The 143rd Annual Meeting of the Pharmaceutical Society of Japan (Sapporo)
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Session Details

Poster Presentation(A) Pharmaceutical Chemistry

[28P1-am1]Chemical reactions/Reaction mechanism/Structure and physical property/Molecular recognition/Others

Tue. Mar 28, 2023 9:00 AM - 10:40 AM JST
Tue. Mar 28, 2023 12:00 AM - 1:40 AM UTC
[Room P1] Gymnasium 1F

[28P1-am1-001]Synthetic method of ynamides through copper-catalyzed diynylation and cycloaddition

○Norihiro Tada1, Akichika Itoh1 (1. Gifu Pharmaceutical University)

[28P1-am1-002S]Development of Regioselective Iodocyclization

○Junya Hirai1, Rikuto Iizuka2, Daiki Lee1, Tohru Nagamitsu1 (1. Grad. Sch. Pharm. Sci., Kitasato Univ, 2. Sch. Science. Sci., Kitasato Univ)

[28P1-am1-003S]Enantioselective Henry reaction catalyzed by copper (II) complexes of multivalent chiral amines

Kenji Yatsuzuka1, ○Ayana Mori1, Chika Sawada1, Midori Kawasaki2, Ryuichi Shirai2 (1. Fac. Pharm. Sci., Doshisha Women's Col., 2. Grad. Sch. Pharm. Sci., Doshisha Women's Col.)

[28P1-am1-004S]Design of Novel Chiral Lithium Amides and
Application to Kinetic Optical Resolution of Racemic Ibuprofen

Midori Kawasaki1, ○Mizuki Fukuda2, Saki Horioka2, Kenji Yatsuzuka2, Ryuichi Shirai1 (1. Grad. Sch. Pharm. Sci., Doshisha Women's Col., 2. Fac. Pharm. Sci., Doshisha Women's Col.)

[28P1-am1-005]Simple immobilization of catalyst by microwave and Flow reaction

○Syunsuke Tenma1, Takuya Iwamura1, Yuhei Saitou1, Yasuyo Mitsutaki1, Kento Sekizuka1, Nami Kawasaki1, Ran Higashisanjou1, Toshinori Nakakita1, Syoji Aoki2, Sigeki Isomura1, Yasuo Sato1 (1. Yokohama University of Pharmacy, 2. E.C.E)

[28P1-am1-006]Aerobic Cross-Dehydrogenative Coupling of Catechols with Persistent Radicals

○Yoshihiro Sohtome1,2, Masumi Sugawara1, Miki Sawamura1, Mai Akakabe1,2, Boobalan Ramadoss2, Mikiko Sodeoka1,2 (1. RIKEN CPR, 2. RIKEN CSRS)

[28P1-am1-007]Synthesis of 2-Imidefuran and 5-Imide-1H-Pyrazole by N-Alkynylimide

○keiji konishi1, Yuta Ino1, Noriko Okamoto1, Takuya Sueda1 (1. Hiroshima International University)

[28P1-am1-008]Efficient Lactam Synthesis using PO(OCH2CF3)3/NaH

○Shota Asai1, Hoshimi Nishimura1, Keigo Kitada1 (1. Fac. of Sci. and Eng., Iwate Univ.)

[28P1-am1-009S]Chemoselective hydrolysis of hydrazone carbamates: its applications for a carbamate-type protecting group for alcohols

○Yui Yoshida1, Yasuhiro Nisikawa1, Momoka Andou1, Mari Momose1, Mayuko Utou1, Osamu Hara1 (1. Meijo Univ)

[28P1-am1-010S]Development of a derivatization method for triazinedione compounds by substitution of the phenoxy group

○Daichi Shimada1, Hikaru Fujita1, Jotaro Kudo1, Ririka Seto1, Munetaka Kunishima1 (1. Faculty of Pharmaceutical Sciences, Institute of Medical, Pharmaceutical, and Health Sciences, Kanazawa University)

[28P1-am1-011S]Phosphazene base-catalyzed intramolecular hydroamination with amide

○Yumika Fujimoto1, Akari Miyawaki1, Junpei Matsuoka1, Yasutomo Yamamoto1 (1. Faculty of Pharmaceutical Sciences, Doshisha Women's College of Liberal Arts)

[28P1-am1-012S]Investigation of piperidine ring construction with silver(I) ions

○Nodoka Onodera1, Riku Sato1, Imaizumi Haruki1, Hiroka Sato1, Koichi Narita1, Yuichi Yoshimura1, Kazuhiro Watanabe1 (1. Fac. Pharm. Sci., Tohoku Med. & Pharm. Univ.)

