Session Details
[27P-pm]Organic Chemistry 2
Thu. Mar 27, 2025 1:30 PM - 5:00 PM JST
Thu. Mar 27, 2025 4:30 AM - 8:00 AM UTC
Thu. Mar 27, 2025 4:30 AM - 8:00 AM UTC
Poster (MARINE MESSE FUKUOKA Hall B: Exhibition Room [1F])
[27P-pm001S]Development of an intramolecular N-N cross-coupling reaction of acridone and carbazole using NaOCl·5H2O
○Junki Sugiyama1, Keisuke Yoshida1, Natsuko Momiyama1, Shinji Kitagaki1 (1. Faculty of Pharmacy, Meijo University)
[27P-pm002S]Synthetic studies of Roehymine
○Ryota Nagao1, Keisuke Yoshida1, Kouki Kameda1, Masaya Kako1, Ryuki Ota1, Shinji Kitagaki1 (1. Faculty of Pharmacy, Meijo University)
[27P-pm003S]Development of oxidative N-N homocoupling reaction of carbazole or acridone using NaOCl·5H2O and application to the total synthesis of Dixiamycin A and B
○Miho Hotta1, Keisuke Yoshida1, Reika Utsugi1, Akari Achiwa1, Shinji Kitagaki1 (1. Faculty of Pharmacy, Meijo University)
[27P-pm004S]Synthetic Studies on Pyridoacridines
○Yuki Nakatani1, Hiromasa Miyoshi2, Risa Kimura1, Hitoshi Takatsu2, Naoyuki Kotoku1,2 (1. Grad. Sch. Pharm. Sci., Ritsumeikan Univ., 2. Coll. Pharm. Sci., Ritsumeikan Univ.)
[27P-pm005S]Studies toward Total Synthesis of Calyciphylline B: Reinvestigation of the BCD Core Construction
Norika Tsuchiya1, ○Kentaro Kako1, Taiki Kurishima1, Yuji Mori1, Takeo Sakai1 (1. Fac. Pharm., Meijo Univ.)
[27P-pm006S]Synthetic studies toward optically active bergamotane sesquiterpenes
○Honoka Takase1, Fumihiro Rokukawa1, Kazuma Matsunaga1, Atsushi Kishida1, Kazuhiko Takatori1 (1. Meiji Pharmaceutical University)
[27P-pm007S]Synthetic studies of antheridiogen–An
○Soichiro Fujiwara1, Satoshi Kaneko1, Kokoro Nagasawa1, Kazuma Matsunaga1, Atsushi Kishida1, Hiroto Nagaoka1, Kazuhiko Takatori1 (1. Meiji Pharmaceutical University)
[27P-pm008S]Synthetic studies of brianthein W
○Kazunori Miyata1, Kyoko Kasai1, Issei Miyamatsu1, Yutaro Numata1, Yuichi Jibiki1, Kazuma Matsunaga1, Atsushi Kishida1, Kazuhiko Takatori1 (1. Meiji Pharmaceutical University)
[27P-pm009]Synthesis of side-chain difluorovitamin D3 with different alkyl length
○FUMIHIRO KAWAGOE1, Hiroya Tabuchi1, Sayuri Mototani2, Kaori Yasuda3, Tomofumi Yatsu2, Toshie Fujishima2, Yoshiki Miyata2, Tsutomu Kimura1, Toshiyuki Sakaki3, Atsushi Kittaka2 (1. Grad. Sch. of Sci., Tokyo Univ. of Sci., 2. Faculty Pharm. Sci., Teikyo Univ., 3. Faculty of Engineering, Toyama Prefectural Univ.)
[27P-pm010S]Highly selective intramolecular O-alkylation of the β-ketoester and synthesis of lilac alcohols
○Ibuki Abe1, Kenichi Harada1, Yuichiro Nakaoka1, Miwa Kubo1, Yoshiyasu Fukuyama1 (1. Pharm. Sci., Tokushima Bunri Univ.)
