Presentation Information

[[A]A404-3am-01]Improving allosteric ligands for in vivo chemogenetic regulation of metabotropic glutamate receptor subtype 1 (mGlu1)

○Keigo Morikawa1, Tomohiro Doura2, Takumi Kondo2, Tomoteru Yamasaki3, Masayuki Fujinaga3, Ming-Rong Zhang3, Wataru Kakegawa4, Shigeki Kiyonaka2,5 (1. Scool of Engineering, Nagoya University, 2. Graduate scool of engineering, Nagoya University, 3. National Institutes for Quantum Science and Technology, 4. Keio University School of Medicine, 5. Research Institute for Quantum and Chemical Innovation, Institutes of Innovation for Future Society, Nagoya University)

Keywords:

Chemogenetics,Pharmacokinetics,G protein-coupled receptor,cell type-specific control,metabotropic glutamate receptor subtype 1