[28P1-am1-013]Synthesis of pentasubstituted 2-aryldihydropyrimidines by Pd-catalyzed/Cu-mediated Liebeskind-Srogl-type cross-coupling reaction

○Yoshio Nishimura1, Kubo Takanori2, Shibuya Nanami1, Shibukawa Ryui1, Cho Hidetsura3 (1. Sch. Pharm. Sci., Ohu Univ., 2. Fac. Pharm., Yasuda Women's Univ., 3. Grad. Sch. Pharm. Sci., XXXX Univ.)

[28P1-am1-014S]The synthesis of chiral spiro oxindoles via oxidative spiro lactonization

○Yuichi Okuaki1, Kosuke Nakashima1, Yasuyuki Matsushima1, Shin-ichi Hirashima1, Tsuyoshi Miura1 (1. Tokyo University of Pharmacy and Life Sciences)

[28P1-am1-015S]Abnormal Strecker reaction of 3-formylindole and synthetics study of Nakijinamine B

○Tomohiro Yazawa1, Masaya Nakajima1, Tetsuhiro Nemoto1 (1. Grad. Sch. Pharm. Sci., Chiba Univ.)

[28P1-am1-016]Interrupted Passerini/ Joullié-Ugi cascade reaction to access highly functionalized furoindoline catalyzed by 3,5,6-trifluoro-2-pyridone

○Takeshi Yamada1, Sentaro Okamoto1 (1. Dept. Mater. Life Chem., Kanagawa Univ.)

[28P1-am1-017S]Synthetic studies of streptonigrin based on gold-catalyzed one-pot synthesis of polysubstituted pyridines

○shuto kosuge1, Kenji Sugimoto1, Kiyoshi Tsuge2, Yuji Matsuya1 (1. Faculty of Pharm. Sci., University of Toyama, 2. Faculty of Sci., University of Toyama)

[28P1-am1-018]Synthetic studies on 1,5-benzoxazepine derivative by N-O bond rearrangement of N-arylisoxazolidine

○Kosaku Tanaka, III1, Motoko Nishidate1, Yoshimitsu Hashimoto1, Nobuyoshi Morita1, Osamu Tamura1 (1. Showa Pharmaceutical University)

[28P1-am1-019S]Ring-opening cyclization of spirocyclopropanes with potassium cyanate

○Hitomi Noro1, Hiroki Iwasaki1, Naoto Kojima1, Hisanori Nambu1 (1. Kyoto Pharm. Univ.)

[28P1-am1-020]Intramolecular Oxidative Cycloaddition of Aldoximes using 2-iodobenzoic acid as catalyst

○Akira Yoshimura1, Irina A Mironova 2, Mekhman S Yusubov2, Nami Ogura1, Tatsuya Suzuki1, Akio Saito3, Akiharu Ueki1 (1. Aomori Univ., 2. Tomsk Polytechnic University, 3. Tokyo University of Agriculture and Technology)

[28P1-am1-021S]Development of one-pot reaction for the synthesis of 1-aminoisoquinoline via isoquinoline N-oxide as reactive intermediate

Hiroki Iwasaki1, ○Rin Nomura1, Masayuki Yamashita1, Naoto Kojima1, Hisanori Nambu1 (1. Kyoto Pharm. Univ.)

[28P1-am1-022S]Development of the cyclization reaction with trifluoroacetamide group as radical precursor mediated by samarium(II) diiodide

Hiroki Iwasaki1, ○Kota Yoshioka1, Mako Hanaki1, Masayuki Yamasita1, Naoto Kojima1, Hisanori Nambu1 (1. Kyoto Pharm. Univ.)

