Presentation Information
[2B-3-02]Identification of ALDH1A1 covalent inhibitor by metabolic phenotypic screening and its application for RIPTAC
*Shohei Uchinomiya1, Rui-kan Yin1, Kazuya Inoue1, Saki Inoue1, Emi Mishiro2, Akinobu SENOO1, Jose Caaveiro1, Naoya Matsunaga1, Akio Ojida1 (1. Graduate School of Pharmaceutical Sciences, Kyushu University, 2. Institute of Transformative Bio-Molecules, Nagoya University)
Keywords:
phenotypic screening,fatty acid beta oxidation,covalent inhibitor,ALDH1A1,RIPTAC