[27P-pm011]Synthetic Studies on Aberrarone (Part 3)
○Miyuki Ishizaki1, Yukino Hihara1, Miyo Kimoto1, Hiroshi Nakamura1 (1. Fac. Pharm. Sci., Josai International University)
[27P-pm012]Daphnia swimming inhibition effect and anti-water mold activity of dehydroantofine analogs
○Miyuu Mori1, Naoto Yamasaki1, Yoshinori Asakawa1, Hirofumi Yamamoto1 (1. Faculty of pharmaceutical Sciences, Tokushima Bunri Univ.)
[27P-pm013S]Synthetic study of Heptelidic acid
○Ai Takeuchi1, Kazuki Yamamoto2, Satoshi Ichikawa2 (1. Pharm. Sci., Hokkaido Univ., 2. Grad. Sch. Pharm. Sci., Hokkaido Univ.)
[27P-pm014S]Synthesis and cytotoxicity evaluation of cadinene-type compounds
○Fumi Oyatsu1, Ryohei Saito-Moriya1, Akihito Yokosuka2, Yoshihiro Mimaki2, Hideki Abe1 (1. Fac. Sci., Japan Women’s Univ., 2. Sch. Pharm., Tokyo Univ. Pharm. Life Sci.)
[27P-pm015]Syntheses and biological activity evaluation of tricyclic natural products and their analogues
○Nanako Inaba1, Mayu Nomura1, Yuta Ogura2, Ryohei Saito-Moriya1, Yuichiro Kawamoto2, Toyoharu Kobayashi2, Akihito Yokosuka3, Yoshihiro Mimaki3, Hisanaka Ito2, Hideki Abe1 (1. Fac. Sci., Japan Women's Univ., 2. Sch. Life Sci., Tokyo Univ. Pharm. Life Sci., 3. Sch. Pharm., Tokyo Univ. Pharm. Life Sci.)
[27P-pm016S]Synthetic Studies of CD Ring Derivatives of Andrastins with FTase Inhibitory Activity
○Fumino Kitamura1, Ayano Kosaka1, Masaru Tanioka1, Tsuyoshi Yamada1, Yuji Matsuya1 (1. Faculty of Pharm. Sci., University of Toyama)
[27P-pm017]Structural “differentiation” of vitamin D and characterization of its novel 19-homo analogues.
○Toshie Fujishima1,2, Atsuki Wada2, Masayuki Morikawa2, Kasumi Une2 (1. Faculty of Pharmaceutical Sciences, Teikyo University, 2. Faculty of Pharmaceutical Sciences at Kagawa Campus, Tokushima Bunri University)
[27P-pm018]Peptide Synthesis by Fragment Condensation Reaction Utilizing Silylating Reagent
○Kotaro Ishihara1, Tomohiro Hattori1, Hisashi Yamamoto1 (1. Peptide Research Center, Chubu Univ.)
[27P-pm019S]Development of late-stage modification synthesis of α-amino phosphate-containing peptides by addition of indole to N-Nps-imino phosphonamide
○Ayaka Mitsuyasu1, Takuya Sakakibara1, Tsubasa Inokuma1, Ken-ichi Yamada1 (1. Grad. Sch. Pharm. Sci., Tokushima Univ.)
[27P-pm020S]Total Synthesis of Amatyemides A and B
○Wakana Osaka1, Rikito Suzuki1,2, George F Neuhaus3, Xinhui Yu3, Kerry L McPhail3, Shinya Oishi1,2 (1. Kyoto Pharm. Univ., 2. Grad. Sch. Pharm. Sci., Kyoto Univ., 3. Oregon State Univ.)
[27P-pm021]Suppression of the diketopiperazine (DKP) by-products in N-methylated peptide synthesis: Efficacy of fluorous silyl protecting group
Kotaro Ishihara1, ○Shoma Naganuma1, Yuna Hagiwara1, Yu Mochizuki2, Yamato Kato1, Akihiro Nagaya3, Takayuki Nagatsuka3, Takayuki Shioiri1,2, Masato Matsugi1,2 (1. Grad. Sch. Agric., Meijo Univ., 2. Fac. Agric., Meijo Univ., 3. Nissan Chemical Corp.)
