[31P-am] Total synthesis 2/Chemical reaction development 3/ Other synthetic studies 3 | The 144th Annual Meeting of the Pharmaceutical Society of Japan (Yokohama)

The 144th Annual Meeting of the Pharmaceutical Society of Japan (Yokohama)

Session Details

Poster Presentation(A) Pharmaceutical Chemistry

Total synthesis 2/Chemical reaction development 3/ Other synthetic studies 3

Sun. Mar 31, 2024 8:30 AM - 12:00 PM JST
Sun. Mar 31, 2024 11:30 PM - 3:00 AM UTC

[Poster 1] Exhibition Hall AB (1F)

[31P-am001S]Synthetic studies on dinapinones A1 and A2

Ayumi Ueno¹, ○Daiki Eto¹, Daiki Lee¹, Shiho Arima¹, Taichi Ohshiro¹, Ryuji Uchida², Hiroshi Tomoda¹, Tohru Nagamitu¹ (1. Sch. Pharm, Kitasato Univ., 2. Facul. Pharm. Sci., Tohoku Med. Pharm. Univ.)

[31P-am002S]Synthetic study of ellagic acid derivatives with Hes1 dimer inhibition

○Daiki Kawabata¹, Midori A. Arai¹ (1. Fac. Sci. Tec., Keio Univ.)

[31P-am003S]Synthetic study on celludinone B

○Shunya Shiraki¹, Tomoka Sato¹, Taichi Ohshiro¹, Hiroshi Tomoda¹, Tohru Nagamitsu¹ (1. Sch. Pharm., Kitasato Univ.)

[31P-am004]Total synthesis of entonalactam B isolated from the fungi belonging to the Xylariaceae family

○Hitoshi Kamauchi¹, Yoshiaki Sugita¹ (1. Faculty of Pharmaceutical and Sciences Josai University)

[31P-am005S]Asymmetric total synthesis of β-carboline alkaloid (S)-brevicolline and its derivatives.

○Koharu Sakoguchi¹, Ruka Kamimoto¹, Takashi Nishiyama¹, Yuka Nagatsuka(Handa)¹, Yuki Sato¹, Noriyuki Hatae², Tominari Choshi¹ (1. Fukuyama Univ., 2. Yokohama Univ of Pharmacy.)

[31P-am006S]Total synthesis of staurosporinone by cyclocarbonylation reaction.

○Shunsuke Doi¹, Takasi Nishiyama¹, Toshio Motoyashiki¹, Noriyuki Hatae², Tominari Choshi¹ (1. Fukuyama univ., 2. Yokohama univ.)

[31P-am007S]Synthesis of β-carboline alkaloid evollionine A.

○Rinya Asano¹, Takashi Nishiyama¹, Tominari Choshi¹ (1. Fukuyama University)

[31P-am008S]Total synthesis of calothrixin B and its analogs.

○Takumi Ueda¹, Takashi Nishiyama¹, Toshio Motoyashiki¹, Noriyuki Hatae², Tominari Choshi¹ (1. Fukuyama University, 2. Yokohama University of Pharmacy)

[31P-am009S]Total synthesis indolo[3,2-a]carbazole alkaloid racemosin B.

○Yuta Uchida¹, Takashi Nishiyama¹, Nanaka Fukada¹, Tominari Choshi¹ (1. Fukuyama University)

[31P-am010S]Development and research of a novel pyrrolo[2,3-c]carbazole skeleton construction method targeting Dictyodendrin B.

○Soma Tsuji¹, Takashi Nishiyama¹, Noriyuki Hatae², Tominari Choshi¹ (1. Fukuyama University, 2. Yokohama University of Pharmacy)

[31P-am011]Synthesis of benzimidazole-4,7-dione and evaluation of antitumor activity

○nishiyama takashi¹, Ryoya Shono¹, Toshio Motoyashiki¹, Noriyuki Hatae², Tominari Choshi¹ (1. Fukuyama Univ., 2. Yokohama Univ. Pharm.)

[31P-am012]Total Synthesis of (+)-Monocillin II

Naoki Kokaji¹, Naru Ishikura¹, Akinobu Matsuzawa¹, ○Shogo Kamo¹, Kazuyuki Sugita¹ (1. Hoshi Univ.)

