Session Details

[[A]A404-3am]16. Natural Products Chemistry, Chemical Biology

Fri. Mar 28, 2025 9:00 AM - 11:10 AM JST
Fri. Mar 28, 2025 12:00 AM - 2:10 AM UTC
[A]A404(A404, Bldg. 1, Area 3 [4F])

[[A]A404-3am-01]Improving allosteric ligands for in vivo chemogenetic regulation of metabotropic glutamate receptor subtype 1 (mGlu1)

○Keigo Morikawa1, Tomohiro Doura2, Takumi Kondo2, Tomoteru Yamasaki3, Masayuki Fujinaga3, Ming-Rong Zhang3, Wataru Kakegawa4, Shigeki Kiyonaka2,5 (1. Scool of Engineering, Nagoya University, 2. Graduate scool of engineering, Nagoya University, 3. National Institutes for Quantum Science and Technology, 4. Keio University School of Medicine, 5. Research Institute for Quantum and Chemical Innovation, Institutes of Innovation for Future Society, Nagoya University)

[[A]A404-3am-02]Strategy to increase the affinity of inhibitors to engineered adenosine A2A receptors for chemogenetic control

○Shinichi Oki1, Yuma Matsuoka2, Tomohiro Doura2, Shigeki Kiyonaka3 (1. School of Engineering, Nagoya University, 2. Graduate School of Engineering, Nagoya University, 3. Research Institute for Quantum and Chemical Innovation, Institute of Innovation for Future Society, Nagoya University)

[[A]A404-3am-03]Investigation of the binding mode of stylissatin A on lysosomal PPCA and development of its analogs for anti-obesity agents

○Dewi Luthfiana1, Yiting Sun1, Ayumi Dakiiwa1, Takahiro Shibata1, Masaki Kita1 (1. Nagoya University)

[[A]A404-3am-04]Small Molecule-Mediated Paralytic Effect on Movement Regulation in Symbiotic Dinoflagellates

○Carlos Augusto Loayza-Cassano1, Hiroshi Yamashita 2, Yuta Tsunematsu1, Masaki Kita1 (1. Graduate School of Bioagricultural Sciences, Nagoya University, 2. Fisheries Technology Institute, Japan Fisheries Research and Education Agency)

[[A]A404-3am-05]Synthesis of Nanographenes with Ca2+ Triggered “Turn-On” Blinking Properties toward Super-Resolution Biosensing

○Zhiqiang Gao1, Hao Zhao1, Akimitsu Narita1 (1. Okinawa Institute of Science and Technology)

[[A]A404-3am-06]Self-Blinking Nanographene with Cationic Side Chains for Super-Resolution Bioimaging of Live-Cell Membrane

○Hao Zhao1, Xingfu Zhu2, Xiaomin Liu2, Mischa Bonn2, Akimitsu Narita1,2 (1. Okinawa Institute of Science and Technology Graduate University, 2. Max Planck Institute for Polymer Research)

Break

[[A]A404-3am-07]Tetrazine-based fluorogenic probe toward leaflet-selective polarity imaging of cell membranes

○Yusei Otsuka1, Tomoya Yamamoto1,2, Kazuya Kikuchi1,2 (1. Graduate School of Engineering, Osaka University, 2. Immunology Frontier Research Center, Osaka University)

[[A]A404-3am-08]Development of Fluorogenic Probes for Monitoring Protein-protein Interactions with Reversible Labeling Strategy

○Jiatong Li1, Masafumi Minoshima1, Kazuya Kikuchi1,2 (1. Graduate School of Engineering, Osaka University, 2. Immunology Frontier Research Center, Osaka University)

[[A]A404-3am-09]Development of Red-fluorescent Probe for Reversible Protein Labeling

○Nana Otani1, Masafumi Minoshima1, Kazuya Kikuchi1,2 (1. Graduate School of Engineering, Osaka Univ, 2. Immunology Frontier Research Center, Osaka Univ)

[[A]A404-3am-10]Development of a novel Raman probe for glutathione

○Yuta Murao1, Hiroyoshi Fujioka1, Minoru Kawatani1, Spencer John Spratt2, Kazuhiro Kuruma2, Yasuyuki Ozeki2, Mako Kamiya1,3 (1. Department of Life Science and Technology, Institute of Science Tokyo, 2. Research Center for Advanced Science and Technology, The University of Tokyo, 3. Research Center for Autonomous Systems Materialogy (ASMat), Institute of Science Tokyo)

[[A]A404-3am-11]Development of photo-switchable Raman probe with simultaneous detection

○SATOSHI MATSUMOTO1, Hiroyoshi Fujioka1, Minoru Kawatani1, Hikaru Akaboshi2, Spencer John Spratt2, Kazuhiro Kuruma2, Yasuyuki Ozeki2, Mako Kamiya1,3 (1. Institute of Science Tokyo Department of Life Science and Technology, 2. The Univ. of Tokyo Research Center for Advanced Science and Technology, 3. Research Center for Autonomous Systems Materialogy)

[[A]A404-3am-12]Synthesis and functional elucidation of fatty acid glyceride derivatives with cytoprotective activity

○Yuki Utsugi1, Leo Kwon1, Yuki Sakata1, Kenji Matsuno2, Osamu Ohno1 (1. Kogakuin Univ., 2. Yasuda Women’s Univ.)