The 144th Annual Meeting of the Pharmaceutical Society of Japan (Yokohama)
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Session Details

Poster Presentation(A) Pharmaceutical Chemistry

Chemical reaction development 2/Reaction mechanism/computational chemistry/Molecular recognition

Sat. Mar 30, 2024 1:30 PM - 5:00 PM JST
Sat. Mar 30, 2024 4:30 AM - 8:00 AM UTC
[Poster 1] Exhibition Hall AB (1F)

[30P-pm001]Efficient preparation of nitroalkenes using benzaldehyde derivatives as the starting materials

○Yuka Arai1, Hisao Kansui2, Tomoko Mineno1 (1. Faculty of Pharm., Takasaki Univ. of Health and Welfare, 2. Faculty of Pharmaceutical Sci., Sojo Univ.)

[30P-pm002]Functional group conversion from aldehydes to nitroalkenes based on the aromatic heterocycles

○Yukiho Araki1, Hisao Kansui2, Tomoko Mineno1 (1. Faculty of Pharm., Takasaki Univ. of Health and Welfare, 2. Faculty of Pharmaceutical Sci., Sojo Univ.)

[30P-pm003S]Conversion of swertiamarin isolated from Swertia Herb to 4-acyloxygentianine.

Sakurako Shimizu1, Hinata Matsuo1, ○Ryoya Kaneko1, Takaya Noguchi1, Yasuaki Hirai2, Mikio Fujii1 (1. Grad. Sch. Pharm., Int. Univ. Health Welf., 2. Mt. Fuji Inst. Nat. Biol., Showa Univ.)

[30P-pm004S]Development of 1,4-Benzoxazepin-5-one Synthesis via Palladium-Catalyzed Heteroannulation

Masahiro Abe1, ○Megumu Kawamoto1, Akiho Mizukami1, Tetsutaro Kimachi1, Kiyofumi Inamoto1 (1. Sch. Pharm. Sci., Mukogawa Women's Univ.)

[30P-pm005S]3,1-Benzoxazin-4-one synthesis by gold-catalyzed heteroannulation

Masahiro Abe1, ○Mai Takano1, Mizukami Akiho1, Kimachi Tetsutaro1, Kiyofumi Inamoto1 (1. Sch. Pharm. Sci., Mukogawa Women's Univ.)

[30P-pm006S]Development of Minisci-Type Remote Heteroarylation of Fluorinated Compounds via 1,5-HAT

Masahiro Abe1, ○Yumeno Matsuoka1, Kuku Inoue1, Mizukami Akiho1, Kimachi Tetsutaro1, Kiyofumi Inamoto1 (1. Grad. Sch. Pharm. Sci., Mukogawa Women's Univ.)

[30P-pm007S]Development of Remote Diazenylation of Fluorinated Compounds via 1,5-Hydrogen Atom Transfer

Masahiro Abe1, ○Airu Kataoka1, Aoi Hirata1, Nagisa Yano1, Akiho Mizukami1, Tetutaro Kimachi1, Kiyofumi Inamoto1 (1. Sch. Pharm. Sci., Mukogawa Women's Univ.)

[30P-pm008]Development of aza-Friedel–Crafts reactions of N-acyliminium ions catalyzed by boronic acids with amino acid derivatives

○Akira Nakamura1, Yuito Kamei1, Yusuke Azuma1, Jyunpei Matsuoka1, Tomohiro Maegawa1 (1. Sch. Pharm. Sci., Kindai Univ.)

[30P-pm009S]Gold-catalyzed Synthesis of Poly-Substituted Pyrroles

○Yukinori Umezawa1, Nobuyoshi Morita1, Hitomi Chiaki1, Yoshimitsu Hashimoto1, Osamu Tamura1 (1. Showa Pharm. Univ.)

[30P-pm010S]Photoacid-induced Mukaiyama aldol reaction of isocoumarins and its application to polysubstituted arene synthesis

○Rio Aikawa1, Yu Hirashima1, Hirotaka Hotta1, Teru Kawazoe1, Takashi Matsumoto1, Hikaru Yanai1 (1. Tokyo Univ. Pharm. Life Sci.)