[31P-am013S]Convergent total syntheses of corallocins A–C

○Kazuki Hori¹, Tomoya Mashiko¹, Shunsuke Onuma¹, Yuta Nakazato¹, Yuta Katsumura¹, Akihiko Kasamatsu¹, Shinya Adachi¹, Akinobu Matsuzawa¹, Shogo Kamo¹, Kazuyuki Sugita¹ (1. Hoshi Univ.)

[31P-am014S]Total syntheses of furanocoumarins

○Yuko Kotaka¹, Masaya Nakajima^2,3, Tetsuhiro Nemoto³ (1. Fac. Pharm. Sci., Chiba Univ., 2. Grad. Sch. Pharm. Sci., Univ. Tokyo., 3. Grad. Sch. Pharm. Sci., Chiba Univ.)

[31P-am015S]Total Synthesis of (±)-Minimiflorin Oriented to Na⁺/K⁺-ATPase Inhibitors

○Wataru Yamawaki¹, Hiroshi Aoyama², Makoto Sako², Kenichi Murai², Kuniaki Suzuki³, Mitsuhiro Arisawa² (1. School of Pharmaceutical Sciences, Osaka University, 2. Graduate School of Pharmaceutical Sciences, Osaka University, 3. Graduate School of Dental Medicine, Hokkaido University)

[31P-am016S]Synthesis of meso-Cyanoporphyrins Using Electrochemical Method

○Ayane Mizunuma¹, Satoshi Hayashi¹, Masahiro Noji¹, Toshikatsu Takanami¹ (1. Meiji Pharmaceutical Univ.)

[31P-am017S]Synthesis of Benzaldehyde Bearing a Stable Boronic Acid Ester Group

○Kota Kawase¹, Satoshi Hayashi¹, Masahiro Noji¹ (1. Meiji Pharmaceutical Univ.)

[31P-am018S]Electrogenerated Acid-Catalyzed Domino Substitution/Cyclization for the Synthesis of Tetrahydroquinolines

○Kakeru Maeda¹, Tsugumi Abe¹, Satoshi Hayashi¹, Masahiro Noji¹ (1. Meiji Pharmaceutical Univ.)

[31P-am019S]Electrogenerated Acid-Catalyzed Dehydrative Substitution of Benzylic Alcohols with Sulfonamides

○Yuki Nakayama¹, Satoshi Hayashi¹, Masahiro Noji¹ (1. Meiji Pharmaceutical Univ.)

[31P-am020S]Electrochemical Mono-Chlorination of Porphyrins

○Kouki Katou¹, Satoshi Hayashi¹, Seiya Yamashita¹, Toshikatsu Takanami¹, Masahiro Noji¹ (1. Meiji Pharmaceutical Univ.)

[31P-am021S]Electrochemical Regioselective meso-Tiocyanation of Porphyrins

○Kodai Takayama¹, Satoshi Hayashi¹, Masahiro Noji¹ (1. Meiji Pharmaceutical Univ.)

[31P-am022]Hypervalent iodine-catalyzed oxidative C(sp³)–H amination for the synthesis of δ-lactam derivatives

○Hirotaka Sasa¹, Miki Okada¹, Manaka Tanigawa¹, Tomoka Higuchi¹, Takuya Matsumoto¹, Minoru Ozeki¹, Toshifumi Dohi², Ikuo Kawasaki¹ (1. Department of Pharmacy, Mukogawa Women's University, 2. College of Pharmaceutical Sciences, Ritsumeikan University)

[31P-am023S]A Copolymer Catalyst Capable of Molecular Recognition

Yusuke Kuroda^1,2, ○Yusei Fujii¹, Kiyosei Takasu¹ (1. Grad. Sch. Pharm. Sci., Kyoto Univ., 2. The Hakubi Center for Advanced Research)

[31P-am024S]Asymmetric construction of chiral phosphorous center by using chiral sulfonamide

○Yurika Kambara¹, Ayase Matsumoto¹, Sayaka Yamada¹, Mizuki Nakamoto¹, Miku Murata¹, Sakura Nakai¹, Tomoe Ishiura¹, Akari Miyawaki¹, Junpei Matsuoka², Yasutomo Yamamoto¹ (1. Doshisha Women's College of Liberal Arts, 2. Kindai University)

[31P-am025]Synthesis of 2-(2-piperidinyl)indole analogues for use in the catalytic synthesis of 9-hydroxyphenalenone

○Hirokazu Tsukamoto^1,2, Jun Nakamura¹, Keiko Suzuki¹, Shota Shigematsu¹, Hina Ikekame¹, Ayane Ikeda¹, Yumi Nomura², Takayuki Doi² (1. Dept. Pharm. Sci., Yokohama Univ. Pharm., 2. Grad. Sch. Pharm. Sci., Tohoku Univ.)