[28P1-am1-023S]Asymmetric Diels-Alder reaction of tropolones with maleimides using thiourea fusedγ-amino alcohol organocatalyst

○Hayato Oda1, Zubeda Begum2, Chigusa Seki2, Yuko Okuyama3, Eunsang Kwon4, Koji Uwai2, Michio Tokiwa5, Suguru Tokiwa5, Mitsuhiro Takeshita5, Hiroto Nakano2 (1. Faculty of Science and Engineering, Muroran Institute of Technology, 2. Graduate School of Engineering, Muroran Institute of Technology, 3. Faculty of Pharmaceutical Sciences, Tohoku Medical and Pharmaceutical University, 4. Graduate School of Science, Tohoku University Research and Analytical Center for Giant Molecules, 5. Tokiwakai Group)

[28P1-am1-024S]Selective synthesis of nitrogen-doped polycyclic aromatic hydrocarbons and their optical properties

○Teru Kawazoe1, Yuto Hagiyama2, Kazumasa Funabiki2, Takashi Matsumoto1, Hikaru Yanai1 (1. Tokyo Univ. Pharm. Life Sci., 2. Fac. Eng., Gifu Univ. )

[28P1-am1-025S]Synthesis and Structural Characterization of Cyclic Compounds Containing Two Sulfonamide Structures

○Takato Koideya1, Ryuji Toshima1, Yoshiki Konno1, Takehiro Yamagishi1,2, Kyosuke Kaneda1,2 (1. Hokkaido University of Science, 2. Creation Reserch Institute of Life Science in KITA-no-DAICHI)

[28P1-am1-026]New Synthetic Methods for Bicyclic Hydantoins

○Tomoya Katakura1, Eiji Kishi2, Ryu Watanabe2, Jun-ichi Yamaguchi2 (1. Kanagawa Institute of Technology, 2. Kanagawa institute of Technology)

[28P1-am1-027S]Synthetic Method for Indolyl 2-Phosphonates by Ring Expansion of Benzocyclobutenone Oxime Sulfonates

○Yusuke Kanno1, Juri Sakata1, Hidetoshi Tokuyama1 (1. Grad. Sch. Pharm. Sci., Tohoku Univ.)

[28P1-am1-028]Halocyclization of alkenylthioester

Rinako Saegusa1, ○hiroki shigehisa1 (1. Musashino Univ.)

[28P1-am1-029]Construction of naphtho[1,8-bc]thiophene via intramolecular cyclization of allynylthioether

○Noriyuki Hatae1, Takashi Nishiyama2, Yuuki Ichikawa1, Tominari Choshi2 (1. Yokohama University of Pharmacy, 2. Faculty of Pharmaceutical Sciences, Fukuyama University)

[28P1-am1-030S]Synthesis of Multi-fused Aromatic Heterocycles by Oxidative Functionalization of Hydroquinones

○Takaaki Aijima1, Keiichiro Nakajima1, Shuji Akai1, Yoshinari Sawama1 (1. Grad. Sch. Pharm. Sci., Osaka Univ.)

[28P1-am1-031S]Enantioselective 1,3-Dipolar [6+4] Cycloaddition Reactions Using Peptide Organocatalysts

○Ayako Suzuki1, Zubeda Begum2, Chigusa Seki2, Yuko Okuyama3, Kwon Eunsaug4, Koji Uwai2, Michio Tokiwa5, Suguru Tokiwa5, Mitsuhiro Takeshita5, Hiroto Nakano2 (1. Faculty of Science and Engineering, Muroran Institute of Technology, 2. Graduate School of Engineering, Muroran Institute of Technology, 3. Faculty of Pharmaceutical Sciences, Tohoku Medical and Pharmaceutical University, 4. Graduate School of Science, Tohoku University Research and Analytical Center for Giant Molecules, 5. Tokiwa Group)

[28P1-am1-032]Environmentally Friendly Synthesis of Tetrahydrofurans by Gold Catalyst

○Nobuyoshi Morita1, Issei Shimada1, Kosaku III Tanaka1, Yoshimitsu Hashimoto1, Osamu Tamura1 (1. Showa Pharmaceutical University, Laboratory of Organic Chemistry)

