Session Details

[S15☆]Development of New Warhead-Construction Reactions for Enhanced DNA-Encoded Library (DEL) Synthesis and Their Application to DEL Production

Fri. Mar 27, 2026 1:10 PM - 3:10 PM JST
Fri. Mar 27, 2026 4:10 AM - 6:10 AM UTC
Room 17 (A201)
Organizer: Hiroyuki Miyachi (Drug Discovery Initiative, Grad. Sch. Pharm. Sci., Univ. of Tokyo), Motomu Kanai (Grad. Sch. Pharm. Sci., Univ. of Tokyo)

オーガナイザー趣旨説明
宮地 弘幸(東大院薬 創薬機構)

[S15-1]Research on the construction of warhead-DEL with low-molecular-weight compounds

○Takashi Osawa1 (1. Grad. Sch. Pharm. Sci., Osaka Univ.)

[S15-2]Construction of DEL with a natural product mimetic macrocycle as war head

○Teigo Asai1 (1. Grad. Sch. Pharm. Sci., Tohoku Univ.)

[S15-3]Synthesis of DNA encoded library with biologically active scaffold derived from amino acid.

○Katarzyna Joanna Malawska1, Masashi Suzuki2, Junko Sasaki2, Masaki Koshimizu2, Kazuma Kaitoh3, Hiroyuki Miyachi2, Motomu Kanai1 (1. Grad. Sch. Pharm. Sci., Univ. of Tokyo, 2. Drug Discovery Initiative, Grad. Sch. Pharm. Sci., Univ. of Tokyo, 3. Cat. Chem. Res. Inst., AIST)

[S15-4]Practical DEL synthesis through industry–academia collaboration: Insights from the field

○Masashi Suzuki1 (1. Drug Discovery Initiative, Grad. Sch. Pharm. Sci., Univ. of Tokyo)

総括
金井 求(東大院薬)