 (1. Sch. Pharm., Kitasato Univ.)

[30P-am032]Synthetic study of tricyclic diterpenoid homoverrucosanol

○Shinnosuke Okazaki1, Shiori Yamashita1, Isshin Nishimura1, Kazuo Kamaike1, Koichiro Ota1, Hiroaki Miyaoka1 (1. Tokyo Univ. of Pharm. and Life Sci.)

[30P-am033]Synthetic study of long-chain ether lipid botryococcoid ethers

○Yuha Maeda1, Sara Yamazaki1, Madoka Sugiyama1, Mina Yoshimura1, Lisa Onai1, Aoi Kadokura1, Atsuko Miura1, Kazuo Kamaike1, Shinnosuke Okazaki1, Koichiro Ota1, Hiroaki Miyaoka1 (1. TUPLS)

[30P-am034]Total synthesis and structure revision of saniculamoid D

○Koichiro Ota1, Kazuo Kamaike1, Hiroaki Miyaoka1 (1. TUPLS)

[30P-am035]Synthesis of mohangic acid C analogues

○Keisuke Takahashi1, Mai Sato1, Misato Shibuya1, Nana Hasegawa1, Kasumi Matsuo1, Ayu Watanabe1, Ayane Iioka1, Takuya Tsukamoto1, Shoko Kikkawa1, Isao Azumaya1, Taichi Kusakabe1, Keisuke Kato1 (1. Toho Univ.)

[30P-am036S]Synthesis of Cyclopentenone Type Natural Products Bearing α-Keto Vinyl Carbinol Moiety

○Chihiro Shizuma1, Natsuki Asada1, Karin Negoro1, Noboru Hayama1, Hiroki Yoneyama1, Yoshihide Usami1 (1. Osaka Med. & Pharm. Univ.)

[30P-am037S]Synthetic study of Actinollides anti-trypanosomal agent

○Wataru Terauchi1, Akito Watanabe1, Yoshihiko Noguchi1,2, Yuki Inahashi1,2, Masato Iwatsuki1,2, Aki Ishiyama1,2, Tomoyasu Hirose1,2, Toshiaki Sunazuka1,2 (1. Grad.Sch.of Infect. Ctl., Kitasato Univ., 2. Ōmura Satoshi Memorial Inst., Kitasato Univ.)

[30P-am038S]Modular Approach toward Total Synthesis of Ivermectin

○Masaya Ogawa1, Goh Sennari1,2, Ryo Saito1, Shougo Sato1, Tomoyasu Hirose1,2, Toshiaki Sunazuka1,2 (1. Grad. Sch. of Infect. Ctl., Kitasato Univ., 2. Ōmura Satoshi Memorial Inst., Kitasato Univ.)

[30P-am039S]Synthetic studies of oxidized phospholipids that have prostane structure

○Natsuki Ishiyama1, Hiroaki Matoba1, Makoto Yoritate1, Ken-ichi Yamada1, Go Hirai1 (1. Grad. Sch. Pharm. Sci., Kyushu Univ.)

[30P-am040]Syntheses of novel compounds to control the differentiation of Neopyropia tenera.

○Momoka Takahashi1, Hiroto Kaku1, Naoto Yamasaki1, Yoshinori Asakawa1, Hirofumi Yamamoto1 (1. Faculty of Pharmaceutical Sciences Tokushima Bunri University)

[30P-am041S]Studies on the oxidative cyclization reaction toward the synthesis of aaptamine skeleton

Yuki Nakatani1, ○Hitoshi Takatsu2, Risa Kimura1, Naoyuki Kotoku1,2 (1. Grad. Sch. Pharm. Sci., Ritsumeikan Univ., 2. Coll. Pharm. Sci., Ritsumeikan Univ.)

[30P-am042S]Drug discovery and development of novel AMDCs using Duocarmycin derivatives.

Akihiro Shimizu1, ○Shunya Homma1, Naoya Miyamoto1, Yuya Inagaki1, Juri Sakata1, Hidetoshi Tokuyama1 (1. Grad. Sch. Pharm. Sci., Tohoku Univ.)

[30P-am043S]Structure-activity relationship of Fentanyl derivatives

○Haruka Sakata1, Hironobu Arita1, Shuntaro Kikukawa1, Tsukasa Tomizawa1, Masahiko Funada2, Kenichi Tomiyama3, Hidetsugu Tabata4, Kayo Nakamura1, Tetsuta Oshitari4, Hideaki Natsugari5, Hideyo Takahashi1 (1. Faculty of Pharmaceutical Sciences, Tokyo University of Science , 2. Faculty of Pharmaceutical Sciences, Shonan University of Medical Sciences, 3. Section of Addictive Drug Research, Department of Drug Dependence Research, National Institute of Mental Health, National Center of Neurology and Psychiatry, 4. Faculty of Pharma-Science, Teikyo University, 5. Faculty of Pharmaceutical Sciences, The University of Tokyo)

[30P-am044S]Synthetic study of novel metabolites of abiraterone

○Ryuji Higashida1, Noboru Hayama1, Yukina Nishi1, Shizuyo Horiyama2, Hiroki Yoneyama1, Jun Haginaka3, Yoshihide Usami1 (1. Fac. Pharm., Osaka Med. Pharm. Univ., 2. Sch. Pharm. Pharmaceut. Sci., Mukogawa Women's Univ., 3. Inst. Biosci., Mukogawa Women's Univ.)