[30P-pm011S]Phosphazene base-catalyzed addition of enolate to alkenes and its application to lignan synthesis

○Saki Nikaido1, Honoka Nodao1, Akari Miyawaki1, Junpei Matsuoka2, Yasutomo Yamamoto1 (1. Doshisha Women's College of Liberal Arts, 2. Kindai University)

[30P-pm012]Effect of additives in the formation reaction of [3.3](2,2')(4,4’-bithiazolopane) skeleton exhibiting c-Met inhibitory activity

Akira Matsutsuru1, ○Tatsuya Takimoto1, Koji Aoki1, Makito Kimura1, Takumi Sei1, Kazuhito Hioki1, Hideaki Sasaki1, De-qi Yuan1 (1. Fac. Pharm. Sci., Kobe Gakuin Univ.)

[30P-pm013]Effects of substituents on C-H arylation reaction to 2-amino-1-phenylethanol

○Karin Shigematsu1, Motofumi Miura1, Masaharu Toriyama1 (1. School of Pharmacy, Nihon University)

[30P-pm014S]Iron-porphyrin Catalyzed Dearomative Arene Cyclopropanation Reaction

○Qitong Dai1, Jun Ueda1, Shingo Harada1, Tetsuhiro Nemoto1 (1. Grad. Sch. Pharm. Sci., Chiba Univ.)

[30P-pm015S]Ag-Catalyzed C5-Selective C-H Functionalization of Indoles

○Tomohiro Isono1, Mai Yanagawa2, Shingo Harada2, Tetsuhiro Nemoto2 (1. Fac. Pharm. Sci., Chiba Univ, 2. Grad. Sch. Pharm. Sci., Chiba Univ)

[30P-pm016S]Phosphazene base-catalyzed intramolecular hydroalkoxylation of hydroxyalkene

○Miyu Kawamoto1, Noriko Yamashita1, Mio Yamanoue1, Akari Miyawaki1, Junpei Matsuoka2, Yasutomo Yamamoto1 (1. Doshisha Women's College of Liberal Arts, 2. Kindai University)

[30P-pm017S]Diastereocontrolled synthesis of spirocyclopentanones using chiral molecular recognition under equilibrium condition

○Karen Hayashi1, Kei Kitamura1, Hiroto Kaku1 (1. Fac. Pharm. Sci., Tokushima Bunri Univ.)

[30P-pm018S]Pd-Catalyzed Intramolecular Cyclization–Thiocarbonylation
Cascade Using Thioesters

○Ryunosuke Ito1 (1. ASE. Waseda Univ.)

[30P-pm019]6-Iodo-2-pyridone-catalyzed ester aminolysis through acid-base double activation mechanism

○Takeshi Yamada1, Nanako Tsuji1, Mioko Nasu1, Shiori Itami1, Tomoe Kometani1, Manabu Hatano1 (1. Kobe Pharmaceutical Univ.)

[30P-pm020S]Regio- and enantioselective bromocyclization of difluoroalkenes enabled by Lewis/Brønsted base concerted catalysis with chiral bisphosphine oxide

○Ryo Hirokawa1, Yuki Nakahara2, Shotaro Uchida1, Kenji Yamashita1,2, Yoshitaka Hamashima1,2 (1. Grad. Sch. Pharm. Sci., Univ. of Shizuoka, 2. Sch. Pharm. Sci., Univ. of Shizuoka)

[30P-pm021S]Synthetic study of pendant of Tebipenem Pivoxil

○Noa Fujiwara1, Mayu Iida1, Yumeno Yoshihara1, Chihiro Shimizu1, Mai Yamamoto1, Kee Nishio1, Kazuhiko Hayashi1 (1. Kinjo Gakuin University)

[30P-pm022S]Ring expansion of 1,3-indandione-derived spirocyclopropanes with sulfur ylide

○Rika Sakai1, Hikaru Fujii1, Hiroki Iwasaki1, Hisanori Nambu1 (1. Kyoto Pharm. Univ.)

