Session Details
[28-18-am]Drug Seeds, Screening 2
Fri. Mar 28, 2025 8:30 AM - 10:11 AM JST
Fri. Mar 28, 2025 11:30 PM - 1:11 AM UTC
Fri. Mar 28, 2025 11:30 PM - 1:11 AM UTC
Room 18 (MARINE MESSE FUKUOKA Hall B: Conference Room2-2 [2F])
Chair: Tadashi Shimizu, Takuya Kobayakawa
[28-18-am01S]Exploration and Synthesis of Drug Candidate Compounds Using Machine Learning
○Takaya Matsumura1, Hiroto Otsuka2, Hiroyuki Morimoto3, Yuri Katou1, Kaori Ota4, Shunsuke Tanaka4, Makoto Furutachi4, Eiji Kawanishi1, Francesca Grisoni5, Motohiro Nishida1, Tomoyuki Miyao6, Takashi Oshima1 (1. Grad. Sch. Pharm. Sci., Kyushu Univ., 2. Fac. Pharm. Sci. Kyushu Univ., 3. Grad. Sch. Eng. Kyutech., 4. Fac. Pharm. Sci. Fukuoka Univ., 5. TU/e, 6. NAIST)
[28-18-am02S]Development of a Massive Fluorogenic Probe Library Based on Bayesian Optimization toward the Discovery of Novel Biomarker Enzymes
○Daiki Ishimoto1, Ryo Tachibana1, Yasuteru Urano1,2 (1. Grad. Sch. Pharm. Sci., Univ. Tokyo, 2. Grad. Sch. Med, Univ. Tokyo)
[28-18-am03S]Construction of a PROTAC library using click chemistry and direct screening to identify HDAC PROTACs.
○Mirei Hayashi1, Yukihiro Itoh1, Yasunobu Yamashita1, Yuri Takada1, Takayoshi Suzuki1 (1. SANKEN, Osaka Univ.)
[28-18-am04S]Recording by Synthesis for enhancement of chemical space, structural diversity, and quality in DNA-Encoded Library
○Masumi Shirakawa1, Ryosuke Ueki1, Jumpei Morimoto1, Shinsuke Sando1 (1. Grad. Sch. Eng. The Univ. of Tokyo)
Break
[28-18-am05S]Identification of small molecules that inhibit SARS-CoV-2 infection by targeting RBD
○Suzuka Makita1, Kaito Koyama1, Katsumi Ohta2, Taiki Ichida2, Ryota Fukai2, Yasushi Takebayashi2,3, Hisashi Murakami1,2, Naohisa Ogo1,2, Akira Asai1,2 (1. Sch. Pharm. Sci., Univ. Shizuoka, 2. Grad. Div. Pharm. Sci., Univ. Shizuoka, 3. Nippon Light Metal Company, Ltd.)
[28-18-am06S]Compound screening for discovering existing drugs selectively targeting CSC-like cells
○Shoki Fujita1, Siori Yanai2, Kao Suzuki1, Satoko Otsuguro1, Yusuke Ohta2, Takao Nomura2, Katsumi Maenaka2,3 (1. Undergrad. Sch. Pharm. Sci., Hokkaido Univ., 2. Grad. Sch. Pharm. Sci., Hokkaido Univ., 3. Grad. Sch. Pharm. Sci., Kyusyu Univ.)
[28-18-am07S]Searching for antimicrobial agents against latent MAC bacteria from microbial resources.
○Yosuke Kamioka1, Satoru Shigeno1, Satoshi Ote1, Hiroshi Tomoda1, Taichi Ohshiro1 (1. Grad. Sch. Pharm. Sci., Kitasato Univ.)
[28-18-am08S]Screening for anti-fatty liver disease compounds from Kitasato Natural Compound Library
○Haruka Murai1, Keisuke Kobayashi1, Taichi Ohshiro1 (1. Grad. Sch. Pharm. Sci., Kitasato Univ.)