Session Details
[28-64-pm2]Drug discovery, structure-activity relationship 4
Sat. Mar 28, 2026 3:30 PM - 5:30 PM JST
Sat. Mar 28, 2026 6:30 AM - 8:30 AM UTC
Sat. Mar 28, 2026 6:30 AM - 8:30 AM UTC
Room 64 (Collaboration Commons, RINPUKAN [1F]) (2)
Discusser: Tomoya Hirano, Tsutsumi Tomohiro
[28-64-pm2-28S]Synthesis of acyclic retinoid derivatives and comparison of their activity in Hepatocellular Carcinoma cell lines
○Rina Naito1, Noriyoshi Tanaka1, Xian-Yang Qin2, Naoki Hirokawa1, Kazuma Mizuno1, Ichiro Yajima1, Yoshitomo Suhara1 (1. Grad. Shibaura institute of Technology, 2. RIKEN Center for Integrative Medical Sciences)
[28-64-pm2-29S]Synthesis and Biological Evaluation of Chennat-Type 1,4-Dihydropyridines as SIRT1 Inhibitors
○Rio Furutani1, Kurumi Yamamoto2, Chisato Onozawa2, Kaho Hentona2, Yosinori Okuno2, Shigeki Isomura2, Miho Sawada1, Yukiko Moriyama1, Yukihiro Itoh1,3, Yasuo Sato2, Takayoshi Suzuki1 (1. SANKEN, The University of Osaka, 2. Department of Medicinal Chemistry, Yokohama University of Pharmacy, 3. Laboratory for Biomaterials and Bioengineering, Institute of Integrated Research, Institute of Science Tokyo)
[28-64-pm2-30S]Structure-Activity Relationship Study of Dihydroquinazolinone Derivatives Targeting Nuclear Receptor Nr4a1
○Kosuke Toyoda1, Yoshinori Taguchi2, Hijiri Kishikawa2, Kohei Sato1, Nobuyuki Mase1, Ichiro Takasaki3, Narumi Tetsuo1,2 (1. Grad. Sch. Integ. Sci., Shizuoka Univ., 2. Grad. Sch. Med. Photonics, Shizuoka Univ., 3. Grad. Sch. Pharm. -Med. Sci., Toyama Univ.)
[28-64-pm2-31S]Synthesis of Novel Vitamin K Derivatives with Enhanced Neural Differentiation Induction Activity through Quinone Ring Modifications
○Miho Iwano1, Tatsuya Kaneko1, Yoshitomo Suhara1 (1. Grad. Engineering and Science, Shibaura Institute of Technology)
[28-64-pm2-32S]Structure and properties of oxygen-independently activatable photosensitizers
○Reiko Kyogoku1, Yumika Matsushita1, Kaori Shimoda2, Samina Aslam2, Yoshimasa Tanaka2, Toshihide Maki2 (1. Fac. Pharm. Nagasaki University, 2. Grad. Sch. Biomed. Sci. Nagasaki University)
[28-64-pm2-33S]Development of novel antibacterial lead compounds against nontuberculous mycobacteria based on natural MraY inhibitors
○Miharu Hikosaka1, Kazuki Yamamoto1, Motoko Shinohara2, Yusuke Minato2, Toyotaka Sato3, Motohiro Horiuchi3, Satoshi Ichikawa1 (1. Grad. Sch. Pharm. Sci., Hokkaido Univ., 2. Center for Infectious Disease Research., Fujita Health Univ.,, 3. Grad. Sch. Vet. Med., Hokkaido Univ.)
[28-64-pm2-34S]Synthesis and Evaluation of Sulfonamide-Containing ortho-Naphthoquinones as STAT3 Inhibitors
○Masaki Kawabata1, Mitsuaki Yamashita1, Yoichi Fukuda1, Akira Iida1 (1. Grad. Sch. Agri., Kindai Univ.)
[28-64-pm2-35S]Synthesis and Structure-Activity Relationship Studies of Antitumor Furanonaphthoquinones with STAT3 Inhibitory Activity
○Shosei Yabushita1, Mitsuaki Yamashita1, Akira Iida1 (1. Grad. Sch. Agri Sci., Kindai Univ.)
[28-64-pm2-36S]Optimized Ultrasound-Assisted Extraction and Bioactive Profile of Mitragyna speciosa Leaves for Cosmeceutical Applications
○Thasang Thavanapong1, Worrapan Poomanee1, Pimporn Leelapornpisid1, Mathukorn Sainakham1, Nathupakorn Dechsupa2, Siripat Chaichit1, Nara Yaowiwat3 (1. Pharm. Sci., Chiang Mai Univ., 2. Radio. Tech., Chiang Mai Univ., 3. Cos. Sci., Mae Fah Luang Univ.)