[31P-am026S]Rapid N-Alkylation of N-Sulfonylcarbamates with Alkyl Chloroformate.

○Mao Kawata¹, Yusuke Takahashi¹, Tomoki Takagi¹, Yusuke Kasai¹, Hiroshi Imagawa¹ (1. Faculty of Pharmaceutical Sciences, Tokushima Bunri University)

[31P-am027S]Gold-Catalyzed Synthesis of Cyclobutanes

○Hitomi Chiaki¹, Naho Ishii¹, Nobuyoshi Morita¹, Yoshimitsu Hashimoto¹, Osamu Tamura¹ (1. Showa Pharm. Univ.)

[31P-am028S]Intramolecular [2+2] photocycloaddition of enone

Yousuke Yamaoka^1,2, Shingo Minamikawa², ○Shoei Nakamura¹, Hideto Miyabe¹, kiyosei Takasu² (1. Sch. of Pharm. Hyogo Med. Univ. , 2. Grad. Sch. Pharm. Sci. Kyoto Univ.)

[31P-am029]Practical Selective Monooxidation Reactions of Symmetric Dialdehydes in Mainly Aqueous Solvents

Pullaiah Kattanguru¹, Ren Ogawa¹, Yutaro Suzuki¹, ○Satomi Niwayama¹ (1. Muroran Institute of Technology)

[31P-am030]Study of the Petasis reaction using alkanediones

○Shigeo Sugiyama¹, Yumi Ikegami¹, Yu Shirahama¹, Ryo Hashimoto¹, Motoki Ito¹, Kazuhiro Higuchi¹ (1. Meiji Pharm. Univ.)

[31P-am031S]Study of the Petasis reaction using cyclic alkanedione; two-step synthesis of Tiletamine

○Yuka Yahata¹, Kae Saitou¹, Airi Morita¹, Sakura Yamada¹, Haruka Taki¹, Motoki Ito¹, Kazuhiro Higuchi¹, Shigeo Sugiyama¹ (1. Meiji Pharm. Univ.)

[31P-am032S]Synthesis of 1,5-Diketones by Metal-Free Enyne Cycloisomerization

○Hiroto Hashi¹, Shoyo Ho¹, Akira Tsubouchi¹, Akio Saito¹ (1. Grad. Sch. Eng., Tokyo Univ. Agric. Tech.)

[31P-am033S]Selective synthesis of superacidic carbon acids through the reaction of simple alkenes with 1,1-bis(triflyl)ethylene

Shoki Hoshikawa¹, ○Leon Sano¹, Takashi Matsumoto¹, Hikaru Yanai¹ (1. Tokyo Univ. Pharm. Life Sci.)

[31P-am034]Organocatalytic Enantioselective Decarboxylative Aldol Reaction

○Takuya Kanemitsu¹, Kazuhiro Nagata², Kiyoshi Fukuhara², Kenichi Nakamura¹, Tetsuo Yamasaki¹ (1. School of Pharmaceutical Sciences, Kyushu University of Health and Welfare, 2. School of Pharmacy, Showa University)

[31P-am035]2,4-trans selective acetalization of 1,2-diols derived from glycerol

○Ryuji Kyan¹, Tatsuki Sera¹, Nono Kawachi¹, Akira Shigenaga¹ (1. Fac. Pharm. and Pharm. Sci., Fukuyama Univ.)

[31P-am036]Development of Metal-Free Oxidative Amination Reaction of Aromatic Compound with Heteroatom

○koji morimoto^1,2, Kana Yanase¹, Sana Kanemitsu¹, Kentaro Toda¹, Hitoshi Takeuchi¹, Toshifumi Dohi^1,2, Yasuyuki Kita² (1. College of Pharmaceutical Sciences, Ritsumeikan University, 2. Research Organization of Science and Technology, Ritsumeikan University)

[31P-am037S]Novel conversion method of cyclopentane-1,3-dione moiety: Construction of 5/5/4 tricyclic systems and its mechanistic studies

○Makoto Kobayashi¹, Tomonari Sasage², Keiji Tanino³, Seiichi Nakamura¹, Kazutada Ikeuchi¹ (1. Grad. Sch. Pharm. Sci., Nagoya City Univ., 2. Grad. Sch. Chem. Sci. Engine., Hokkaido Univ., 3. Fac. Sci., Hokkaido Univ.)