[27P-pm022S]Development of a Method for Simultaneous Synthesis of Both Epimers of α-Indolylglycine-Containing Peptide
○Rui Shiozawa1, Kana Masui1, Tsubasa Inokuma1, Ken-ichi Yamada1 (1. Gras. Sch. Pharm. Sci., Tokushima Univ.)
[27P-pm023]Three-component azepine synthesis by gold/magnesium orthogonal relay catalysis
○Kenji Sugimoto1,2, Shuto Kosuge2, Yoshihiro Kiraku2, Kiyoshi Tsuge3, Yuji Matsuya2 (1. Grad. Sch. Life and Environmental Sci., Kyoto Pref. Univ., 2. Faculty of Pharm. Sci., Univ. of Toyama, 3. Faculty of Sci., Univ. of Toyama)
[27P-pm024S]Asymmetric hydrolysis of tropic acid β-lactone with new cincona alkaloid-derived chiral phase-transfer catalysts
Midori Kawasaki1, ○Rio Maruyama2, Nagisa Aono2, Takahiro Shirai3, Kenji Yatsuzuka2, Ryuichi Shirai1 (1. Grad. Sch. Pharm. Sci., Doshisha Women's Col., 2. Fac. Pharm. Sci., Doshisha Women's Col., 3. Grad. Sch. Biomed. Health Sci., Hiroshima Univ.)
[27P-pm025]Photoinduced electron transfer-directed alkylation of ynamides
Yousuke Yamaoka1,2, Daigo Kajiwara2, Hikaru Saito2, ○Takuma Tsujimoto1, Kiyosei Takasu2, Hideto Miyabe1 (1. Sch. of Pharm. Hyogo Med. Univ. , 2. Grad. Sch. Pharm. Sci. Kyoto Univ.)
[27P-pm026S]Photodegradation of pharmaceuticals using vitamin B2 as a photosensitizer
○Noa Ito1, Yuka Kimura1, Mayuko Suga1, Kayo Nakamura1, Hidetsugu Tabata2, Tetsuta Oshitari2, Hideaki Natsugari3, Hideyo Takahashi1 (1. Pharm. Sci., Tokyo Univ. Sci., 2. Pharm. Sci., Teikyo Univ., 3. Pharm. Sci., Tokyo Univ.)
[27P-pm027]Construction of piperidine ring and formal synthesis of Julifloridine using hypervalent iodine and diphenyl diselenide
○Yoshihiro Natori1, Hideaki Wakamatsu1, Yukako Saito1, Asako Kaise1, Kentaro Yamaguchi2, Tadashi Hyodo2, Yuichi Yoshimura1 (1. Faculty of Pharmaceutical Sciences, Tohoku Medical and Pharmaceutical University, 2. Faculty of Pharmaceutical Sciences at Kagawa Campus, Tokushima Bunri University)
[27P-pm028]Development of a 1,3,5-triazine skeleton formation via ring cleavage of 2-alkynyl-3-hydroxyisoindolin-1-one
○Noriko Okamoto1, Takuya Sueda1 (1. Faculty of Pharmaceutical Sciences, Hiroshima International University)
[27P-pm029S]Regioselective Hydroacylation of 3-Azacyclohexyne
○Kentaro Kagami1, Nanako Ishibashi1, Ayane Kayano1, Masanori Tayu1, Sayaka Ohrui1, Nozomi Saito1 (1. Meiji Pharm. Univ.)
[27P-pm030]Development of N-difluoroiodomethylation of imidazoles using trifluoroiodomethane
○Ryuichi Nishiyori1, Munenori Inoue1 (1. SCRI)
[27P-pm031S]Development of chiral DMAP type catalyst and application to reactions
○Yuria Kato1, Tomoki Mukai1, Taiki Asai1, Shinya Kimura1, Masamichi Yamanaka1, Masashi Yokoya1 (1. Meiji Pharm. Univ.)