[30P-pm023S]Asymmetric Fluoro-Ether Cyclization of Enamides under Dicarboxylate Phase-Transfer Catalysis

○Chihiro Kanefusa1, Lio Kurihara2, Hiromichi Egami1,2, Yoshitaka Hamashima1,2 (1. Grad. Sch. Pharm. Sci., Univ. of Shizuoka, 2. Sch. Pharm. Sci., Univ. of Shizuoka)

[30P-pm024S]Dearomative C-C bond cleavage reaction of benzyl alcohols using hypervalent iodine(III) reagents

○Takeru Nakamura1, Koshi Higashiyama1, Haruka Taniguchi1, Hideyasu China2, Toshifumi Dohi1 (1. College of Pharmaceutical Sciences, Ritsumeikan University, 2. Faculty of Bioscience, Nagahama Institute of Bio-Science and Technology)

[30P-pm025S]Synthesis of multi-substituted pyrrolidines by Hofmann–Löffler-type cyclization of optically active amines

○Yuita Tanaka1, Hirotaka Sasa2, Kotaro Kikushima1, Toshifumi Dohi1 (1. Ritsumeikan Univ, 2. Mukogawa Women's Univ)

[30P-pm026S]Synthesis of Benzoazepinones by Sequential Coupling with Hypervalent Iodine Reagents

○Arisu Kasai1, Naoki Miyamoto2, Kotaro Kikushima1, Yasuyuki Kita3, Toshifumi Dohi1,3 (1. College of Pharmaceutical Sciences, Ritsumeikan University, 2. Grad. Sch. Pharm. Sci., Ritsumeikan Univ., 3. Research Organization of Science and Technology, Ritsumeikan University)

[30P-pm027S]Oxidative Decarboxylation of 4-Hydroxybenzoic acids using Hypervalent Iodine(III) Reagent and Bromide Salt

○Koyo Onoda1, Sae Matsumoto1, Hiromi Hamamoto1 (1. Fac. Agr., Meijo Univ.)

[30P-pm028S]Synthesis of Bromofuranone via Oxidative Decarboxylation of 2-Furancarboxylic acid

Hiromi Hamamoto1, ○Kasumi Kato1, Fumiaki Kato1, Ukako Inukai1 (1. Fac. Agr., Meijo Univ.)

[30P-pm029S]Mechanochemical Synthesis of Cyclic Carbonate Derivatives

○Naohito Tomita1, Takashi Ikawa1, Hironao Sajiki1 (1. Gifu Pharm. Univ.)

[30P-pm030S]Synthesis of cyclic acetals by gold and Lewis acid-promoted cascade ring opening-cyclization of alkynylazetidines with phenols

○Toya Kariya1, Yoshida Masahiro1 (1. Faculty of Pharmaceutical Sciences, Tokushima Bunri University)

[30P-pm031S]Dearomative enantio- and siteselective fluorination of hydroxy pyridine derivatives

○Kousuke Sakimoto1, Hiromichi Egami1, Yoshitaka Hamashima1 (1. Grad. Sch. Pharm. Sci., Shizuoka Univ.)

[30P-pm032S]Construction of 1,4-oxazepine skeleton by palladium-catalyzed cascade cyclization of propargylic carbonates

○Akira Kurosaka1, Shiomi Shinya1, Yoshida Masahiro1 (1. Fac. of Pharm. Sci., Tokushima Bunri Univ.)

[30P-pm033S]Pyrroloindoline synthesis by palladium-DHTP-catalyzed C3-selective arylation/cyclization of tryptamine derivatives

○Haruna Jimbo1, Miyuki Yamaguchi1, Hideyuki Konishi1, Kei Manabe1 (1. Univ. of Shizuoka)

[30P-pm034]Bi-directional nitroaldol reaction -Studies on substrate and stereoselectivity-

○Erika Iwasaki1, Yoko Asakura1, Momo Sakai1, Yusuke Akagi1, Toshiya Komatsu1 (1. Fac. Pharm. Sci., Teikyo Heisei Univ.)

