Presentation Information

[2P-047]Salt bridge interaction of an arginine residue in EP4 receptor with carboxyl group of prostaglandin is required for β-arrestin activation.

Kaisei Mori, Yuki Mori, Erina Ymazaki, Saori Numata, Tosiko Sugimoto, Tomoaki Inazumi, Soken Tutiya, Yukihiko Sugimoto (Dept. Pharmaceut. Biochem., Grad. Sch. Pharm. Sci., Kumamoto Univ.)
キーテクノロジー:BRET

Keywords:

GPCR,プロスタグランジン,β-arrestin,バイアス型作動薬

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