[27P-pm032S]Diastereoselective synthesis of fused cyclic amines bearing consecutive tetrasubstituted carbons by a cascade reaction
Kaito Totsuka1, ○Haruka Katayama1, Ayame Taki1, Yuji Mori1, Takeo Sakai1 (1. Fac. Pharm., Meijo Univ.)
[27P-pm033S]Study on the N-alkylation of amines with primary benzyl cationoids
○Ayato Kataoka1, Kazuyuki Kosha2, Kazuhito Hioki1, Keiko Hojo1, Hikaru Fujita2, Munetaka Kunishima1,2 (1. Kobe Gakuin Univ., 2. Kanazawa Univ.)
[27P-pm034S]Boronic acid-catalyzed peptide bond formation utilizing amino acid-derived inert esters
○Airi Takahashi1, Naoya Takahashi2, Naoyuki Shimada1 (1. Department of Chemistry, Nihon Univ., 2. Department of Pharmaceutical Sciences, Kitasato Univ.)
[27P-pm035S]Synthesis of trans-fused carbocycles by the three-component coupling/6-endo cyclization sequence: improvement and application
○Mari Ando1, Eisaku Ohashi2, Ryuji Ando2, Ryuki Kawaguchi1, Seiichi Nakamura2 (1. Fac. Pharm. Sci., Nagoya City Univ., 2. Grad. Sch. Pharm. Sci., Nagoya City Univ.)
[27P-pm036S]Boronic acid/palladium hybrid catalysis for regio- and stereo-selective glycosylation of carbohydrates
○Atsunari Kanda1, Kazuma Irisawa1, Makoto Wakatsuki2, Naoyuki Shimada1 (1. Department of Chemistry, Nihon Univ., 2. Department of Pharmaceutical Sciences, Kitasato Univ.)
[27P-pm037S]Boronic acid-catalyzed regioselective propargylation of carbohydrates
○Kai Nitanda1, Daichi Sato2, Naoyuki Shimada1 (1. Department of Chemistry, Nihon Univ., 2. Department of Pharmaceutical Sciences, Kitasato Univ.)
[27P-pm038S]Development of a one-pot reaction for the sequential acylation of α-D-glucose to the 6- and 2-positions.
○Rui Ishikawa1, Kazuki Usuguchi1, Akira Takagi1, Kensuke Okuda1 (1. Kobe Pharm. Univ.)
[27P-pm039]Synthesis of diverse heterocycles based on MHAT/RPC mechanism
○hiroki shigehisa1, Takuma Sugimura1, Ren Yamada2, Wataru Kanna2, Tsuyoshi Mita3,4, Satoshi Maeda2,3,4, Szarłan Bartłomiej5 (1. Musashino Univ., 2. Fac. of Sci., Hokkaido Univ., 3. WPI-ICReDD, Hokkaido Univ., 4. JST-ERATO, 5. Adam Mickiewicz Univ. in Poznań)
[27P-pm040S]Ring-closing disulfenylation of alkenoic thioester
○Kanaru Sasaki1, Miari Kurihara1, Hiroki Shigehisa1 (1. Musashino Univ.)
[27P-pm041S]Development of highly active 2-pyridone catalysts for ester aminolysis and their mechanistic elucidation
Takeshi Yamada1, ○Mahiro Tamura1, Nanako Tsuji1, Marin Gogami2, Takeshi Yoshikawa2, Ken Sakata2, Manabu Hatano1 (1. Fac. Pharm. Sci. Kobe Pharmaceutical Univ., 2. Fac. Pharm. Sci. Toho Univ.)
[27P-pm042S]Solution phase peptide synthesis using phenol-derived hydrophobic soluble tag
Takeshi Yamada1, ○Waka Oda1, Mioko Nasu1, Manaka Fujita1, Manabu Hatano1 (1. Kobe Pharmaceutical Univ.)