[31P-am038]Synthesis of indoxyl derivatives by indolin-2,3-acetonides

○Tetsu Tsubogo¹, Tatsuya Furube¹, Karen Sato¹, Koji Yamada¹ (1. Health Sciences Univ. of Hokkaido)

[31P-am039S]Development of red-light-driven radical cyclization reaction catalyzed by zinc porphyrin catalyst and its application to natural product synthesis

○Yusuke Okanishi¹, Otoki Takemoto¹, Sanpou Kawahara¹, Satoshi Hayashi², Toshikatsu Takanami², Takehiko Yoshimitsu¹ (1. Grad. Sch. Pharm. Sci., Okayama Univ., 2. Meiji Pharm. Univ.)

[31P-am040S]γ-Selective Aldol Condensation Using β-Diketones

○Rina Tanaka¹, Kyosuke Sugihara², Hitoshi Abe² (1. Fac. Eng., Toyama Univ., 2. Grad. Sch. Sci. and Eng., Toyama Univ.)

[31P-am041S]Development of N-N cross coupling reaction between carbazoles and acridones by using NaOCl･5H₂O

○Natsuko Momiyama¹, Mirei Ueda¹, Keisuke Yoshida¹, Shinji Kitagaki¹ (1. Meijo University)

[31P-am042S]Development of pyridine N-oxide catalyzed dimesylation of epoxides via ring-opening
reaction

○Saki Hasegawa¹, Kana Hashimoto¹, Keisuke Yoshida¹, Shinji Kitagaki¹ (1. Meijo University)

[31P-am043S]Effect of β-alkoxy group on electron-deficient alkene on the regioselectivity in the phosphine-catalyzed (2+3) annulation reaction of allenoates

○Kyoka Kishimoto¹, Daiki Uchida¹, Ayane Nishino¹, Akane Uchida¹, Hiroto Takeuchi¹, Hiroshi Aoyama², Keisuke Yoshida¹, Shinji Kitagaki¹ (1. Meijo University, 2. Graduate School of Pharmaceutical Sciences, Osaka University)

[31P-am044S]Photoinduced Diels-Alder reaction of benzocyclobutenone

○Yukiko Ikeda¹, Masaru Tanioka¹, Yuji Matsuya¹ (1. Faculty of Pharm. Sci., University of Toyama)

[31P-am045S]Design, Synthesis and Evaluation of Photoresponsive Propertied of Chiral Macro Cyclic Compounds Containing an Azobenzene-unit.

○Shotaro Otaki¹, Ryota Shibauchi¹, Toshifumi Tojo¹, Norio Tanada³, Yoshiyuki Kageyama³, Shin Aoki^1,2 (1. Grad. Sch. Pharm. Sci., Tokyo Univ. of Science., 2. Res. Inst. for Sci., Tokyo Univ. of Science., 3. Grad. Sch. Sci., Hokkaido Univ.)

[31P-am046]Synthetic Studies on Novel 4-HydroxypyrazoleDerivatives by Ring Transformation of Pyrazole-Propargyl Alcohols (3)

○Takafumi Fujita¹, Eiichi Masumoto¹, Fumi Okabe-Nakahara¹, Hiroshi Maruoka¹ (1. Fac. Pharm. Sci., Fukuoka Univ.)

[31P-am047]Synthetic Studies of Novel Spiro[benzoxazine-2,4′-pyrazole] Derivatives

○Eiichi Masumoto¹, Mai Horioka¹, Takafumi Fujita¹, Fumi Okabe-Nakahara¹, Hiroshi Maruoka¹ (1. Fac. Pharm. Sci., Fukuoka Univ.)

[31P-am048S]Synthetic Studies of fused Tricyclic Pyrazolo[3,4-b]pyridine Derivatives.

Fumi Okabe-Nakahara¹, ○Minori Konta¹, Takafumi Fujita¹, Eiichi Masumoto¹, Hiroshi Maruoka¹ (1. Fac. Pharm. Sci., Fukuoka Univ.)

[31P-am049S]Synthetic Studies of fused Tricyclic Pyrido[2,3-d]pyrimidine Derivatives.

