Session Details
[28-18-am]Drug Design 2
Fri. Mar 28, 2025 10:20 AM - 11:44 AM JST
Fri. Mar 28, 2025 1:20 AM - 2:44 AM UTC
Fri. Mar 28, 2025 1:20 AM - 2:44 AM UTC
Room 18 (MARINE MESSE FUKUOKA Hall B: Conference Room2-2 [2F])
Chair: Kohei Tsuji, Shinsuke Inuki
[28-18-am09S]Omics-based drug design using generative artificial intelligence
○Yuki Matsukiyo1,2, Yuko Sakajiri2, Kaho Yamabe3, Saki Oshima3, Chika Tohzawa4, Tomokazu Shibata1, Ryusuke Sawada5, Takuya Okada3,4, Hisashi Mori6, Naoki Toyooka3,4, Yoshihiro Yamanishi2 (1. Grad. Sch. of Comp. Sci. and Sys. Eng., Kyushu Inst. of Tech., 2. Grad. Sch. of Inf., Nagoya Univ., 3. Grad. Sch. of Pharm.-Med. Sci., Univ. of Toyama, 4. Fac. of Eng., Univ. of Toyama, 5. Grad. Sch. of Med., Dent. and Pharm. Sci., Okayama Univ., 6. Fac. of Med., Univ. of Toyama)
[28-18-am10S]Development of novel STING antagonists
○Hitomi Terauchi1,2, Taiyo Toita3, Genichiro Tsuji2, Syoichi Ishida3, Toru Ekimoto3, Kei Terayama3, Yosuke Demizu1,2,3 (1. Grad. Sch. Med., Dent. and Pharm. Sci., Okayama Univ, 2. NIHS, 3. Grad. Sch. Med. Life. Sci., Yokohama City Univ.)
[28-18-am11S]Development of Spirocyclopropane-Based Peptidomimetics Targeting α-Helix Hot Spots
○Yuki Yamazaki1, Ryotaro Sakashita1, Tomoki Kuwahara1, Masanori Nagatomo1, Koh Takeuchi2, Satoshi Shuto1, Mizuki Watanabe1 (1. Facul. Pharma. Sci., Hokkaido Univ., 2. Grad. Sch. Pharm. Sci., Tokyo Univ.)
[28-18-am12S]Development of octaarginine-linked CDP-ribitol derivative for substrate supplementation therapy
○Kyosuke Ohira1, Atsuhiko Taniguchi1,2, Rina Kobayashi1, Kei Mukaiyama1, Yui Furuya1, Kazuki Oka1, Sho Konno1,2, Akihiro Taguchi1,2, Hiroshi Manya3, Tamao Endo3, Motoi Kanagawa4, Yoshio Hayashi2,5 (1. Sch. Pharm., Tokyo Univ. Pharm. Life Sci., 2. Grad. Sch. Pharm., Tokyo Univ. Pharm. Life Sci., 3. Tokyo Metro. Inst. Gerontol., 4. Grad. Sch.Med., Ehime Univ., 5. Sch. Life Sci., Tokyo Univ. Pharm. Life Sci.)
[28-18-am13S]Intracellular Nrf2 activation effect of naphthalene-2-acetamide derivatives bearing azetidine skeleton
○Sayuri Inoue1, Saki Yamauchi1, Daisuke Inoue1, Daisuke Yasuda1, Tomoyuki Ohe2, Tomoya Hirano1 (1. Fac. Pharm, Osaka Medcial and Phamaceutical Univ., 2. Fac. Pharm, Keio Univ.)
[28-18-am14S]Identification of small molecules that bind to heterochromatin protein 1 (HP1)
○Akari Tokuyama1, Yasunobu Yamashita1, Ryo Maeda2, Yuri Takada1, Yukihiro Itoh1, Makoto Tachibana2, Takayoshi Suzuki1 (1. SANKEN, Osaka Univ., 2. FBS, Osaka Univ.)
[28-18-am15S]Search and optimization of antimalarial seeds derived from fungi
○Taichi Okano1, So-ichiro Kimura1, Hiroki Nakahara1, Shuji Yoshioka1, Yoshihiro Watanabe1,2, Goh Sennari1,2, Mizuki Hashimoto3, Hiroki Kojima1,2, Kenichi Nonaka4, Akihiro Sugawara1,2, Yuki Inahashi1,2, Takahiro Ishii5, Toshiaki Teruya6, Aki Ishiyama1,2, Rei Hokari1,2, Tomoyasu Hirose1,2, Toshiaki Sunazuka1,2, Masato Iwatsuki1,2 (1. Grad. Sch. Infection Control Sci., Kitasato Univ., 2. Ōmura Satoshi Memorial Inst., Kitasato Univ., 3. Sch. Sci., Kitasato Univ., 4. Fac. Life & Environ. Sci., Teikyo Univ. Sci., 5. Fac. Agric., Univ. Ryukyus, 6. Fac. Edu., Univ. Ryukyus)