[27P-pm043S]Concise synthesis of polyacyloxy cyclic ethers from polyols and carboxylic acids using sulfonic acid catalyst
Takeshi Yamada1, ○Mike Matsuda1, Anri Kimura1, Saya Takenouchi1, Mizuki Sugahara1, Mai Yoshioka1, Yuhei Monta1, Manabu Hatano1 (1. Kobe Pharmaceutical Univ.)
[27P-pm044S]Synthesis of 2-fluorodienes by Lewis acid-mediated Suzuki-Miyaura Cross-Coupling
○Runa Nakamura1, Takashi Niwa2 (1. Sch. Pharm. Sci., Kyushu Univ., 2. Grad. Sch. Pharm. Sci., Kyushu Univ.)
[27P-pm045S]Preparation of optically active paraconyl alcohol through consecutive acyl substitution
○Airi Kokawa1, Yuuna Nishioka1, Kei Kitamura1, Hiroto Kaku1 (1. Fac. Pharm. Sci., Tokushima Bunri Univ.)
[27P-pm046S]Gold-catalyzed synthesis of cyclobutanes in ionic liquid
○Naho Ishii1, Hitomi Chiaki1, Miyu Yamashita1, Yoshimitsu Hashimoto1, Osamu Tamura1, Nobuyoshi Morita1 (1. Showa Pharm. Univ.)
[27P-pm047S]Palladium-Catalyzed α-Arylation of Ketones mediated by Lewis acid
○Ryo Kajiyama1, Takashi Niwa2 (1. Sch. Pharm. Sci., Kyushu Univ., 2. Grad. Sch. Pharm. Sci., Kyushu Univ.)
[27P-pm048S]Structural diversification strategy of cyclic hydrosilanes leading to synthesis of novel silicon-containing compounds
○Ryusei Kitagawa1, Hiroki Matsui1, Akira Matsumoto1, Chao Wang1, Keiichi Hirano1 (1. Grad. Sch. Pharm. Sci., Kanazawa Univ.)
[27P-pm049S]Development of chloroalkylation of carboxylic acids using bromochloromethane
Junpei Matsuoka1, ○Haato Tsuda1, Natsumi Kuraoka 1, Yao Hiroki1, Tomohiro Maegawa1 (1. School of Pharmaceutical Sciences, Kindai University)
[27P-pm050]Mechanistic studies on a palladium-catalyzed α-alkylation of ketones
○Yasunari Monguchi1, Taisei Sakai1, Yuki Yoshino1, Kotaro Yamashita1, Miku Takamaru1, Kazutaka Koga1, Sayuri Yokoyama1 (1. Daiichi University of Pharmacy)
[27P-pm051S]γ-Selective Substitution of 1,3-Diketones and Synthesis of Unsymmetrical Curcumin Derivatives
○Rina Tanaka1, Kyosuke Sugihara1, Arata Kumazaki2, Hitoshi Abe1 (1. Grad. Sch. Sci. and Eng., Toyama Univ., 2. Fac. Eng., Toyama Univ.)
[27P-pm052]Continuous flow synthesis of cyclobutenes via lithium ynolates
○aki kohyama1, motoki namioka1, hiroshi takikawa1, yousuke yamaoka2, kiyosei takasu1 (1. Grad. Sch. Pharm. Sci., Kyoto Univ., 2. Sch. Pharm., Hyogo Med. Univ.)
[27P-pm053S]Telescoping synthesis of 2-acylindoles from 2-aminochalcones
○Yuto Matsumura1, Takeru Kanazawa1, Kyoko Okamura1, Akira Nakamura1, Junpei Matsuoka1, Tomohiro Maegawa1 (1. School of Pharmaceutical Sciences, Kindai University)
[27P-pm054S]Development of new PMB-Type protecting groups focusing on the o-substituent effect
Junpei Matsuoka1, ○Tatsuya Katagiri1, Seiya Higashioka1, Tomohiro Maegawa1 (1. School of Pharmaceutical Sciences, Kindai University)
[27P-pm055S]Sulfur compounds-mediated halogenation of electron-deficient aromatic compounds
Junpei Matsuoka1, ○Riko Okaguchi1, Yuna Yano1, Tomohiro Maegawa1 (1. School of Pharmaceutical Sciences, Kindai University)
[27P-pm056S]Crystal structures of N-methyl-N-phenylthiophene carboxamides
○Ruka Ikeda1, Ai Ito1, Hirokazu Karasawa1, Midori Hakuno1, Ryu Yamasaki1, Iwao Okamoto1 (1. Showa Pharm. Univ.)