Fumi Okabe Nakahara¹, ○Mari Kobayashi¹, Takafumi Fujita¹, Eiichi Masumoto¹, Hiroshi Maruoka¹ (1. Fac. Pharm. Sci., Fukuoka Univ.)

[31P-am050S]Synthetic Studies of fused Tricyclic Pyrazolo[3,4-b]pyridine Derivatives.

Fumi Okabe-Nakahara¹, ○Nanako Shimizu¹, Ayaka Ide¹, Ayano Kabu¹, Takafumi Fujita¹, Eiichi Masumoto¹, Hiroshi Maruoka¹ (1. Fac. Pharm. Sci., Fukuoka Univ.)

[31P-am051S]Synthetic Studies of fused Tricyclic Pyrrolo[2,3-b]pyridine Derivatives.

Fumi Okabe Nakahara¹, ○Sayako Jimi¹, Takafumi Fujita¹, Eiichi Masumoto¹, Hiroshi Maruoka¹ (1. Fac. Pharm. Sci., Fukuoka Univ.)

[31P-am052S]Exploration of novel anti-human cytomegalovirus agent based on the structure of Sophovicine B

○Daiki Suzuki¹, Ayaka Ishiyama¹, Yoshihiro Natori¹, Asako Kaise¹, Yuichi Yoshimura¹ (1. Faculty of Pharmaceutical Sciences, Tohoku Medical and Pharmaceutical University)

[31P-am053S]Development of new discriminative color test reagents for cannabis extracts.

○Hikari Nishiguchi¹, Kayo Nakamura¹, Riho Hamajima¹, Hidetsugu Tabata², Tetsuta Ositari², Hideaki Natsugari³, Hideyo Takahashi¹ (1. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2. Faculty of Pharma-Science, Teikyo University, 3. Faculty of Pharmaceutical Sciences, The University of Tokyo)

[31P-am054S]Development of the synthetic method of peptide analogs bonded at amino group site of amino acids

○Ryusei Uozumi¹, Takashi Kano¹, Norihiro Tada¹, Akichika Itoh¹ (1. Gifu Pharmaceutical University)

[31P-am055S]Creation of Bioactive Substances with Flavonoid Skeletons

○Mayu Hiromori¹, Ayaka Fujimura², Hiroki Suzuki², Yuma Tsujimura², Mami Watano², Ayumi Imayoshi², Masaharu Shin-Ya³, Maiko Nakashio³, Eriko Ohgitani³, Osam Mazda³, Kazunori Tsubaki² (1. Faculty of Life and Environment, Kyoto Prefectural University, 2. Graduate School of Life and Environmental Science, Kyoto Prefectual University, 3. Department of Immunology, Kyoto Prefectural University of Medicine)

[31P-am056]Nucleophilic substitution versus β-elimination of β-hydroxyesters in Mitsunobu reaction and choline phosphate esterification

○Takayasu YAMAUCHI¹, Mayu Shimizu¹, Ayano Shiragiyama¹, Manaka Fukuda¹ (1. Hoshi Univ.)

[31P-am057S]Synthesis of organic fluorescent dyes bearing a nitrogen ylide-based group that exhibits strong π-electron donating ability

○Naoto Kuchiki¹, Hikaru Fujita¹, Takanari Arai¹, Munetaka Kunishima^1,2 (1. Faculty of Pharmaceutical Sciences, Institute of Medical, Pharmaceutical, and Health Sciences, Kanazawa University, 2. Faculty of Pharmaceutical Sciences, Kobe Gakuin University)

[31P-am058]Synthesis of β,β’,β’’-trifluoro-tert-butyl ethers/thio ethers as a novel partial fluorinated motif

○atsushi tarui¹, David O'Hagan² (1. Pharm. Sci., Setsunan Univ., 2. Univ. St Anderws)

[31P-am059S]Development of recyclable chiral phosphoric acid catalyst bearing hydrophobic anchor

○Shoya Nakamura¹, Haruna Aozaki¹, Tsubasa Inokuma¹, Kenichi Yamada¹ (1. Sch. Pharm. Sci., tokushima Univ.)

[31P-am060S]Utility of the epoxide ring-opening reaction and efficiency of the synthetic route for the cyclic polyglycerol synthesis

○Mizuki Noda¹, Yu Saeki¹, Noriyuki Nakajima^1,2, Yasuhito Koyama^1,2, Masahiro Hamada^1,2 (1. Toyama Pref. Univ., 2. Biotech. Res. Center, Toyama Pref. Univ.)