Presentation Information
[3A-1-01]GPCR chemogenetics for enhancing the therapeutic potential of approved inhibitors
*Yuma Matsuoka1, Tomohiro Doura1, Yoshifumi Ueda2, Duy Phuoc Tran3, Hidetsugu Asada4, Haruki Omatsu2, Tatsuki Hori3, So Iwata4,5, Akio Kitao3, Nobuaki Takahashi2, Shigeki Kiyonaka1,6 (1. Graduate School of Engineering, Nagoya University, 2. Graduate School of Engineering, Kyoto University, 3. School of Life Science and Technology, Science Tokyo, 4. Graduate School of Medicine, Kyoto University, 5. Graduate School of Biostudies, Kyoto University, 6. Research Institute for Quantum and Chemical Innovation, Nagoya University)
Keywords:
Chemogenetics,GPCR,approved inhibitors,tumor microenvironment,A2AR