[28P1-am1-033S]Gold/Platinum-Catalyzed Construction of Bicyclo[3.3.1]/[3.3.0] Ketal Skeletons

○Hitomi Chiaki1, Nobuyoshi Morita1, Kousaku Tanaka III1, Yoshimitsu Hashimoto1, Osamu Tamura1 (1. Showa Pharmaceutical University)

[28P1-am1-034S]Examination of ring opening reaction of spirocyclopropane derivatives mediated by samarium(II) diiodide

Hiroki Iwasaki1, ○Tomohito Yamashita1, Naoto Kojima1, Hisanori Nambu1 (1. Kyoto Pharm. Univ.)

[28P1-am1-035]Regioselective asymmetric reaction of furan derivatives using organocatalyst

○Hiroshi Akutsu1, Keigo Tamai1, Yutaro Toshikage1, Ryota Tominaga1, Kosuke Nakashima2, Shin-ich Hirashima2, Akihiro Yoshida1, Tsuyoshi Miura2, Takashi Yamanoi1 (1. Fac. of. Pharm. and Pharmceut. Sci., Josai Univ., 2. Pharm., Tokyo Univ. of Pharm. and Life Sci.)

[28P1-am1-036]Dehydrative amination of benzhydrols with aminopyridines utilizing Au(III)/TPPMS catalyst system in water

○Hidemasa Hikawa1, Taku Nakayama1, Shunki Nakamura1, Shoko Kikkawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)

[28P1-am1-037S]The reaction used picolinamide with aldehydes in non-polar solvent

○Taku Nakayama1, Sayaka Fujiki1, Hidemasa Hikawa1, Shoko Kikkawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)

[28P1-am1-038S]Gold(Ⅲ)-catalayzed Friedel-Crafts alkylation of nitroanilines in water

○Akane Fukuda1, Hidemasa Hikawa1, Isao Azumaya1 (1. Pharm. Sci., Toho Univ.)

[28P1-am1-039S]Synthesis of imidazopyridine via Pd-catalyzed transfer hydrogenative cascade reaction of nitropyridines with benzyl alcohols in water.

○Reita Mashimo1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)

[28P1-am1-040S]Pd-catalyzed dehydrative/decarboxylative coupling of carboxylic acids with alcohols in water.

○Naohiro Tahara1, Taku Nakayama1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)

[28P1-am1-041S]Creation and structural analysis of inclusion crystals of aromatic diimide-based macrocycles containing ketones

○Sakito Nanbara1, Masahide Tominaga1, Tadashi Hyodo1, Masatoshi Kawahata2, Kentaro Yamaguchi1 (1. Pharm. Sci., Tokushima Bunri Univ., 2. Showa Pharmaceutical Univ.)

[28P1-am1-042S]Preparation and structural elucidation of inclusion crystals built from aromatic diimide-based macrocycles and liquid guests with triple bonds

○Masahiro Uematsu1, Masahide Tominaga1, Tadashi Hyodo1, Masatoshi Kawahata2, Kentaro Yamaguchi1 (1. Pharm. Sci., Tokushima Bunri Univ., 2. Showa Pharmaceutical Univ.)

[28P1-am1-043S]Dimeric structures of molecular tweezers bearing naphthalimide and adamantane units in the crystalline state

○Tadashi Hyodo1, Kiyoe Matsui2, Masahide Tominaga1,2, Kentaro Yamaguchi1,2 (1. Grad. Sch. Pharm Sci., Tokushima Bunri Univ., 2. Pharm Sci., Tokushima Bunri Univ.)

[28P1-am1-044S]Development of non-directed C-H activation using CBS catalyst analogs as bifunctional ligand

○Miho Ibara1, Daisuke Sawada1 (1. Grad. Sch. Med. Dent. Pharm. Sci., Okayama Univ.)

[28P1-am1-045S]C-H activation cooperatively catalyzed by transition metal and bifunctional ligand

○Koki Yano1, Daisuke Sawada1 (1. Grad. Sch. Med. Dent. Pharm. Sci., Okayama Univ.)
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