[30P-am045S]Synthetic studies of new derivatives based on Andrastins’ C,D ring fragment

○Fumino Kitamura1, Ayano Kosaka1, Masaru Tanioka1, Yuji Matsuya1 (1. Faculty of Pharm. Sci., University of Toyama)

[30P-am046]Synthesis of α-trifluoromethyl α-(4-pentenyl)glycine and application to tethering of peptide side chains

○Atsushi Ueda1, Ken Matsuta1, Takuma Kato2, Mitsunobu Doi2, Masakazu Tanaka1 (1. Grad. Sch. Biomed. Sci., Nagasaki Univ., 2. Fac. Pharm., Osaka Med. Pharm. Univ.)

[30P-am047S]Synthetic Study on Histicorrugatin Containing Cyclic Amidine Backbone

○Shoya Kawai1, Yoshinori Taguchi2, Kohei Sato1, Nobuyuki Mase1, Hiroyuki Hutamata1, Tetsuo Narumi1,2 (1. Fac. Eng., Shizuoka Univ., 2. Grad. Sch. Med. Photonics, Shizuoka Univ.)

[30P-am048S]Synthetic Study on Amyloid Peptide β49

○Taiyo Hagiwara1, Shoko Tanaka2, Kohei Sato1,2, Nobuyuki Mase1,2, Akio Fukumori3, Tetsuo Narumi1,2 (1. Fac. Eng., Shizuoka Univ., 2. Res. Inst. Green Sci. Tech., Shizuoka Univ., 3. Pharm. Sci., Osaka Med. Fharm. Univ.)

[30P-am049S]Diastereoselective Synthesis of Chloroalkene Dipeptide Isosteres Containing α,α-Disubstituted Amino Acid

○Harui Miyata1, Sayuri Takeo2, Yui Suruga1, Kohei Sato1, Nobuyuki Mase1, Tetsuo Narumi1,2 (1. Fac. Eng., Shizuoka Univ., 2. Grad. Sch. Med. Photonics, Shizuoka Univ.)

[30P-am050S]Enantioselective synthesis of cyclopropane amino acid using bisphenymenthyl alkylidenemalonate

○Shinya Sotohara1, Tsubasa Inokuma1, Ken-ichi Yamada1 (1. Sch. Pharm. sci., Tokushima Univ.)

[30P-am051S]Asymmetric epoxidation using helical peptides with carbocyclic α,α-disubstituted α-amino acids having cross-linking motif.

○Akihiro Iyoshi1, Atsushi Ueda1, Tomohiro Umeno1, Kazuhiro Hirayama1, Takuma Kato2, Mitsunobu Doi2, Masakazu Tanaka1 (1. Grad. Sch. Biomed. Sci., Nagasaki Univ., 2. Fac. Pharm., Osaka. Med. Pharm. Univ.)

[30P-am052]Synthesis of beta-mercaptoamino acid derivatives and installation of glycan tag

○junpei abe1, Yumi Fujioka1, Teppei Miwa1, Yuta Maki1,2, Ryo Okamoto1,2, Yasuhiro Kajihara1,2 (1. Grad. Sch. Sci., Osaka Univ., 2. FRC, Grad. Sch. Sci., Osaka Univ.)

[30P-am053]Synthesis of elastin-like peptide analogues by ammonia-Ugi reaction

○Keisuke Tomohara1, Satoru Kusaba2, Naoki Tanaka2, Takeru Nose1,2 (1. Faculty of Arts and Science, Kyushu Univ., 2. Grad. Sch. Sci., Kyushu Univ.)

[30P-am054S]Preparation of N-Nps-α-iminophosphonamide for development of a synthetic method for α-aminophosphate-containing peptides

○Ayaka Mitsuyasu1, Takuya Sakakibara1, Tsubasa Inokuma1, Ken-ichi Yamada1 (1. Sch. Pharm. Sci., Tokushima Univ.)

[30P-am055]Synthesis and analysis of stability of 6-unsubstituted 2-aryl-1,4-dihydropyrimidine tautomers by Pd-catalyzed/CuCl-mediated Liebeskind-Srogl-type cross-coupling reaction

○Yoshio Nishimura1, Keito Taira1, Yusuke Yamamoto1, Takanori Kubo2, Hidetsura Cho3 (1. Sch. Pharm. Sci., Ohu Univ., 2. Fac. Pharm., Yasuda Women's Univ., 3. Grad. Sch. Pharm. Sci., Tohoku Univ.)