[30P-pm035S]Fluorination reaction of 1-Azabicyclo[1.1.0]butane (ABB)

○Mayu Iida1, Noa Fujiwara1, Yumeno Yoshihara1, Chihiro Shimizu1, Mai Yamamoto1, Kee Nishio1, Kazuhiko Hayashi1 (1. Kinjo Gakuin University)

[30P-pm036S]Synthesis of a nitroxyl-radical catalyst having methoxymethyl groups at the α-position and its application to the mechanistic studies of the oxidation of silyl ethers

○Ryosuke Arai1, Kaori Sakamoto1, Eri Miyazaki1, Yusuke Kobayashi1, Takumi Furuta1, Shohei Hamada1 (1. Kyoto Pharmaceutical University)

[30P-pm037]Elucidation of the stereocontrol mechanisms of chemical and enzymatic intramolecular Diels-Alder cycloaddition reactions for the formation of bioactive decalins

Takumi Kariya1, Hayato Hasegawa2, Taro Udagawa3, Mieko Tsuji1, Yusaku Inada1, Shingo Nagano2, Naoki Kato4, Tatsuo Suzutani5, Tasuku Hirayama1, ○Hideko Nagasawa1 (1. Gifu Pharm. Univ., 2. Grad. Sch. Eng. Tottori Univ., 3. Gifu Univ., 4. Agric. Setsunan Univ., 5. Fukushima Med. Univ.)

[30P-pm038S]Origin of large secondary kinetic isotope effect in deuterium labeling of chiral phase-transfer catalyst

○Sei Murayama1, Hiroshi Naka1,2 (1. Grad. Sch. of Pharm. Sci., Kyoto Univ., 2. CPiER-DSR, Kyoto Univ.)

[30P-pm039]Molecular behavior and properties in aqueous solutions of β-cyclodextrin derivative with secondary hydroxy groups of two adjacent glucose units being heterobifunctionalized

○Kazutaka Koga1, Shun Yasunaga2, Makoto Fukudome2, De-Qi Yuan2 (1. Fac. Pharm., Daiichi Univ. of Pharm., 2. Fac. Pharm. Sci., Kobe Gakuin Univ.)

[30P-pm040S]Inclusion and selectivity of cyclic ethers and esters by a disubstituted adamantane bearing nitrophenol

○Hayahide Makino1, Masahide Tominaga1, Masatoshi Kawahata2, Kentaro Yamaguchi1 (1. Tokushima Bunri Univ.,Pharm.Sci.Kagawa., 2. Showa Pharmaceutical Univ.)

[30P-pm041S]Structural analysis of co-inclusion crystals with two types of host molecules

○Ryusei Kamada1, Masahide Tominaga1, Tadashi Hyodo1, Kentaro Yamaguchi1 (1. Tokushima Bunri Univ.,Pharm.Sci.Kagawa.)

[30P-pm042]Mechanism of Chiral Recognition of Diketopiperazines containing Proline Residues using (-)-Epigallocatechin-3-O-gallate

○Takashi Ishizu1, Yuka Fujitani1, Haruka Kamei1, Runa Nishio1 (1. Faculty of Pharmacy and Pharmaceutical Sciences, Fukuyama University)

[30P-pm043]Characterization of drug inclusion behavior by using porous crystals of halogen-containing cyclic compounds

○Tadashi Hyodo1, Masahide Tominaga1, Kentaro Yamaguchi1 (1. Tokushima Bunri Univ., Pharm. Sci. Kagawa.)

[30P-pm044S]The synthesis and gelation abilities evaluation of amphiphilic bis-urea

○Minami Ishii1, Shinya Kimura1, Masashi Yokoya1, Masamichi Yamanaka1 (1. Meiji Pharm. Univ.)

[30P-pm045S]Synthesis of Cyclic Monourea and Gelation by Ring-Opening Reaction

○Noriaki Kimishima1, Shinya Kimura1, Masashi Yokoya1, Masamichi Yamanaka1 (1. Meiji Pharm. Univ.)
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