The 145th Annual Meeting of the Pharmaceutical Society of Japan (Fukuoka)
Advanced Search

Session Details

Oral Presentation(A) Pharmaceutical Chemistry

[28-17-am]Chemical Biology 4

Fri. Mar 28, 2025 8:30 AM - 10:11 AM JST
Fri. Mar 28, 2025 11:30 PM - 1:11 AM UTC
Room 17 (MARINE MESSE FUKUOKA Hall B: Conference Room2-1 [2F])
Chair: Shinichi Sato, Kazuya Matsuo
8:30 AM - 8:42 AM JST(11:30 PM - 11:42 PM UTC)

[28-17-am01]Turn-ON type proximity labeling method for profiling intracellular protein complexes

○TAKUMI KARIYA1, Shinichi Sato2,3, Keita Nakane2,3, Mikiko Sodeoka1, Kosuke Dodo1 (1. RIKEN CSRS, 2. FRIS. Tohoku Univ., 3. Grad. Sch. Life Sciences, Tohoku Univ.)
8:42 AM - 8:54 AM JST(11:42 PM - 11:54 PM UTC)

[28-17-am02S]Studies toward tyrosine modification via oxime transfer

○Shuhei Terada1, Yuki Yamanashi1, Motomu Kanai1 (1. Grad. Sch. Pharm. Sci., The Univ. of Tokyo)
8:54 AM - 9:06 AM JST(11:54 PM - 12:06 AM UTC)

[28-17-am03]Visible-light-induced proximity labeling based on genetically encoded fluorescent proteins

○Zhengyi Liu1, Takahiro Kuchimaru2, Tetsuya Kadonosono3, Shinichi Sato1 (1. Frontier Research Institute of Interdisciplinary Sciences, Tohoku Univ., 2. Center for Molecular Medicine, Jichi Medical Univ., 3. School of Life Science and Technology, Institute of Science Tokyo)
9:06 AM - 9:18 AM JST(12:06 AM - 12:18 AM UTC)

[28-17-am04S]Development of a novel covalent inhibitor for glutaminase 1 with lysine-targeted warhead

○Xiwen Xiao1, Hibiki Okuno1, Saki Inoue1, Shohei Uchinomiya1, Akio Ojida1 (1. Grad. Sch. Pharm. Sci., Kyushu Univ.)
9:18 AM - 9:23 AM JST(12:18 AM - 12:23 AM UTC)

Break

9:23 AM - 9:35 AM JST(12:23 AM - 12:35 AM UTC)

[28-17-am05S]Development of multi-kinase inhibitors using spatiotemporaly-controlled lysine warheads

○Yudai Tanaka1, Atsuya Tanigawa1, Ryo Tetsukawa1, Naoki Zenmyo1, Naoya Shindo1, Akio Ojida1 (1. Grad. Sch. Pharm. Sci., Kyushu Univ.)
9:35 AM - 9:47 AM JST(12:35 AM - 12:47 AM UTC)

[28-17-am06S]Development of covalent KRAS G12D inhibitors using lysine reactive chemistry

○Ryo Tetsukawa1, Yudai Tanaka1, Atsuya Tanigawa1, Naoki Zenmyo1, Naoya Shindo1, Akio Ojida1 (1. Grad. Sch. Pharm. Sci., Kyushu Univ.)
9:47 AM - 9:59 AM JST(12:47 AM - 12:59 AM UTC)

[28-17-am07S]Cyclic Thioureas as Novel Lysine-Selective Covalent Warheads

○Xincheng Lin1, Naoya Shindo1, Akio Ojida1 (1. Grad. Sch. Pharm. Sci., Kyushu Univ.)
9:59 AM - 10:11 AM JST(12:59 AM - 1:11 AM UTC)

[28-17-am08]Synthesis and Evaluation of Astatine-211-labeled Fibroblast Activation Protein Inhibitor(FAPI) for Targeted alpha-therapy medicine

○Masayuki Takamatsu1, Atsushi Shimoyama1, Ayaka Aso1, Taketo Toda1, Yuichiro Kadonaga1,2, Yoshifumi Shirakami2,3, Tadashi Watabe2,3, Taku Yoshiya4, Masayoshi Mochizuki4, Kazuhiro Ooe3, Atsushi Toyoshima3, Hiromitsu Haba5, Yang Wang5, Jens Cardinale6, Frederik Lars Giesel6, Kazuko Nakashima Kaneda1,3, Koichi Fukase1,3 (1. Grad. Sch. Sci., Osaka Univ., 2. Grad. Sch. Med., Osaka Univ., 3. IRS, Osaka Univ., 4. Peptide Institute, Inc., 5. RIKEN, 6. University Hospital Düsseldorf)
Back to Category List