[30P-am056]Design and synthesis of a novel water-soluble vizantin

○Rinka Bekku1, Naoto Yamasaki1, Takashige Kawakami1, Masahisa Inoue1, Yoshinori Asakawa1, Hirofumi Yamamoto1 (1. Faculty of Pharmaceutical Sciences Tokushima Bunri University)

[30P-am057S]Improvement of the Synthesis and purification of Cyclic Oligosaccharides by One-pot Glycosylation of Glycosyl Donor/Acceptors.

○Tatsuya Yamada1, Gouta Ishigami1, Toshifumi Tojo1, Yasuyuki Yamada2, Shin Aoki1,3,4 (1. Grad. Sch. Pharm. Sci., Tokyo Univ. of Sci., 2. Res. Cent. for Mater. Sci., Naoya Univ., 3. Res. Inst. for Sci & Tech., Tokyo Univ. of Sci., 4. Res. Inst. for Biomed. Sci., Tokyo Univ. of Sci.)

[30P-am058S]Development of a Facile β-D-Glucuronidation Reaction by Using Methyl 1,2,3,4-Tetra-O-acetyl-D-glucuronate as a Glycosyl Donor

○Tianqi DU1, Yuki Sakai1, Kaneko Kimiyoshi2, Yasuyuki Matsushima3, Tsuyoshi Miura3, Tetsuya Kajimoto1 (1. Pharm. Sci., Ritsumeikan Univ., 2. Res. Org. Sci. & Tech., Ritsumeikan Univ., 3. Pharm. Sci., Tokyo Univ. Pharm. & Life Sci.)

[30P-am059S]Synthesis of 4’-substituted adenosine derivatives targeting SARS-CoV-2 RNA polymerase

○Kotomi Otsuki1, Ayami Takayama1, Makoto Roppongi2, Shinichiro Hattori3, Nobuyo Kuwata3, Hiroaki Mitsuya3, Kiju Konno1 (1. International University of Health and Welfare, Department of Pharm. Sci., 2. Center for Industry-University Innovation Support of Utsunomiya Univ, 3. National Center for Global Health and Medicine, Department of Refractory Viral Infection)

[30P-am060S]Synthesis of carbovir derivatives as therapeutic agents for adenovirus infections

○Eri Hasegawa1, Nachi Watanabe1, Kotomi Otsuki1, Makoto Roppongi2, Shinichiro Hattori3, Nobuyo Kuwata3, Hiroaki Mitsuya3, Kiju Konno1 (1. International University of Health and Welfare, Department of Pharm. Sci., 2. Center for Industry-University Innovation Support of Utsunomiya Univ, 3. National Center for Global Health and Medicine, Department of Refractory Viral Infection)

[30P-am061S]Synthesis of 4'-substituted carbocyclic nucleosides targeting SARS-CoV-2 RNA polymerase

○Nachi Watanabe1, Eri Hasegawa1, Kotomi Otsuki1, Makoto Roppongi2, Shinichiro Hattori3, Nobuyo Kuwata3, Hiroaki Mitsuya3, Kiju Konno1 (1. International University of Health and Welfare, Department of Pharm. Sci., 2. Center for Industry-University Innovation Support of Utsunomiya Univ, 3. National Center for Global Health and Medicine, Department of Refractory Viral Infection)

[30P-am062]Preparation of thymidine derivatives functionalized at 5'-position as monomer units and their conjugation of phosphate diesters for novel strategies to oligonucleotide synthesis

○Risa Yamaguchi1, Yoshiaki Kitamura1,2,3,4 (1. Fac. Eng., Gifu Univ., 2. Grad. Sch. Nat. Sci. Tech., Gifu Univ., 3. United Grad. Sch. Drug Discov. Med. Info. Sci., Gifu Univ., 4. Ctr. One Med. Innov. Transl. Res., Gifu Univ.)

[30P-am063S]Novel synthetic route for 1′-C,3′-O-propylene-bridged altritol nucleic acid

○Tomoki Yoshimura1, Takashi Nakamura2, Takao Yamaguchi2, Satoshi Obika2,3 (1. Sch. Pharm. Sci., Osaka Univ.,, 2. Grad. Sch. Pharm. Sci., Osaka Univ., 3. OTRI, Osaka Univ.)

[30P-am064S]Design and synthesis of amphiphilic supramolecular catalysts for catalytic hydrolysis of Phosphate Monoester.

○Ayane Nomoto1, Hirokazu Okamoto1, Toshifumi Tojo1, Shin Aoki1,2,3 (1. Grad. Sch. Pharm. Sci., Tokyo Univ. of Sci., 2. Res. Inst. for Sci. & Tech., Tokyo Univ. of Sci., 3. Res. Inst. for Biomed. Sci., Tokyo Univ. of Sci.)

[30P-am065S]Synthesis of Bisoxazoline- Pyridylamide Frameworks for Chiral Z-Type Ligands

○Shingo Kuge1, Mayuka Tsutaka1, Ryo Murakami1, Fuyuhiko Inagaki1 (1. Fac. Pharm. Sci., Kobegakuin Univ.)
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