[27P-pm057S]Synthesis and structural properties of N-vinylamide bearing fluorine aromatics
○Hiroto Koide1, Ryu Yamasaki1, Souichiro Urushiyama1, Ai Ito1, Iwao Okamoto1 (1. Showa Pharm. Univ.)
[27P-pm058S]Crystal structures and conformational preferences of aromatic amides bearing 5-membered aromatic ring
○Mako Endo1, Ai Ito1, Marino Asato1, Yuki Asami1, Ryu Yamasaki1, Iwao Okamoto1 (1. Showa Pharm. Univ.)
[27P-pm059S]Toward the synthesis of oxoazananobelts which have an amide bridged paracyclophane structure
○Haruka Kato1, Hisato Takahashi1, Hyuma Masu2, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ., 2. CAI, Chiba Univ.)
[27P-pm060S]Synthesis and chiroptical properties of chiral tetraphenyladamantane derivatives having four different substituents
○Hikaru Yasukawa1, Sae Maeda1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)
[27P-pm061S]The steric effect of terminal substituents on energy barriers for racemization of an oxoaza[5]helicene
○Hazuki Yasuno1, Ryo Ikeda1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)
[27P-pm062S]Trapacycles: Design and Synthesis of Rhombus-shaped Macrocycles
○Sei Murayama1, Hiroshi Naka1,2 (1. Grad. Sch. of Pharm. Sci., Kyoto Univ., 2. CPiER-DSR, Kyoto Univ.)
[27P-pm063S]Synthesis and optical properties of chiral spherical amides with fluorescent emitting moieties
○Takahiro Yajima1, Daiki Koike1, Hyuma Masu2, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ., 2. CAI, Chiba Univ.)
[27P-pm064S]Synthesis and optical properties of C3-symmetric aromatic spherical amides with two kinds of substituents
○Mikito Shimoda1, Daiki Koike1, Hyuma Masu2, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ., 2. CAI, Chiba Univ.)
[27P-pm065S]Synthesis of cyclic hydroxamic acid derivatives whose structure changes in response to the external environment
○Saki Tanaka1, Sara Tomita1, Hidemasa Hikawa1, Shoko Kikkawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)
[27P-pm066S]Development of fluorescein-based water-compatible NIR-II photoredox catalyst
○Masaya Oyama1, Masaru Tanioka1, Chen Shiyu1, Tsuyoshi Yamada1, Yuji Matsuya1 (1. Faculty of Pharm. Sci., University of Toyama)
[27P-pm067S]Development of packing material method to obtain crystals suitable for single crystal X-ray crystallographic analysis by co-crystallization
○Tomokatsu Enda1, Shoko Kikkawa1, Hidemasa Hikawa1, Isao Azumaya1 (1. Fac. Pharm. Sci., Toho Univ.)
[27P-pm068S]Solvent Trigger: Effortless CO2 Release from Aralkylamines through Retro Neutralizartion
○Narumi Iwamoto1, Hiroto Tanishima2, Risa Otsuka1, Ayaka Uchida1, Ryo Murakami1, Fuyuhiko Inagaki1 (1. Grad.Sch.Pharm.Sci.,Kobegakuin Univ., 2. Grad.Sch. Pharm.Sci.,Kobegakuin Univ.)
[27P-pm069]Development of boron compound analysis method using fluorescrent boron sensor
○Yoshihide Hattori1, Miki Ishimura1, Yoichiro Ohta1, Hiroshi Takenaka1, Mitsunori Kirihata (1. Res. Cen. BNCT, Osaka Metropolitan Univ.)